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GPR
Bimatoprost acid
CAS:38344-08-0
Bimatoprost acid is a metabolically stable analog of PGF2 and has a potential antagonistic activity …
Formula:
C23H32O5
Purity:
99.19%
Molecular weight:
388.5
Estimated delivery in United States, on Thursday 3 Feb 2022
APD 668
CAS:832714-46-2
APD668 is a potent GPR119 agonist with EC50 of 2.7 nM and 33 nM for …
Formula:
C21H24FN5O5S
Purity:
99.74%
Color and Shape:
solid
Molecular weight:
477.51
Estimated delivery in United States, on Thursday 3 Feb 2022
GW 9508
CAS:885101-89-3
GW9508 is a potent and selective agonist for FFA1 (GPR40), stimulates insulin secretion in a …
Formula:
C22H21NO3
Color and Shape:
solid
Molecular weight:
347.41
Estimated delivery in United States, on Thursday 3 Feb 2022
Azathioprine
CAS:446-86-6
Azathioprine, an immunosuppressive agent, inhibits purine synthesis and GTP-binding protein Rac1 activation.
Formula:
C9H7N7O2S
Purity:
100.00%
Color and Shape:
Pale Yellow Crystals From 50% Aq Acetone Physical Description Pale Yellow Crystals Or Yellowish Powder Decomposes At 243-
Molecular weight:
277.26
Estimated delivery in United States, on Thursday 3 Feb 2022
AZD1981
CAS:802904-66-1
AZD1981 is an effective and specific CRTh2 (DP2) receptor antagonist (IC50: 4 nM), showing >1000-fold …
Formula:
C19H17ClN2O3S
Purity:
99.54%
Color and Shape:
solid
Molecular weight:
388.87
Estimated delivery in United States, on Thursday 3 Feb 2022
GSK1292263
CAS:1032823-75-8
GSK1292263 is a GPR119 agonist and has been investigated for the treatment of DIABETES MELLITUS, …
Formula:
C23H28N4O4S
Purity:
98.34%
Color and Shape:
solid
Molecular weight:
456.56
Estimated delivery in United States, on Thursday 3 Feb 2022
Palosuran
CAS:540769-28-6
Palosuran (ACT-058362) is a new potent and specific antagonist of the human UT receptor.
Formula:
C25H30N4O2
Purity:
98.04%
Color and Shape:
solid
Molecular weight:
418.53
Estimated delivery in United States, on Thursday 3 Feb 2022
TUG891
CAS:1374516-07-0
TUG-891 is a G protein-coupled receptor (GPCR) expressed in intestine, adipocytes, and pro-inflammatory macrophages that …
Formula:
C23H21FO3
Purity:
99.21%
Color and Shape:
solid
Molecular weight:
364.41
Estimated delivery in United States, on Thursday 3 Feb 2022
GSK137647A
CAS:349085-82-1
GSK137647A is a selective FFA4 agonist.
Formula:
C16H19NO3S
Purity:
99.26%
Color and Shape:
solid
Molecular weight:
305.39
Estimated delivery in United States, on Thursday 3 Feb 2022
TAK875
CAS:1000413-72-8
TAK875 is a potent, selective and orally bioavailable GPR40 agonist.
Formula:
C29H32O7S
Purity:
99.82%
Color and Shape:
solid
Molecular weight:
524.63
Estimated delivery in United States, on Thursday 3 Feb 2022
TC-O 9311
CAS:444392-31-4
TC-O 9311 is a potent GPR139 agonist.
Formula:
C20H19N3O4
Purity:
99.81%
Color and Shape:
Solid
Molecular weight:
365.38
Estimated delivery in United States, on Thursday 3 Feb 2022
AH 7614
CAS:6326-06-3
AH 7614 is a selective and potent free fatty acid receptor 4 (FFA4/GPR120) antagonist.
Formula:
C20H17NO3S
Molecular weight:
351.42
Estimated delivery in United States, on Thursday 3 Feb 2022
CAY10595
CAS:916047-16-0
CAY10595 is a potent antagonist of the CRTH2/DP2 receptor (Ki: 10 nM).
Formula:
C20H13Cl2FN2O5
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
451.23
Estimated delivery in United States, on Thursday 3 Feb 2022
VER155008
CAS:1134156-31-2
VER-155008 is a potent Hsp70 family inhibitor with IC50 of 0.5 μM, 2.6 μM, and …
Formula:
C25H23Cl2N7O4
Purity:
99.55%
Color and Shape:
solid
Molecular weight:
556.4
Estimated delivery in United States, on Thursday 3 Feb 2022
G-1
CAS:881639-98-1
G-1 is a nonsteroidal, high-affinity and selective GPR30 agonist (Ki: 11 nM).
Formula:
C21H18BrNO3
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
412.28
Estimated delivery in United States, on Thursday 3 Feb 2022
GPR40 Agonist 2
CAS:1147729-48-3
GPR40 Agonist 2 is a GPR40 agonist extracted from patent WO2009054479A1. It can be used …
Formula:
C24H30O3
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
366.49
Estimated delivery in United States, on Thursday 3 Feb 2022
MK-6892
CAS:917910-45-3
MK-6892 is a selective and full agonist for the high-affinity nicotinic acid receptor GPR109A (Ki: …
Formula:
C19H22N4O5
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
386.4
Estimated delivery in United States, on Thursday 3 Feb 2022
TAK-875 Hemihydrate
CAS:1374598-80-7
TAK-875 is a selective GPR40 agonist with EC50 of 14 nM, 400-fold more potent than …
Formula:
C29H32O7SH2O
Purity:
98.0%
Color and Shape:
solid
Molecular weight:
533.63
Estimated delivery in United States, on Thursday 3 Feb 2022
GW-1100
CAS:306974-70-9
GW-1100 is a selective antagonist of GPR40 (pIC50: 6.9). GW1100 also plays the role of …
Formula:
C27H25FN4O4S
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
520.58
Estimated delivery in United States, on Thursday 3 Feb 2022
FTBMT
CAS:1358575-02-6
FTBMT is a selective GPR52 agonist (EC50: 75 nM) and has antipsychotic and procognitive properties.
Formula:
C19H16F4N4O
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
392.35
Estimated delivery in United States, on Thursday 3 Feb 2022
MBX2982
CAS:1037792-44-1
MBX-2982 is a selective, orally-available GPR119 agonist, used for the treatment of diabetes.
Formula:
C22H24N8OS
Color and Shape:
solid
Molecular weight:
448.54
Estimated delivery in United States, on Thursday 3 Feb 2022
GPR84 antagonist 8
CAS:1445846-30-9
GPR84 antagonist 8 is a selective GPR84 antagonist.
Formula:
C23H23N3O5
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
421.45
Estimated delivery in United States, on Thursday 3 Feb 2022
GLPG0974
CAS:1391076-61-1
GLPG0974 is an antagonist of free fatty acid receptor-2 (IC50: 9 nM).
Formula:
C25H25ClN2O4S
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
485
Estimated delivery in United States, on Thursday 3 Feb 2022
Palosuran hydrochloride 540769-28-6(free base
Palosuran is a new potent and specific antagonist of the human UT receptor with an …
Formula:
C25H31ClN4O2
Purity:
99.75%
Color and Shape:
solid
Molecular weight:
454.99
Estimated delivery in United States, on Thursday 3 Feb 2022
Benzyl nicotinate
CAS:94-44-0
Benzyl Nicotinate is a agonist of GPR109A receptor and GPR109B receptor
Formula:
C13H11NO2
Purity:
98.22%
Color and Shape:
Yellow Liquid
Molecular weight:
213.23
Estimated delivery in United States, on Thursday 3 Feb 2022
Firuglipel
CAS:1371591-51-3
Firuglipel is an orally available and selective agonist of GPR119.
Formula:
C25H26FN3O5
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
467.49
Estimated delivery in United States, on Thursday 3 Feb 2022
hGPR91 antagonist 1
CAS:1314796-00-3
hGPR91 antagonist 1 is a potent and selective hGPR91 antagonist (IC50: 7 μM).
Formula:
C31H23F4N3O
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
529.53
Estimated delivery in United States, on Thursday 3 Feb 2022
Pamoic acid
CAS:130-85-8
Pamoic acid is the orphan G protein-coupled receptor GPR35 agonist. Pamoic acid activates ERK and …
Formula:
C23H16O6
Purity:
99.99%
Color and Shape:
Fine Yellow Powder
Molecular weight:
388.37
Estimated delivery in United States, on Thursday 3 Feb 2022
PU-H54
CAS:1454619-13-6
PU-H54 is a purine-based inhibitor of Grp94. It is a Grp94-selective resorcinol-based inhibitor isolated through …
Formula:
C18H19N5S
Molecular weight:
337.45
Estimated delivery in United States, on Thursday 3 Feb 2022
CRTh2 antagonist 1
CAS:1379445-54-1
CRTh2 antagonist 1 is a CRTh2 antagonist (IC50: 89 nM).
Formula:
C23H25N3O5S
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
455.53
Estimated delivery in United States, on Thursday 3 Feb 2022
JNJ63533054
CAS:1802326-66-4
JNJ-63533054 is a potent and selective agonist of hGPR139 with an EC50 = 16 nM.
Formula:
C17H17ClN2O2
Purity:
99.87%
Color and Shape:
Solid
Molecular weight:
316.78
Estimated delivery in United States, on Thursday 3 Feb 2022
CID 2745687
CAS:264233-05-8
CID 2745687 is a GPR35 antagonist that inhibited the effects at human GPR35 of cromolyn …
Formula:
C17H19F2N5O2S
Molecular weight:
395.43
Estimated delivery in United States, on Thursday 3 Feb 2022
Grp94 Inhibitor-1
CAS:2234897-35-7
Grp94 Inhibitor-1 is a potent, selective Grp94 inhibitor (IC50 : 2 nM).
Formula:
C22H28N2O2
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
352.47
Estimated delivery in United States, on Thursday 3 Feb 2022
NF-56-EJ40
CAS:2380230-73-7
NF-56-EJ40 is a high-affinity and highly selective antagonist of human SUCNR1 (GPR91) (IC50 of 25 …
Formula:
C27H29N3O3
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
443.54
Estimated delivery in United States, on Thursday 3 Feb 2022
GPR120 receptor agonist
CAS:1234844-11-1
A potent and selective GPR120 receptor agonist.
Formula:
C22H25ClO4
Purity:
99.52%
Color and Shape:
Solid
Molecular weight:
388.89
Estimated delivery in United States, on Thursday 3 Feb 2022
CRTh2 antagonist 2
CAS:780763-95-3
CRTh2 antagonist selective and potent CRTH2 antagonist, IC5010 nM. CRTh2 antagonist 2 can be used …
Formula:
C26H23ClN4O3
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
474.94
Estimated delivery in United States, on Thursday 3 Feb 2022
HA15
CAS:1609402-14-3
HA15 targets specifically BiP/GRP78/HSPA5. HA15 exhibits anti-cancerous activity on all melanoma cells tested, including cells …
Formula:
C23H22N4O3S2
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
466.58
Estimated delivery in United States, on Thursday 3 Feb 2022
Kisspeptin-10, human (TFA)(374675-21-5,FREE)
Kisspeptin-10, human TFA is a potent vasoconstrictor and angiogenesis inhibitor. Kisspeptin-10, human TFA acts as …
Formula:
C63H83N17O14C2HF3O2
Purity:
100.00%
Color and Shape:
solid
Molecular weight:
1416.46
Estimated delivery in United States, on Thursday 3 Feb 2022
APD597
CAS:897732-93-3
APD597 is a GPR119 agonist, used in the treatment of type 2 diabetes.
Formula:
C21H29N5O6S
Purity:
99.63%
Color and Shape:
solid
Molecular weight:
479.55
Estimated delivery in United States, on Thursday 3 Feb 2022
Ramatroban
CAS:116649-85-5
Ramatroban (BAY u3405) is a thromboxane A(2) (TxA(2)) antagonist marketed for allergic rhinitis. It has …
Formula:
C21H21FN2O4S
Purity:
99.96%
Color and Shape:
Crystalline Solid
Molecular weight:
416.47
Estimated delivery in United States, on Thursday 3 Feb 2022
Kisspeptin-10, rat acetate(478507-53-8 free base)
Endogenous ligand for the rodent kisspeptin receptor (KISS1, GPR54).
Formula:
C65H87N17O17
Molecular weight:
1378.45
Estimated delivery in United States, on Thursday 3 Feb 2022
Fevipiprant
CAS:872365-14-5
Fevipiprant is a selective, potent, reversible competitive CRTh2 antagonist.
Formula:
C19H17F3N2O4S
Purity:
99.32%
Color and Shape:
solid
Molecular weight:
426.41
Estimated delivery in United States, on Thursday 3 Feb 2022
AR 231453
CAS:733750-99-7
AR 231453 is a selective and orally available GPR119 agonist,can stimulate -cell replication and improve …
Formula:
C21H24FN7O5S
Purity:
99.31%
Color and Shape:
solid
Molecular weight:
505.52
Estimated delivery in United States, on Thursday 3 Feb 2022
RTI-13951-33
CAS:2244884-08-8
RTI-13951-33 is an effective and brain-penetrant GPR88 agonist (EC50: 25 nM, in GPR88 cAMP functional …
Formula:
C28H33N3O3
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
459.58
Estimated delivery in United States, on Thursday 3 Feb 2022
GPR120 Agonist 1
CAS:1628448-77-0
GPR120 Agonist 1 is a selective GPR120 agonist. In GPR120 transfected HEK293 cells, GPR120 Agonist …
Formula:
C20H12ClF6NO3S
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
495.82
Estimated delivery in United States, on Thursday 3 Feb 2022
DC260126
CAS:346692-04-4
DC260126 is a small-molecule antagonist of FFA1 (GPR40)
Formula:
C16H18FNO2S
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
307.38
Estimated delivery in United States, on Thursday 3 Feb 2022
MS21570
CAS:65373-29-7
MS21570 as a GPR171 antagonist based on its ability to block,with an IC50 of 220 …
Formula:
C10H11N3S2
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
237.34
Estimated delivery in United States, on Thursday 3 Feb 2022
CAY10471 Racemate
CAS:844639-57-2
CAY 10471 is a potent, highly selective CRTH2/DP 2 receptor antagonist. CAY10471 binds to the …
Formula:
C21H21FN2O4S
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
416.47
Estimated delivery in United States, on Thursday 3 Feb 2022
Latanoprost
CAS:130209-82-4
Latanoprost is a prostaglandin F2alpha analogue and a prostanoid selective FP receptor agonist with an …
Formula:
C26H40O5
Purity:
99.76%
Color and Shape:
Pale Yellow Oil
Molecular weight:
432.59
Estimated delivery in United States, on Thursday 3 Feb 2022
TC-O9311
CAS:444932-31-4
TC-O9311 is an effective agonist of GPR139 (EC50 = 39 nM in CHO-K1 cells expressing …
Formula:
C20H19N3O4
Purity:
99.12%
Molecular weight:
365.39
Estimated delivery in United States, on Thursday 3 Feb 2022
Setipiprant
CAS:866460-33-5
Setipiprant is an orally available, selective CRTH2 antagonist (IC50: 6.0 nM). CRTH2 is a G …
Formula:
C24H19FN2O3
Purity:
99.71%
Color and Shape:
solid
Molecular weight:
402.42
Estimated delivery in United States, on Thursday 3 Feb 2022
Setogepram sodium salt
CAS:1254472-97-3
Setogepram sodium salt is an orally active GPR40 agonist and is an antagonist or inverse …
Formula:
C13H17NaO2
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
228.26
Estimated delivery in United States, on Thursday 3 Feb 2022
3-chloro-5-hydroxybenzoic Acid
CAS:53984-36-4
3-chloro-5-hydroxy Benzoic Acid (3-chloro-5-hydroxy BA) is an agonist of GPR81 (EC50 : 16 µM)
Formula:
C7H5ClO3
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
172.57
Estimated delivery in United States, on Thursday 3 Feb 2022
AM-4668
CAS:1011531-27-3
AM-4668 is a type 2 diabetes GPR40 agonist. For GPR40, in A9 cells (GPR40 IP3 …
Formula:
C24H19F3N2O4S
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
488.48
Estimated delivery in United States, on Thursday 3 Feb 2022
GSK256073
CAS:862892-90-8
GSK256073 is an orally active GPR109A agonist. GSK256073 also is a long-lasting and non-flushing HCA2 …
Formula:
C10H13ClN4O2
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
256.69
Estimated delivery in United States, on Thursday 3 Feb 2022
AS 1269574
CAS:330981-72-1
AS 1269574 is a potent, orally available GPR119 agonist. AS1269574 has the potential for the …
Formula:
C13H14BrN3O
Purity:
99.98%
Molecular weight:
308.18
Estimated delivery in United States, on Thursday 3 Feb 2022
Dihydromunduletone
CAS:674786-20-0
Dihydromunduletone (DHM) is a carotenoid derivative and selective strong adhesion G protein-coupled receptor (aGPCR) (GPR56 …
Formula:
C25H28O6
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
424.49
Estimated delivery in United States, on Thursday 3 Feb 2022
Setogepram
CAS:1002101-19-0
Setogepram is an orally active GPR40 agonist and is an antagonist or inverse agonist of …
Formula:
C13H18O2
Purity:
99.38%
Color and Shape:
solid
Molecular weight:
206.28
Estimated delivery in United States, on Thursday 3 Feb 2022
GTPL5846
CAS:83797-69-7
6-OAU(GTPL5846; 6-n-octylaminouracil) is a surrogate agonist of GPR84; activates human GPR84 in the presence of …
Formula:
C12H21N3O2
Purity:
99.01%
Color and Shape:
solid
Molecular weight:
239.31
Estimated delivery in United States, on Thursday 3 Feb 2022
BI-671800
CAS:1093108-50-9
BI-671800 is a highly specific and potent antagonist of chemoattractant receptor-homologous molecule on Th2 cells …
Formula:
C25H26F3N5O3
Purity:
98.06%
Molecular weight:
501.5
Estimated delivery in United States, on Thursday 3 Feb 2022
GPR4 antagonist 1
CAS:1197879-16-5
GPR4 antagonist 1 is a GPR4 antagonist (IC50: 189 nM).
Formula:
C27H37N5
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
431.62
Estimated delivery in United States, on Thursday 3 Feb 2022
cangrelor tetrasodium
CAS:163706-36-3
Cangrelor tetrasodium is a reversible and selective antagonist of platelet P2Y12, with prompt and potent …
Formula:
C17H21Cl2F3N5Na4O12P3S2
Purity:
100.00%
Color and Shape:
solid
Molecular weight:
864.29
Estimated delivery in United States, on Thursday 3 Feb 2022
AM-1638
CAS:1142214-62-7
AM-1638 is a full agonist of GPR40/FFA1 (EC50: 0.16 μM).
Formula:
C33H35FO4
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
514.63
Estimated delivery in United States, on Thursday 3 Feb 2022
YUM70
CAS:423145-35-1
YUM70 is a potent and selective glucose-regulated protein 78 (GRP78) inhibitor(with an IC50 of 1.5 …
Formula:
C21H19ClN2O4
Molecular weight:
398.84
Estimated delivery in United States, on Thursday 3 Feb 2022
GPR40/FFAR1 modulator 1
CAS:874755-26-7
GPR40/FFAR1 modulator 1 is an agonist and an allosteric modulator for Gq-coupled free fatty acid …
Formula:
C21H19N5O3
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
389.41
Estimated delivery in United States, on Thursday 3 Feb 2022
Timapiprant
CAS:851723-84-7
OC000459 is a potent and selective D prostanoid receptor 2 (DP2) antagonist (IC50: 13 nM).
Formula:
C21H17FN2O2
Purity:
99.89%
Color and Shape:
solid
Molecular weight:
348.37
Estimated delivery in United States, on Thursday 3 Feb 2022
Urotensin II (114-124), human acetate
Urotensin II (114-124), human acetate is an 11-amino acid residue peptide, is a potent vasoconstrictor …
Formula:
C66H89N13O20S2
Purity:
100.00%
Molecular weight:
1448.63
Estimated delivery in United States, on Thursday 3 Feb 2022
NE 52-QQ57
CAS:1401728-56-0
NE 52-QQ57 is a selective, and orally available antagonist of GPR4(IC50 : 70 nM),with anti-inflammatory …
Formula:
C24H28N6O
Purity:
99.93%
Color and Shape:
Solid
Molecular weight:
416.52
Estimated delivery in United States, on Thursday 3 Feb 2022
CID1231538
CAS:354126-20-8
CID1231538 is a potent GPR35 antagonist.
Formula:
C26H22ClN3O3S2
Molecular weight:
524.05
Estimated delivery in United States, on Thursday 3 Feb 2022
Kisspeptin 234 acetate(1145998-81-7 free base)
kisspeptin receptor (KISS1, GPR54) antagonist; kisspeptin-10 analog. Inhibits kisspeptin-10 stimulation of inositol phosphate (IP) (IC50 …
Formula:
C65H82N18O15
Molecular weight:
1355.46
Estimated delivery in United States, on Thursday 3 Feb 2022
Urotensin II, mouse TFA (9047-55-6 free base)
Urotensin II, mouse TFA is an endogenous ligand for the orphan GPR14 or SENR. It …
Formula:
C78H101N18F3O21S2
Molecular weight:
1747.88
Estimated delivery in United States, on Thursday 3 Feb 2022
Urotensin II, mouse acetate (9047-55-6 free base)
Urotensin II, mouse acetate is an endogenous ligand for the orphan GPR14 or SENR. It …
Formula:
C78H104N18O21S2
Purity:
97.86%
Molecular weight:
1693.91
Estimated delivery in United States, on Thursday 3 Feb 2022
TUG-770
CAS:1402601-82-4
TUG-770 is a highly potent agonist of free fatty acid receptor 1 (FFA1/GPR40, EC50: 6 …
Formula:
C19H14FNO2
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
307.32
Estimated delivery in United States, on Thursday 3 Feb 2022
AMG 837 calcium hydrate
CAS:1259389-38-2
AMG 837 calcium hydrate is a potent GPR40 agonist(EC50: 13 nM) with highly selective over …
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
455.45
Estimated delivery in United States, on Thursday 3 Feb 2022
MK-7246
CAS:1218918-62-7
MK-7246 is a potent and specific CRTH2 antagonist (Ki: 2.5 nM).
Formula:
C21H21FN2O4S
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
416.47
Estimated delivery in United States, on Thursday 3 Feb 2022
