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Angiogenesis
Subcategories of "Angiogenesis"
Show 8 more subcategories
Products of "Angiogenesis"
Regorafenib
CAS:755037-03-7
Formula:
C21H15ClF4N4O3
Purity:
>98.0%(HPLC)
Color and Shape:
White to Light yellow to Light orange powder to crystal
Molecular weight:
482.82
Estimated delivery in United States, on Tuesday 25 Jan 2022
2-Methoxy--estradiol
CAS:362-07-2
Formula:
C19H26O3
Purity:
>97.0%(GC)
Color and Shape:
White to Light yellow powder to crystal
Molecular weight:
302.41
Estimated delivery in United States, on Tuesday 25 Jan 2022
SKLB1002
CAS:1225451-84-2
Formula:
C13H12N4O2S2
Purity:
>98.0%(HPLC)
Color and Shape:
White to Light yellow powder to crystal
Molecular weight:
320.39
Estimated delivery in United States, on Tuesday 25 Jan 2022
(±)-Thalidomide
CAS:50-35-1
Formula:
C13H10N2O4
Purity:
>98.0%(HPLC)(N)
Color and Shape:
White to Almost white powder to crystal
Molecular weight:
258.23
Estimated delivery in United States, on Tuesday 25 Jan 2022
Gefitinib
CAS:184475-35-2
Formula:
C22H24ClFN4O3
Purity:
>98.0%(T)(HPLC)
Color and Shape:
White to Light yellow powder to crystal
Molecular weight:
446.91
Estimated delivery in United States, on Tuesday 25 Jan 2022
Genipin
CAS:6902-77-8
Formula:
C11H14O5
Purity:
>97.0%(GC)
Color and Shape:
White to Almost white powder to crystal
Molecular weight:
226.23
Estimated delivery in United States, on Tuesday 25 Jan 2022
Bestatin, Ubenimex
CAS:58970-76-6
Bestatin (or ubenimex), an antibiotic of natural origin, is a specific, competitive inhibitor of many …
Formula:
C16H24N2O4
Purity:
99.5%
Color and Shape:
White Powder
Molecular weight:
308.17361
Estimated delivery in United States, on Tuesday 25 Jan 2022
Stem Cell Proliferation Inhibitor, AcSDKP, Goralatide, Thymosin b4 (1-4)
CAS:120081-14-3
The bioactive tetrapeptide goralatide which corresponds to the N-terminus of Thymosin b4, is a physiological …
Formula:
C20H33N5O9
Purity:
98.7%
Color and Shape:
White
Molecular weight:
487.22783
Estimated delivery in United States, on Tuesday 25 Jan 2022
Thymosin a1
CAS:62304-98-7
Bachem ID: 4095878.
Formula:
C129H215N33O55
Purity:
95.6%
Color and Shape:
White Lyophilisate
Molecular weight:
3106.50413
Estimated delivery in United States, on Tuesday 25 Jan 2022
Angiotensin I/II (1-7)
CAS:51833-78-4
Angiotensin (1-7), DRVYIHP, an enzymatically produced peptide of the renin-angiotensin system, shows pharmacologically distinct, tissue-specific …
Formula:
C41H62N12O11
Purity:
99.3%
Color and Shape:
White Powder
Molecular weight:
898.4661
Estimated delivery in United States, on Tuesday 25 Jan 2022
H-Lys-Pro-OH
CAS:52766-27-5
This dipeptide has the potential as a very promising healing agent in ulcer therapy. Daily …
Formula:
C11H21N3O3
Purity:
> 99%
Color and Shape:
White
Molecular weight:
243.15829
Estimated delivery in United States, on Tuesday 25 Jan 2022
LL-37 amide
CAS:597562-32-8
LL-37 amide is an antimicrobial peptide with angiogenic activity.
Formula:
C205H341N61O52
Purity:
97.3%
Color and Shape:
White Lyophilisate
Molecular weight:
4489.59141
Estimated delivery in United States, on Tuesday 25 Jan 2022
LL-37
CAS:154947-66-7
LL-37 is an antimicrobial peptide with angiogenic activity. It corresponds to the C-terminal sequence (134-170) …
Formula:
C205H340N60O53
Purity:
96.7%
Color and Shape:
White
Molecular weight:
4490.57543
Estimated delivery in United States, on Tuesday 25 Jan 2022
Thymosin a1
CAS:62304-98-7
Thymosin a1, originally isolated from calf thymus, acts as an immunomodulator. Additionally, the peptide showed …
Formula:
C129H215N33O55
Molecular weight:
3106.50413
Estimated delivery in United States, on Tuesday 25 Jan 2022
Momelotinib Mesylate
CAS:1056636-07-7
Momelotinib Mesylate is an ATP-competitive JAK1/JAK2 inhibitor (IC50: 11 nM/18 nM). It has 10-fold selectivity …
Formula:
C24H26N6O5S
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
510.57
Estimated delivery in United States, on Tuesday 1 Feb 2022
HS-10296
CAS:1899921-05-1
Hs-10296 is an inhibitor of EGFR activation mutation and tolerant mutation of EGFR T790M, which …
Formula:
C30H35N7O2
Purity:
99.85%
Color and Shape:
Solid
Molecular weight:
525.66
Estimated delivery in United States, on Tuesday 1 Feb 2022
Entrectinib
CAS:1108743-60-7
Entrectinib is an inhibitor of TrkA (IC50: 1.7 nM), TrkB (IC50: 0.1 nM), and TrkC …
Formula:
C31H34F2N6O2
Purity:
99.49%
Color and Shape:
solid
Molecular weight:
560.64
Estimated delivery in United States, on Tuesday 1 Feb 2022
Ginsenoside Rg3
CAS:14197-60-5
Ginsenoside Rg3 possess an ability to inhibit the lung metastasis of tumor cells via inhibition …
Formula:
C42H72O13
Purity:
99.53%
Color and Shape:
solid
Molecular weight:
785.02
Estimated delivery in United States, on Tuesday 1 Feb 2022
Withanolide A
CAS:32911-62-9
Withanolide A extends the lifespan in human EGFR-driven cancerous Caenorhabditis elegans.
Formula:
C28H38O6
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
470.6
Estimated delivery in United States, on Tuesday 1 Feb 2022
AST 487
CAS:630124-46-8
AST 487 is a RET kinase inhibitor, inhibiting RET autophosphorylation and activation of downstream effectors. …
Formula:
C26H30F3N7O2
Purity:
99.56%
Color and Shape:
solid
Molecular weight:
529.56
Estimated delivery in United States, on Tuesday 1 Feb 2022
SU5208
CAS:62540-08-3
SU5208 is a compound with bioactivity.SU5208 inhibits vascular endothelial growth factor receptor-2 (VEGFR2).
Formula:
C13H9NOS
Purity:
100.00%
Color and Shape:
solid
Molecular weight:
227.28
Estimated delivery in United States, on Tuesday 1 Feb 2022
KX2-391
CAS:897016-82-9
KX2-391 is a highly selective Src kinase inhibitor that has demonstrated efficacy in pre-Clinicalal animal …
Formula:
C26H29N3O3
Purity:
99.43%
Color and Shape:
solid
Molecular weight:
431.53
Estimated delivery in United States, on Tuesday 1 Feb 2022
Mutated EGFR-IN-1
CAS:1421372-66-8
Mutated EGFR-IN-1 is a useful intermediate for the inhibitors design for mutated EGFR, such as …
Formula:
C25H31N7O
Purity:
99.73%
Color and Shape:
solid
Molecular weight:
445.56
Estimated delivery in United States, on Tuesday 1 Feb 2022
Cyasterone
CAS:17086-76-9
Cyasterone, a natural EGFR inhibitor, can inhibit the growth of A549 and MGC823 cells, via …
Formula:
C29H44O8
Purity:
99.32%
Color and Shape:
solid
Molecular weight:
520.66
Estimated delivery in United States, on Tuesday 1 Feb 2022
NCT503
CAS:1916571-90-8
NCT-503 is an inhibitor of 3-phosphoglycerate dehydrogenase (PHGDH), inhibiting serine synthesis from 3-phosphoglycerate in cells.
Formula:
C20H23F3N4S
Purity:
98.91%
Color and Shape:
Solid
Molecular weight:
408.49
Estimated delivery in United States, on Tuesday 1 Feb 2022
Tesevatinib
CAS:781613-23-8
Tesevatinib is an orally available, multi-target tyrosine kinase inhibitor (IC50s: 0.3, 16, 1.5, 8.7, and …
Formula:
C24H25Cl2FN4O2
Molecular weight:
491.39
Estimated delivery in United States, on Tuesday 1 Feb 2022
LDN214117
CAS:1627503-67-6
LDN-214117 is a potent and selective ALK2 inhibitor.
Formula:
C25H29N3O3
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
419.52
Estimated delivery in United States, on Tuesday 1 Feb 2022
O-Nornuciferine
CAS:3153-55-7
O-Nornuciferine reveals distinct in vitro hERG blockages measured in HEK293 cells with the IC50 value …
Formula:
C18H19NO2
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
281.35
Estimated delivery in United States, on Tuesday 1 Feb 2022
Inulicin
CAS:33627-41-7
Inulicin, an active compound isolated from Inula Britannica L, inhibits VEGF-mediated activation of Src and …
Formula:
C17H24O5
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
308.37
Estimated delivery in United States, on Tuesday 1 Feb 2022
(Z)-Semaxinib
CAS:194413-58-6
Semaxanib (SU5416) is a potent and selective VEGFR(Flk-1/KDR) inhibitor (IC50: 1.23 μM), 20-fold more selective …
Formula:
C15H14N2O
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
238.28
Estimated delivery in United States, on Tuesday 1 Feb 2022
Erdafitinib
CAS:1346242-81-6
Erdafitinib is a quinoxaline derivative compound, acts on FGFR1/2/3/4.
Formula:
C25H30N6O2
Purity:
99.04%
Color and Shape:
solid
Molecular weight:
446.55
Estimated delivery in United States, on Tuesday 1 Feb 2022
TL02-59 dihydrochloride
CAS:2415263-06-6
TL02-59 dihydrochloride is an orally active inhibitor of Src-family kinase Fgr (IC50: 0.03 nM).
Formula:
C32H36Cl2F3N5O4
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
682.56
Estimated delivery in United States, on Tuesday 1 Feb 2022
Olmutinib
CAS:1353550-13-6
Olmutinib is an orally available small molecule, a mutant-selective inhibitor of epidermal growth factor receptor …
Formula:
C26H26N6O2S
Purity:
99.00%
Molecular weight:
486.59
Estimated delivery in United States, on Tuesday 1 Feb 2022
Ponatinib
CAS:943319-70-8
Ponatinib is an orally available, multitargeted kinase inhibitor (IC50s: 0.37/1.1/1.5/2.2/5.4 nM for Abl, PDGFR, VEGFR2, …
Formula:
C29H27F3N6O
Purity:
99.58%
Color and Shape:
solid
Molecular weight:
532.56
Estimated delivery in United States, on Tuesday 1 Feb 2022
AV-412
CAS:451493-31-5
AV-412 is an EGFR inhibitor (EGFR, EGFR T790M, EGFR L858R, EGFR L858R/T790M and ErbB2 with …
Formula:
C41H44ClFN6O7S2
Purity:
99.85%
Color and Shape:
solid
Molecular weight:
851.41
Estimated delivery in United States, on Tuesday 1 Feb 2022
BAY 87-2243
CAS:1227158-85-1
BAY 87-2243 is a potent and selective inhibitor of hypoxia-inducible factor-1 (HIF-1).
Formula:
C26H26F3N7O2
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
525.53
Estimated delivery in United States, on Tuesday 1 Feb 2022
JAK-IN-11
CAS:916742-11-5
JAK-IN-11 is a potent and selective inhibitor of JAK, has the potential for the skin …
Formula:
C23H22FN5O4S
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
483.52
Estimated delivery in United States, on Tuesday 1 Feb 2022
Gefitinib
CAS:184475-35-2
Gefitinib is an EGFR tyrosine kinase inhibitor and can inhibit Tyr1173, Tyr992, Tyr1173 and Tyr992 …
Formula:
C22H24ClFN4O3
Purity:
100.00%
Color and Shape:
Light-Yellow Crystalline Powder
Molecular weight:
446.91
Estimated delivery in United States, on Tuesday 1 Feb 2022
AG 555
CAS:133550-34-2
AG 555 is an EGFR tyrosine kinase inhibitor.
Formula:
C19H18N2O3
Purity:
99.50%
Color and Shape:
solid
Molecular weight:
322.36
Estimated delivery in United States, on Tuesday 1 Feb 2022
Dovitinib Lactate
CAS:915769-50-5
Dovitinib (TKI258) Lactate is the Lactate of Dovitinib, which is a multitargeted RTK inhibitor, mostly …
Formula:
C24H27FN6O4
Purity:
99.17%
Molecular weight:
482.51
Estimated delivery in United States, on Tuesday 1 Feb 2022
Vactosertib Hydrochloride
CAS:1352610-25-3
Vactosertib Hydrochloride is an orally active and ATP-competitive ALK5 inhibitor (IC50: 12.9 nM). It has …
Formula:
C22H19ClFN7
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
435.88
Estimated delivery in United States, on Tuesday 1 Feb 2022
Crizotinib
CAS:877399-52-5
Crizotinib is an ATP-competitive small-molecule tyrosine kinases inhibitor of c-MET (IC50: 8 nM) and ALK …
Formula:
C21H22Cl2FN5O
Purity:
99.00%
Color and Shape:
solid
Molecular weight:
450.34
Estimated delivery in United States, on Tuesday 1 Feb 2022
Regorafenib Hydrochloride
CAS:835621-07-3
Regorafenib Hydrochloride is a new oral multikinase inhibitor of angiogenic, stromal and oncogenic receptor tyrosine …
Formula:
C21H16Cl2F4N4O3
Purity:
100.00%
Color and Shape:
solid
Molecular weight:
519.28
Estimated delivery in United States, on Tuesday 1 Feb 2022
Sennoside B
CAS:128-57-4
Sennoside B is an anthranoid. Anthranoid derivatives are used all over the world as a …
Formula:
C42H38O20
Color and Shape:
Light Yellow Crystal
Molecular weight:
862.74
Estimated delivery in United States, on Tuesday 1 Feb 2022
PF04929113
CAS:908115-27-5
SNX-5422 is a synthetic, novel, small molecule Hsp90 Inhibitor. As an oral formulation that demonstrates …
Formula:
C25H30F3N5O4
Purity:
99.06%
Color and Shape:
solid
Molecular weight:
521.53
Estimated delivery in United States, on Tuesday 1 Feb 2022
Syk Inhibitor II (hydrochloride)
CAS:227449-73-2
Spleen tyrosine kinase (Syk) is a non-receptor tyrosine kinase that, upon phosphorylation, binds to immunoreceptor …
Formula:
C14H17Cl2F3N6O
Color and Shape:
solid
Molecular weight:
413.22
Estimated delivery in United States, on Tuesday 1 Feb 2022
SAR20347
CAS:1450881-55-6
SAR-20347 is an inhibitor of TYK2, JAK1/2/3 (IC50: 0.6/23/26/41 nM).
Formula:
C21H18ClFN4O4
Purity:
99.35%
Color and Shape:
Solid
Molecular weight:
444.85
Estimated delivery in United States, on Tuesday 1 Feb 2022
Epertinib hydrochloride
CAS:2071195-74-7
Epertinib hydrochloride shows potent antitumor activity. Epertinib hydrochloride is a potent, orally active, reversible, and …
Formula:
C30H28Cl2FN5O3
Purity:
99.36%
Color and Shape:
Solid
Molecular weight:
596.48
Estimated delivery in United States, on Tuesday 1 Feb 2022
Lanraplenib monosuccinate
CAS:1800046-97-2
Lanraplenib monosuccinate inhibits SYK activity in platelets via the glycoprotein VI (GPVI) receptor without prolonging …
Formula:
C27H31N9O5
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
561.59
Estimated delivery in United States, on Tuesday 1 Feb 2022
ALK5 Inhibitor IV
CAS:909910-43-6
A 83-01 is a selective inhibitor of TGF- type I receptor ALK5 kinase, type I …
Formula:
C25H19N5S
Purity:
97.00%
Color and Shape:
solid
Molecular weight:
421.52
Estimated delivery in United States, on Tuesday 1 Feb 2022
AG 494
CAS:133550-35-3
AG-494 is an inhibitor of epidermal growth factor receptor kinase.
Formula:
C16H12N2O3
Purity:
99.50%
Color and Shape:
solid
Molecular weight:
280.28
Estimated delivery in United States, on Tuesday 1 Feb 2022
TG 100801 Hydrochloride
CAS:1018069-81-2
TG 100801 Hydrochloride is a prodrug to treat age-related macular degeneration. TG 100572 is a …
Formula:
C33H31Cl2N5O3
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
616.54
Estimated delivery in United States, on Tuesday 1 Feb 2022
Mutated EGFR-IN-3
CAS:2375107-27-8
Mutated EGFR-IN-3 is a ATP-competitive and highly selective allosteric dibenzodiazepinone EGFR(L858R/T790M) and EGFR(L858R/T790M/C797S) inhibitor(IC50 of …
Formula:
C31H29FN4O2
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
508.59
Estimated delivery in United States, on Tuesday 1 Feb 2022
Osimertinib mesylate
CAS:1421373-66-1
Osimertinib (AZD-9291) is an irreversible and mutant selective EGFR inhibitor (IC50s: 12/1 nM for EGFR(L858R) …
Formula:
C29H37N7O5S
Purity:
98.65%
Color and Shape:
solid
Molecular weight:
595.71
Estimated delivery in United States, on Tuesday 1 Feb 2022
TG 100572
CAS:867334-05-2
TG 100572 is a inhibitor of multi-targeted kinase which inhibits receptor tyrosine kinases and Src …
Formula:
C26H26ClN5O2
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
475.97
Estimated delivery in United States, on Tuesday 1 Feb 2022
IBT6A
CAS:1022150-12-4
IBT6A is an impurity of Ibrutinib. Ibrutinib is a Btk inhibitor (IC50: 0.5 nM). IBT6A …
Formula:
C22H22N6O
Purity:
99.88%
Color and Shape:
solid
Molecular weight:
386.45
Estimated delivery in United States, on Tuesday 1 Feb 2022
LDN193189
CAS:1062368-24-4
LDN193189 (DM 3189) is a selective BMP signaling inhibitor, inhibiting the transcriptional activity of ALK2 …
Formula:
C25H22N6
Purity:
99.11%
Color and Shape:
solid
Molecular weight:
406.48
Estimated delivery in United States, on Tuesday 1 Feb 2022
ITK inhibitor 2
CAS:1309784-09-5
ITK inhibitor 2 is a interleukin-2-inducible T-cell kinase (ITK) inhibitor , with an IC50 of …
Formula:
C25H33N5O2
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
435.56
Estimated delivery in United States, on Tuesday 1 Feb 2022
SYP-5
CAS:1384268-04-5
SYP-5 is a novel inhibitor of HIF-1, suppresses tumor cells invasion and angiogenesis.
Formula:
C18H16O3S
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
312.38
Estimated delivery in United States, on Tuesday 1 Feb 2022
PRN1371
CAS:1802929-43-6
PRN1371 is a specific and potent FGFR1-4 and CSF1R inhibitor (IC50s: 0.6/1.3/4.1/19.3/8.1 nM for FGFR1/2/3/4 …
Formula:
C26H30Cl2N6O4
Purity:
99.72%
Color and Shape:
solid
Molecular weight:
561.46
Estimated delivery in United States, on Tuesday 1 Feb 2022
Pexidartinib
CAS:1029044-16-3
Pexidartinib is a capsule formulation containing a small-molecule receptor tyrosine kinase (RTK) inhibitor of KIT, …
Formula:
C20H15ClF3N5
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
417.81
Estimated delivery in United States, on Tuesday 1 Feb 2022
6-Demethoxytangeretin
CAS:6601-66-7
6-Demethoxytangeretin is a citrus flavonoid isolated from Citrus depressa.
Formula:
C19H18O6
Purity:
99.89%
Color and Shape:
solid
Molecular weight:
342.3
Estimated delivery in United States, on Tuesday 1 Feb 2022
SC99
CAS:882290-02-0
SC99 is a selective inhibitor of JAK2-STAT3 activation. SC99 downregulates the expression of STAT3-modulated genes.SC99 …
Formula:
C15H8Cl2FN3O
Molecular weight:
336.15
Estimated delivery in United States, on Tuesday 1 Feb 2022
TAS-115
CAS:1190836-34-0
TAS-115 is a potent inhibitor of VEGFR and hepatocyte growth factor receptor (c-Met/HGFR)-targeted kinase(IC50s of …
Formula:
C27H23FN4O4S
Purity:
99.15%
Color and Shape:
Solid
Molecular weight:
518.56
Estimated delivery in United States, on Tuesday 1 Feb 2022
SAR131675
CAS:1092539-44-0
SAR131675 is an effective and specific VEGFR-3 inhibitor. It inhibited VEGFR-3 tyrosine kinase activity (IC50: …
Formula:
C18H22N4O4
Purity:
98.73%
Color and Shape:
solid
Molecular weight:
358.16
Estimated delivery in United States, on Tuesday 1 Feb 2022
EGFR-IN-5
CAS:2225887-26-1
EGFR-IN-5 is a EGFR inhibitor, EGFR-IN-5 with IC50s of 10.4, 1.1, 34, 7.2 nM for …
Formula:
C31H38FN9O
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
571.69
Estimated delivery in United States, on Tuesday 1 Feb 2022
Mollugin
CAS:55481-88-4
Mollugin may be a JAK2 inhibitor and inhibits LPS-induced inflammatory responses by blocking the activation …
Formula:
C17H16O4
Purity:
99.90%
Color and Shape:
solid
Molecular weight:
284.3
Estimated delivery in United States, on Tuesday 1 Feb 2022
Tandutinib
CAS:387867-13-2
Tandutinib (MLN518, CT53518), an effective FLT3 antagonist (IC50: 0.22 μM), can also inhibit c-Kit and …
Formula:
C31H42N6O4
Purity:
99.74%
Color and Shape:
White Solid
Molecular weight:
562.7
Estimated delivery in United States, on Tuesday 1 Feb 2022
ALK2-IN-2
CAS:2254409-25-9
ALK2-IN-2 is a potent and selective inhibitor of ALK2 (IC50: 9 nM), and over 700-fold …
Formula:
C28H27N5O2S
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
497.61
Estimated delivery in United States, on Tuesday 1 Feb 2022
Sunitinib D10
CAS:1126721-82-1
Sunitinib D10 is a deuterium labeled Sunitinib. Sunitinib is a inhibitor of multi-targeted receptor tyrosine …
Formula:
C22H17D10FN4O2
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
408.54
Estimated delivery in United States, on Tuesday 1 Feb 2022
ZM 39923 HCl
CAS:1021868-92-7
ZM 39923 HCl is an JAK1/3 inhibitor with pIC50 of 4.4/7.1, almost no activity to …
Formula:
C23H25NO·HCl
Purity:
98.05%
Color and Shape:
solid
Molecular weight:
367.91
Estimated delivery in United States, on Tuesday 1 Feb 2022
RTC-5
CAS:1423077-49-9
RTC-5 demonstrated efficacy against a xenograft model of an EGFR driven cancer without the neurotropic …
Formula:
C24H22ClF3N2O3S
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
510.96
Estimated delivery in United States, on Tuesday 1 Feb 2022
Olafertinib
CAS:1660963-42-7
CK-101 (RX-518) is a novel mutant-selective, irreversible, orally available EGFR inhibitor. It can overcome T790M-mediated …
Formula:
C29H28F2N6O2
Purity:
98.43%
Color and Shape:
Solid
Molecular weight:
530.57
Estimated delivery in United States, on Tuesday 1 Feb 2022
GZD856
CAS:1257628-64-0
GZD856 is an orally bioavailable PDGFR/ inhibitor (IC50s: 68.6 and 136.6 nM) with anti-lung cancer …
Formula:
C29H27F3N6O
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
532.56
Estimated delivery in United States, on Tuesday 1 Feb 2022
WZ8040
CAS:1214265-57-2
WZ8040 is a novel mutant-selective irreversible EGFRT790M inhibitor, does not inhibit ERBB2 phosphorylation (T798I).
Formula:
C24H25ClN6OS
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
481.01
Estimated delivery in United States, on Tuesday 1 Feb 2022
Ripretinib
CAS:1442472-39-0
Ripretinib is an orally bioavailable inhibitor of KIT and PDGFRA.
Formula:
C24H21BrFN5O2
Purity:
99.72%
Color and Shape:
Solid
Molecular weight:
510.36
Estimated delivery in United States, on Tuesday 1 Feb 2022
PF-06651600
CAS:1792180-81-4
PF-06651600 is a potent JAK3-selective inhibitor (IC50: 33.1 nM).
Formula:
C15H19N5O
Purity:
99.10%
Color and Shape:
Solid
Molecular weight:
285.34
Estimated delivery in United States, on Tuesday 1 Feb 2022
EGFR-IN-1
CAS:1625677-63-5
EGFR-IN-1 displays strong antiproliferative activity against the H1975 cells and the first line mutant HCC827 …
Formula:
C28H30N6O4
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
514.58
Estimated delivery in United States, on Tuesday 1 Feb 2022
DMOG
CAS:89464-63-1
DMOG, an antagonist of the -ketoglutarate cofactor, is an inhibitor for HIF prolyl hydroxylase.
Formula:
C6H9NO5
Purity:
80.23%
Color and Shape:
solid
Molecular weight:
175.14
Estimated delivery in United States, on Tuesday 1 Feb 2022
E-4031
CAS:113559-13-0
E-4031 is a methanesulfonanilide class III antiarrhythmic agent that prolongs cardiac action potential duration by …
Formula:
C21H29Cl2N3O3S
Molecular weight:
474.44
Estimated delivery in United States, on Tuesday 1 Feb 2022
UNC2025 2HCl (1429881-91-3(free base))
UNC2025 is a potent and orally bioavailable Mer/Flt3 dual inhibitor with IC50 of 0.8/0.74 nM …
Formula:
C28H42Cl2N6O
Purity:
98.56%
Color and Shape:
solid
Molecular weight:
549.62
Estimated delivery in United States, on Tuesday 1 Feb 2022
ALK-IN-5
CAS:2351929-66-1
ALK-IN-5 is a potent, selective, and brain-penetrant inhibitor of anaplastic lymphoma kinase (ALK, IC50: 2.9 …
Formula:
C24H25FN6O3
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
464.49
Estimated delivery in United States, on Tuesday 1 Feb 2022
BMS-935177
CAS:1231889-53-4
BMS-935177 is a potent and selective reversible inhibitor of Brutons tyrosine kinase (Btk), with an …
Formula:
C31H26N4O3
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
502.56
Estimated delivery in United States, on Tuesday 1 Feb 2022
Biochanin A
CAS:491-80-5
Biochanin A is an isoflavone derivative isolated from red clover Trifolium pratense with anticarcinogenic properties. …
Formula:
C16H12O5
Purity:
97.69%
Color and Shape:
Solid
Molecular weight:
284.26
Estimated delivery in United States, on Tuesday 1 Feb 2022
TX1-85-1
CAS:1603845-32-4
TX1-85-1 induces partial degradation of Her3 protein and attenuates Her3-dependent signaling. TX1-85-1 is an irreversible …
Formula:
C32H36N8O3
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
580.68
Estimated delivery in United States, on Tuesday 1 Feb 2022
A 419259
CAS:364042-47-7
A 419259 is a pyrrolo-pyrimidine inhibitor, designed to enhance selectivity towards the Src family (IC50s: …
Formula:
C29H34N6O
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
482.62
Estimated delivery in United States, on Tuesday 1 Feb 2022
AZD2932
CAS:883986-34-3
AZD2932 is a potent and multi-targeted kinase inhibitor VEGFR2, PDGF, Flt-3, and c-Kit.
Formula:
C24H25N5O4
Purity:
97.71%
Color and Shape:
solid
Molecular weight:
447.49
Estimated delivery in United States, on Tuesday 1 Feb 2022
PD 089828
CAS:179343-17-0
PD 089828 is a competitive inhibitor of the receptor tyrosine kinases FGFR1, PDGFR, and EGFR …
Formula:
C18H18Cl2N6O
Purity:
96.78%
Molecular weight:
405.28
Estimated delivery in United States, on Tuesday 1 Feb 2022
CNX774
CAS:1202759-32-7
CNX-774 is a highly specific, irreversible, and orally active BTK inhibitor (IC50<1 nM).
Formula:
C26H22FN7O3
Purity:
98.77%
Color and Shape:
solid
Molecular weight:
499.5
Estimated delivery in United States, on Tuesday 1 Feb 2022
Alofanib
CAS:1612888-66-0
Alofanib is a selective allosteric inhibitor of FGFR2 and has a dramatic inhibitory effect on …
Formula:
C19H15N3O6S
Purity:
99.53%
Color and Shape:
Solid
Molecular weight:
413.4
Estimated delivery in United States, on Tuesday 1 Feb 2022
Afatinib D6
CAS:1313874-96-2
Afatinib D6 (BIBW 2992 D6) is a deuterium-labeled Afatinib. Afatinib is an irreversible EGFR family …
Formula:
C24H19D6ClFN5O3
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
491.98
Estimated delivery in United States, on Tuesday 1 Feb 2022
EGFR mutant-IN-1
EGFR mutant- in-1, A 5-methylpyrimidopyridone derivative are effective selective EGFRL858R/T790M/C797S mutant inhibitors with IC50 of …
Formula:
C34H39ClFN7O2
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
632.17
Estimated delivery in United States, on Tuesday 1 Feb 2022
Chebulic acid
CAS:23725-05-5
Chebulic acid, a phenolcarboxylic acid compound isolated from Terminalia chebula, has potent anti-oxidant activity,which breaks …
Formula:
C14H12O11
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
356.24
Estimated delivery in United States, on Tuesday 1 Feb 2022
IN-1130
CAS:868612-83-3
IN-1130 is a highly selective inhibitor of transforming growth factor- type I receptor kinase (ALK5) …
Formula:
C25H20N6O
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
420.47
Estimated delivery in United States, on Tuesday 1 Feb 2022
SU16f
CAS:251356-45-3
SU16f is a potent and selective PDGFR inhibitor (IC50s: 10 nM, 140 nM, 2.29 μM …
Formula:
C24H22N2O3
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
386.44
Estimated delivery in United States, on Tuesday 1 Feb 2022
Peficitinib
CAS:944118-01-8
Peficitinib (ASP015K, JNJ-54781532) is an orally bioavailable JAK inhibitor. Phase 3.
Formula:
C18H22N4O2
Purity:
98.0%
Molecular weight:
326.39
Estimated delivery in United States, on Tuesday 1 Feb 2022
AZD4547
CAS:1035270-39-3
AZD4547, a new-type specific FGFR inhibitor, targets for FGFR1/2/3 (IC50: 0.2/2.5/1.8 nM in cell-free assays).
Formula:
C26H33N5O3
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
463.57
Estimated delivery in United States, on Tuesday 1 Feb 2022
PF-06700841 (P-Tosylate)
CAS:2140301-96-6
PF-06700841 P-Tosylate is a potent dual inhibitor of Janus kinase 1 (JAK1) and TYK2 (IC50s …
Formula:
C25H29F2N7O4S
Purity:
99.82%
Color and Shape:
Solid
Molecular weight:
561.60
Estimated delivery in United States, on Tuesday 1 Feb 2022
Mobocertinib
CAS:1847461-43-1
Mobocertinib is a potent inhibitor of epidermal growth factor receptor (EGFR) and an antineoplastic agent
Formula:
C32H39N7O4
Purity:
99.72%
Color and Shape:
Solid
Molecular weight:
585.71
Estimated delivery in United States, on Tuesday 1 Feb 2022
CP-547632
CAS:252003-65-9
CP-547632 is a well-tolerated, orally-bioavailable inhibitor of the VEGFR-2 and basic fibroblast growth factor (FGF) …
Formula:
C20H24BrF2N5O3S
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
532.4
Estimated delivery in United States, on Tuesday 1 Feb 2022
