Glucocorticoid Receptor
The glucocorticoid receptor (GR) is a nuclear hormone receptor that mediates the effects of glucocorticoids, a class of steroid hormones involved in the regulation of metabolism, immune response, and stress. Glucocorticoid receptor agonists and antagonists are widely used in the treatment of inflammatory and autoimmune diseases, as well as in cancer therapy. GR modulators are also important tools for studying the physiological and pathological roles of glucocorticoids. At CymitQuimica, we provide a wide range of high-quality glucocorticoid receptor modulators to support your research in endocrinology, immunology, and hormone regulation.
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Budesonide
CAS:51333-22-3
Budesonide (Pulmicort), an anti-inflammatory corticosteroid, has shown the effective glucocorticoid activitie and few mineralocorticoid activities. …
Formula:
C25H34O6
Purity:
99.03% - 99.72%
Color and Shape:
Crystals Solid
Molecular weight:
430.53
Ref: TM-T0094
| 1ml | 54.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
GW-870086
CAS:827319-43-7
GW-870086 is an effective anti-inflammatory agent.
Formula:
C31H39F2NO6
Purity:
99.63%
Color and Shape:
Solid
Molecular weight:
559.64
Ref: TM-T15451
| 2mg | 34.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 113.00 € | ||
| 50mg | 203.00 € | ||
| 100mg | 301.00 € | ||
| 200mg | 435.00 € | ||
| 1mL*10mM (DMSO) | 62.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Mirodenafil
CAS:862189-95-5
Mirodenafil is a PDE-5 inhibitor developed for the treatment of erectile dysfunction.
Formula:
C26H37N5O5S
Purity:
99.89%
Color and Shape:
Solid
Molecular weight:
531.67
Ref: TM-T16079
| 5mg | 52.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 132.00 € | ||
| 50mg | 209.00 € | ||
| 100mg | 333.00 € | ||
| 500mg | 782.00 € | ||
| 1mL*10mM (DMSO) | 70.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Hydrocortisone
CAS:50-23-7
Hydrocortisone is a synthetic glucocorticoid that aids in metabolism, immunity, and inflammation control.
Formula:
C21H30O5
Purity:
98.4% - 99.95%
Color and Shape:
Plates From Alc Or Iso-Propyl Alc Solid
Molecular weight:
362.46
Ref: TM-T1614
| 50mg | 35.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Fluticasone (propionate)
CAS:80474-14-2
Fluticasone propionate (CCI-187881), derived from fluticasone used to remedy asthma and allergic rhinitis, is a …
Formula:
C25H31F3O5S
Purity:
100% - 98.98%
Color and Shape:
Crystalline Solid
Molecular weight:
500.57
Ref: TM-T0188
| 5mg | 49.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 123.00 € | ||
| 50mg | 185.00 € | ||
| 100mg | 269.00 € | ||
| 200mg | 335.00 € | ||
| 500mg | 552.00 € | ||
| 1mL*10mM (DMSO) | 83.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Medroxyprogesterone Acetate
CAS:71-58-9
Medroxyprogesterone Acetate (Farlutin) is a synthetic progestin that is derived from 17-hydroxyprogesterone. Farlutin is a …
Formula:
C24H34O4
Purity:
99.45%
Color and Shape:
White Powder
Molecular weight:
386.52
Ref: TM-T1261
| 200mg | 36.00 € | ||
| 500mg | 47.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Fluocinolone (Acetonide)
CAS:67-73-2
Fluocinolone Acetonide (Flucort-N) is a glucocorticoid derivative used topically in the treatment of various skin …
Formula:
C24H30F2O6
Purity:
99.42% - 99.66%
Color and Shape:
Crystals From Acetone & Hexane Solid
Molecular weight:
452.49
Ref: TM-T0367
| 1g | 62.00 € | ||
| 500mg | 41.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Megestrol acetate
CAS:595-33-5
Megestrol acetate (BDH1298) is an oral progestogen with anti-androgenic properties, used for endometrial and breast …
Formula:
C24H32O4
Purity:
99.72%
Color and Shape:
Crystalline Solid
Molecular weight:
384.51
Ref: TM-T1284
| 1g | 62.00 € | ||
| 500mg | 54.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Nimodipine
CAS:66085-59-4
Nimodipine (BAY-e 9736), a 1, 4-dihydropyridine calcium channel blocker, acts primarily on vascular smooth muscle …
Formula:
C21H26N2O7
Purity:
99.56% - 99.71%
Color and Shape:
Solid
Molecular weight:
418.44
Ref: TM-T0343
| 50mg | 52.00 € | ||
| 100mg | 57.00 € | ||
| 500mg | 83.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Dexamethasone acetate
CAS:1177-87-3
Dexamethasone acetate (NSC 39471) is a potent anti-inflammatory steroid, blocks NF-kB, and lacks salt-retention.
Formula:
C24H31FO6
Purity:
99.22% - 99.65%
Color and Shape:
White Or Almost White Crystalline Powder
Molecular weight:
434.5
Ref: TM-T0947
| 1g | 84.00 € | ||
| 500mg | 49.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Flumethasone
CAS:2135-17-3
Flumethasone (RS-2177) is a glucocorticoid receptor agonist, with anti-inflammatory, antipruritic and vasoconstrictive properties.
Formula:
C22H28F2O5
Purity:
99.91%
Color and Shape:
White Crystalline Powder
Molecular weight:
410.45
Ref: TM-T1124
| 50mg | 35.00 € | ||
| 100mg | 56.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Hydrocortisone acetate
CAS:50-03-3
Hydrocortisone acetate (Cortisol 21-acetate) is the synthetic acetate salt form of hydrocortisone, a corticosteroid with …
Formula:
C23H32O6
Purity:
99.58%
Color and Shape:
White To Off-White Crystalline Powder
Molecular weight:
404.5
Ref: TM-T1243
| 1g | 51.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Hydrocortisone 17-butyrate
CAS:13609-67-1
Hydrocortisone 17-butyrate (Cortisol 17-butyrate) is a glucocorticoid receptor agonist with antiinflammatory, antipruritic and vasoconstrictive effects.
Formula:
C25H36O6
Purity:
98% - 99.01%
Color and Shape:
Solid
Molecular weight:
432.55
Ref: TM-T0270
| 100mg | 34.00 € | ||
| 200mg | 50.00 € | ||
| 500mg | 82.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Esaxerenone
CAS:1632006-28-0
Esaxerenone (XL-550) is a highly potent and selective non-steroidal antagonist of the mineralocorticoid receptor.
Formula:
C22H21F3N2O4S
Purity:
99.68%
Color and Shape:
Solid
Molecular weight:
466.47
Ref: TM-T15246
| 1mg | 69.00 € | ||
| 5mg | 143.00 € | ||
| 10mg | 223.00 € | ||
| 25mg | 432.00 € | ||
| 50mg | 686.00 € | ||
| 100mg | 1,077.00 € | ||
| 500mg | 2,168.00 € | ||
| 1mL*10mM (DMSO) | 159.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Spironolactone
CAS:52-01-7
Spironolactone (SC9420) is an Aldosterone Antagonist. The mechanism of action of spironolactone is as an …
Formula:
C24H32O4S
Purity:
99.63%
Color and Shape:
White Powder
Molecular weight:
416.57
Ref: TM-T0476
| 50mg | 39.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Hydrocortisone Valerate
CAS:57524-89-7
Hydrocortisone Valerate (Westcort) has anti-inflammatory, antipruritic and vasoconstrictive properties.
Formula:
C26H38O6
Purity:
99.69%
Color and Shape:
Solid
Molecular weight:
446.58
Ref: TM-T0276
| 10mg | 34.00 € | ||
| 25mg | 67.00 € | ||
| 50mg | 93.00 € | ||
| 100mg | 171.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Dexamethasone Phosphate disodium
CAS:2392-39-4
Dexamethasone Phosphate disodium (EGP437. Dex-Phos) is a water-soluble form of the synthetic glucocorticoid dexamethasone.
Formula:
C22H28FNa2O8P
Purity:
99.88%
Color and Shape:
White To Off White Powder
Molecular weight:
516.4
Ref: TM-T0947L
| 50mg | 36.00 € | ||
| 100mg | 48.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Dexamethasone
CAS:50-02-2
Dexamethasone: a glucocorticoid agonist; modulates IL receptors; reduces inflammatory miRNA-155 exosomes in macrophage responses.
Formula:
C22H29FO5
Purity:
98% - 99.91%
Color and Shape:
Crystals From Ether (Ntp 1992)
Molecular weight:
392.46
Ref: TM-T1076
| 50mg | 34.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Loteprednol etabonate
CAS:82034-46-6
Loteprednol etabonate (Lotemax) is an ophthalmic analog of the corticosteroid prednisolone with anti-inflammatory activity.
Formula:
C24H31ClO7
Purity:
99.19%
Color and Shape:
Solid
Molecular weight:
466.95
Ref: TM-T0181
| 10mg | 46.00 € | ||
| 25mg | 86.00 € | ||
| 50mg | 151.00 € | ||
| 100mg | 237.00 € | ||
| 200mg | 296.00 € | ||
| 500mg | 492.00 € | ||
| 1mL*10mM (DMSO) | 45.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Halcinonide
CAS:3093-35-4
Halcinonide (Halciderm), a high-efficiency corticosteroid, is served as an anti-inflammatory agent used in topical preparations.
Formula:
C24H32ClFO5
Purity:
99.32% - 99.94%
Color and Shape:
Solid
Molecular weight:
454.96
Ref: TM-T0107
| 1g | 558.00 € | ||
| 10mg | 47.00 € | ||
| 25mg | 64.00 € | ||
| 50mg | 80.00 € | ||
| 100mg | 129.00 € | ||
| 200mg | 200.00 € | ||
| 500mg | 367.00 € | ||
| 1mL*10mM (DMSO) | 44.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
