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JAK
Tyrphostin AG 490
CAS:133550-30-8
Formula:
C17H14N2O3
Purity:
>98.0%(HPLC)(T)
Color and Shape:
Slightly Pale Yellow - Yellow Solid
Molecular weight:
294.31
Estimated delivery in United States, on Thursday 27 Jan 2022
WHI-P154
CAS:211555-04-3
Formula:
C16H14BrN3O3
Purity:
>98.0%(HPLC)
Color and Shape:
White to Yellow to Orange powder to crystal
Molecular weight:
376.21
Estimated delivery in United States, on Thursday 27 Jan 2022
AG490
CAS:133550-30-8
AG-490 (Tyrphostin AG 490) is an inhibitor of EGFR (IC50: 0.1 μM). It is 135-fold …
Formula:
C17H14N2O3
Purity:
98.60%
Color and Shape:
Yellow Solid
Molecular weight:
294.3
Estimated delivery in United States, on Monday 7 Feb 2022
BaricitinibPhosphate
CAS:1187595-84-1
Baricitinib phosphate is a selective orally bioavailable JAK1/JAK2 inhibitor.
Formula:
C16H20N7O6PS
Purity:
98.87%
Color and Shape:
solid
Molecular weight:
469.41
Estimated delivery in United States, on Monday 7 Feb 2022
AT9283
CAS:896466-04-9
AT9283 is an effective multi-targeted inhibitor of JAK2(IC50=1.2 nM) and JAK3(IC50=1.1 nM), Aurora A, Aurora …
Formula:
C19H23N7O2
Purity:
98.45%
Color and Shape:
solid
Molecular weight:
381.43
Estimated delivery in United States, on Monday 7 Feb 2022
Momelotinib
CAS:1056634-68-4
Momelotinib is an orally bioavailable small-molecule inhibitor of Janus kinases 1 and 2 (JAK1/2) with …
Formula:
C23H22N6O2
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
414.46
Estimated delivery in United States, on Monday 7 Feb 2022
Filgotinib
CAS:1206161-97-8
GLPG0634(filgotinib) is a selective JAK1 inhibitor. The IC50 values against JAK1, JAK2, JAK3, and TYK2 …
Formula:
C21H23N5O3S
Purity:
99.09%
Color and Shape:
solid
Molecular weight:
425.5
Estimated delivery in United States, on Monday 7 Feb 2022
Baricitinib
CAS:1187594-09-7
Baricitinib is an orally bioavailable inhibitor of Janus kinases 1 and 2 (JAK1/2), with potential …
Formula:
C16H17N7O2S
Purity:
99.00%
Color and Shape:
solid
Molecular weight:
371.42
Estimated delivery in United States, on Monday 7 Feb 2022
Cerdulatinib
CAS:1198300-79-6
Cerdulatinib is an novel oral dual Syk/JAK inhibitor.
Formula:
C20H27N7O3S
Purity:
98.74%
Color and Shape:
solid
Molecular weight:
445.54
Estimated delivery in United States, on Monday 7 Feb 2022
PP2
CAS:172889-27-9
PP2 is a effective inhibitor of Lck/Fyn (IC50:4/5 nM) , ~100-fold less potent to EGFR, …
Formula:
C15H16ClN5
Purity:
95.65%
Color and Shape:
solid
Molecular weight:
301.77
Estimated delivery in United States, on Monday 7 Feb 2022
WHI-P154
CAS:211555-04-3
WHI-P154 is a potent JAK3 inhibitor.
Formula:
C16H14BrN3O3
Purity:
98.03%
Color and Shape:
solid
Molecular weight:
376.2
Estimated delivery in United States, on Monday 7 Feb 2022
JAK2 Inhibitor V
CAS:195371-52-9
NSC 42834(JAK2 Inhibitor V, Z3) is a novel specific inhibitor of Jak2, inhibiting Jak2-V617F and …
Formula:
C23H24N2O
Purity:
99.15%
Color and Shape:
solid
Molecular weight:
344.45
Estimated delivery in United States, on Monday 7 Feb 2022
Solcitinib
CAS:1206163-45-2
Solcitinib (GSK2586184, GLPG0778) is a JAK1 inhibitor. Solcitinib may be potentially used for the treatment …
Formula:
C22H23N5O2
Purity:
99.68%
Color and Shape:
solid
Molecular weight:
389.18
Estimated delivery in United States, on Monday 7 Feb 2022
SHR0302
CAS:1445987-21-2
SHR0302 is a JAK inhibitor that binds JAK1 with stronger affinity than others (Selectivity for …
Formula:
C18H22N8O2S
Molecular weight:
414.48
Estimated delivery in United States, on Monday 7 Feb 2022
JDTic
CAS:361444-66-8
JDTic has a very long duration of action, with effects in animals seen for up …
Formula:
C28H39N3O3
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
465.63
Estimated delivery in United States, on Monday 7 Feb 2022
JBJ-02-112-05
JBJ-02-112-05 is a potent, mutant-selective, allosteric and orally active EGFR inhibitor with an IC50 of …
Formula:
C27H20N4O2S
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
464.54
Estimated delivery in United States, on Monday 7 Feb 2022
WP1066
CAS:857064-38-1
WP1066 is a inhibitor of JAK2 (IC50: 2.30 μM) and STAT3 (IC50: 2.43 μM) in …
Formula:
C17H14BrN3O
Purity:
99.07%
Color and Shape:
solid
Molecular weight:
356.22
Estimated delivery in United States, on Monday 7 Feb 2022
Pyridone 6
CAS:457081-03-7
Pyridone 6(CMP 6) is a potent and selective inhibitor of JAK1 (IC50=15 nM, murine JAK1), …
Formula:
C18H16FN3O
Purity:
98.70%
Color and Shape:
solid
Molecular weight:
309.34
Estimated delivery in United States, on Monday 7 Feb 2022
Oclacitinib maleate
CAS:1640292-55-2
Oclacitinib is a novel inhibitor of JAK family members with IC50 ranging from 10 to …
Formula:
C15H23N5O2S·C4H4O4
Purity:
99.17%
Color and Shape:
Solid
Molecular weight:
453.51
Estimated delivery in United States, on Monday 7 Feb 2022
JAK3-IN-7
CAS:1263774-57-7
JAK3-IN-7 is an effective and selective JAK3 inhibitor (IC50 <0.01 μM) extracted from patent WO2011013785A1.
Formula:
C17H20N6O
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
324.38
Estimated delivery in United States, on Monday 7 Feb 2022
WHI-P97 HCl 211555-05-4(free base)
WHI-P97 HCl is a potent and selective JAK-3 inhibitor. WHI-P97 had an estimated Ki value …
Formula:
C16H14Br2ClN3O3
Molecular weight:
491.56
Estimated delivery in United States, on Monday 7 Feb 2022
Cucurbitacin I
CAS:2222-07-3
Cucurbitacin I, a natural compound, is a selective inhibitor of JAK2/STAT3 with anti-cancer activity.
Formula:
C30H42O7
Purity:
96.69%
Color and Shape:
solid
Molecular weight:
514.65
Estimated delivery in United States, on Monday 7 Feb 2022
AZ-3
CAS:2228908-91-4
AZ-3 is a potent and selective JAK1 inhibitor (IC50: 34 nM).
Formula:
C20H28FN7
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
385.48
Estimated delivery in United States, on Monday 7 Feb 2022
Oclacitinib
CAS:1208319-26-9
Oclacitinib(PF03394197) is a potent and selective JAKs inhibitor with IC50 of 10-99 nM; not inhibit …
Formula:
C15H23N5O2S
Purity:
97.71%
Color and Shape:
White To Off-White Solid
Molecular weight:
337.44
Estimated delivery in United States, on Monday 7 Feb 2022
JAK3 covalent inhibitor-1
CAS:2300106-50-5
JAK3 covalent inhibitor-1 is a potent and selective janus kinase 3 (JAK3) covalent inhibitor with …
Formula:
C22H17FN6O2S
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
448.47
Estimated delivery in United States, on Monday 7 Feb 2022
Gusacitinib
CAS:1425381-60-7
Gusacitinib (ASN-002) is spleen tyrosine kinase (SYK) and janus kinase (JAK) inhibitor (IC50: 5-46 nM).
Formula:
C24H28N8O2
Purity:
99.58%
Color and Shape:
Solid
Molecular weight:
460.53
Estimated delivery in United States, on Monday 7 Feb 2022
AZD4205
CAS:2091134-68-6
AZD4205 is a selective JAK1 inhibitor (IC50: 73 nM) and weakly inhibits JAK2/JAK3 (IC50: >14.7, …
Formula:
C25H31N9O2
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
489.57
Estimated delivery in United States, on Monday 7 Feb 2022
Curcumol
CAS:4871-97-0
Curcumol, a pure monomer isolated extracted from Rhizoma Curcumaeis, has antitumor activities.
Formula:
C15H24O2
Purity:
99.87%
Color and Shape:
solid
Molecular weight:
236.35
Estimated delivery in United States, on Monday 7 Feb 2022
CEP33779
CAS:1257704-57-6
CEP-33779 is a novel and selective inhibitor of JAK2 with an IC50 of 1.8±0.6 nM.
Formula:
C24H26N6O2S
Purity:
97.00%
Color and Shape:
solid
Molecular weight:
462.57
Estimated delivery in United States, on Monday 7 Feb 2022
MM-589
CAS:2097887-20-0
MM-589 is a potent WD repeat domain 5 (WDR5) inhibitor and mixed lineage leukemia (MLL) …
Formula:
C28H44N8O5
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
572.7
Estimated delivery in United States, on Monday 7 Feb 2022
Ilginatinib maleate
CAS:1354799-87-3
Ilginatinib maleate is a highly active and orally bioavailable inhibitor of JAK2.
Formula:
C25H24FN7O4
Purity:
99.68%
Color and Shape:
Solid
Molecular weight:
505.5
Estimated delivery in United States, on Monday 7 Feb 2022
JAK1-IN-4
CAS:2091134-35-7
JAK1-IN-4 is a selective JAK1 inhibitor (IC50s: 85 nM, 12.8 μM and >30 μM for …
Formula:
C26H32FN9O2
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
521.59
Estimated delivery in United States, on Monday 7 Feb 2022
Tofacitinib
CAS:477600-75-2
Tofacitinib is an oral, small molecule inhibitor of Janus kinases that is used to treat …
Formula:
C16H20N6O
Purity:
100.00%
Color and Shape:
solid
Molecular weight:
312.37
Estimated delivery in United States, on Monday 7 Feb 2022
Ilginatinib
CAS:1239358-86-1
Ilginatinib is a highly active and orally bioavailable inhibitor of JAK2.
Formula:
C21H20FN7
Purity:
99.43%
Color and Shape:
Solid
Molecular weight:
389.43
Estimated delivery in United States, on Monday 7 Feb 2022
Delgocitinib
CAS:1263774-59-9
Delgocitinib is a novel and specific inhibitor of JAK (IC50s: 2.8, 2.6, 13, and 58 …
Formula:
C16H18N6O
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
310.35
Estimated delivery in United States, on Monday 7 Feb 2022
AZD1480
CAS:935666-88-9
AZD1480 is a novel ATP-competitive JAK2 inhibitor (IC50: 0.26 nM), selectivity act against Tyk2 and …
Formula:
C14H14ClFN8
Purity:
97.50%
Color and Shape:
solid
Molecular weight:
348.77
Estimated delivery in United States, on Monday 7 Feb 2022
JAK2-IN-4
CAS:1438284-00-4
JAK2-IN-4 is a selective JAK2/JAK3 inhibitor, with IC50 values of 0.7 nM and 23.2 nM …
Formula:
C23H27N5O4S
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
469.56
Estimated delivery in United States, on Monday 7 Feb 2022
JAK3-IN-6
CAS:1443235-95-7
JAK3-IN-6 is irreversible Janus Associated Kinase 3 (JAK3) inhibitor, with an IC50 of 0.15 nM
Formula:
C19H18N4O3
Purity:
97.34%
Color and Shape:
Solid
Molecular weight:
350.37
Estimated delivery in United States, on Monday 7 Feb 2022
WDR5-0103
CAS:890190-22-4
WDR5-0103 is an effective and specific WD repeat-containing protein 5 (WDR5) antagonist (Kd: 450 nM).
Formula:
C21H25N3O4
Purity:
99.61%
Color and Shape:
solid
Molecular weight:
383.44
Estimated delivery in United States, on Monday 7 Feb 2022
Ilginatinib hydrochloride
CAS:1239358-85-0
Ilginatinib hydrochloride is a highly active and orally bioavailable inhibitor of JAK2.
Formula:
C21H21ClFN7
Purity:
99.55%
Color and Shape:
Solid
Molecular weight:
425.89
Estimated delivery in United States, on Monday 7 Feb 2022
JAK 3 inhibitor IV
CAS:58753-54-1
JAK 3 inhibitor IV is a JAK1/3 inhibitor with pIC50 of 4.4/7.1, almost no activity …
Formula:
C16H19NO
Molecular weight:
241.33
Estimated delivery in United States, on Monday 7 Feb 2022
Jaspamycin
CAS:22242-96-2
Jaspamycin (7-CN-7-C-Ino) does not bind with purified human PKARI. Anti-parasite activity. Jaspamycin (7-CN-7-C-Ino) is a …
Formula:
C12H12N4O5
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
292.25
Estimated delivery in United States, on Monday 7 Feb 2022
Momelotinib sulfate
CAS:1056636-06-6
Momelotinib sulfate is an ATP-competitive JAK1/JAK2 inhibitor (IC50: 11 nM/18 nM). It has 10-fold selectivity …
Formula:
C23H26N6O10S2
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
610.62
Estimated delivery in United States, on Monday 7 Feb 2022
TAK901
CAS:934541-31-8
TAK-901 has been used in trials studying the treatment of Lymphoma, Myelofibrosis, Multiple Myeloma, Myeloid …
Formula:
C28H32N4O3S
Purity:
98.18%
Color and Shape:
solid
Molecular weight:
504.64
Estimated delivery in United States, on Monday 7 Feb 2022
FM381
CAS:2226521-65-7
FM381 is a potent covalent reversible inhibitor of JAK3. FM-381 has an IC50 of 127 …
Formula:
C24H24N6O2
Purity:
98.27%
Color and Shape:
Solid
Molecular weight:
428.49
Estimated delivery in United States, on Monday 7 Feb 2022
JAK-IN-5
CAS:2096999-92-5
JAK-IN-5 is an inhibitor of JAK.
Formula:
C27H31FN6O
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
474.57
Estimated delivery in United States, on Monday 7 Feb 2022
OICR9429
CAS:1801787-56-3
OICR-9429 is a potent antagonist of the interaction that WDR5 effect with peptide regions of …
Formula:
C29H32F3N5O3
Purity:
99.93%
Color and Shape:
Solid
Molecular weight:
555.59
Estimated delivery in United States, on Monday 7 Feb 2022
Tofacitinib Citrate
CAS:540737-29-9
Tofacitinib citrate is a a potent, cell-permeable inhibitor of JAK1/2/3 (IC50s: 1/20/112 nM).
Formula:
C22H28N6O8
Purity:
99.47%
Color and Shape:
solid
Molecular weight:
504.49
Estimated delivery in United States, on Monday 7 Feb 2022
Icaritin
CAS:118525-40-9
Icaritin has hormone regulation activity and cardiovascular function improvement activity. Icaritin has anticancer activity, can …
Formula:
C21H20O6
Purity:
97.69%
Color and Shape:
solid
Molecular weight:
368.38
Estimated delivery in United States, on Monday 7 Feb 2022
JBJ-04-125-02
CAS:2060610-53-7
JBJ-04-125-02 can inhibit cancer cell proliferation and EGFRL858R/T790M/C797S signaling. JBJ-04-125-02 has anti-tumor activities. JBJ-04-125-02 is …
Formula:
C29H26FN5O3S
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
543.61
Estimated delivery in United States, on Monday 7 Feb 2022
S-Ruxolitinib
CAS:941685-37-6
Ruxolitinib S enantiomer is the S-enantiomer of Ruxolitinib. Ruxolitinib is the first potent, selective JAK1/2 …
Formula:
C17H18N6
Purity:
99.79%
Molecular weight:
306.37
Estimated delivery in United States, on Monday 7 Feb 2022
MM-589 TFA
CAS:2097887-21-1
MM-589 TFA is a potent WD repeat domain 5 (WDR5)inhibitor and mixed lineage leukemia (MLL) …
Formula:
C30H45F3N8O7
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
686.72
Estimated delivery in United States, on Monday 7 Feb 2022
Upadacitinib
CAS:1310726-60-3
Upadacitinib (ABT-494) is a selective Janus kinase (JAK) 1 inhibitor, which is being studied for …
Formula:
C17H19F3N6O
Purity:
99.89%
Color and Shape:
solid
Molecular weight:
380.37
Estimated delivery in United States, on Monday 7 Feb 2022
Ruxolitinib (INCB-18424) phosphate
CAS:1092939-17-7
Ruxolitinib phosphate(INCB018424 phosphate) is the first potent, selective, JAK1/2 inhibitor to enter the clinic with …
Formula:
C17H21N6O4P
Purity:
99.72%
Color and Shape:
solid
Molecular weight:
404.36
Estimated delivery in United States, on Monday 7 Feb 2022
AZ 960
CAS:905586-69-8
AZ 960 is an effective ATP competitive JAK2 inhibitor (IC50/Ki: <3 nM and0.45 nM).
Formula:
C18H16F2N6
Purity:
96.02%
Color and Shape:
solid
Molecular weight:
354.36
Estimated delivery in United States, on Monday 7 Feb 2022
Ruxolitinib
CAS:941678-49-5
Ruxolitinib is a potent and selective JAK1/2 inhibitor (IC50: 3.3/2.8 nM) and is relatively less …
Formula:
C17H18N6
Purity:
99.42%
Color and Shape:
solid
Molecular weight:
306.37
Estimated delivery in United States, on Monday 7 Feb 2022
WHI-P131
CAS:202475-60-3
Janex-1 is a cell-permeable, reversible, effective, ATP-competitive, and selective inhibitor of JAK3 (IC50: 78 μM); …
Formula:
C16H15N3O3
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
297.31
Estimated delivery in United States, on Monday 7 Feb 2022
Fedratinib
CAS:936091-26-8
Fedratinib (TG101348) is an ATP-competitive inhibitor of JAK2 (IC50: 3 nM) with significantly less potent …
Formula:
C27H36N6O3S
Purity:
99.00%
Color and Shape:
solid
Molecular weight:
524.68
Estimated delivery in United States, on Monday 7 Feb 2022
BMS-986165
CAS:1609392-27-9
BMS-986165 inhibits IL-12/23 and type I IFN pathways[1][2]. BMS-986165 is a highly selective, orally bioavailable …
Formula:
C20H19D3N8O3
Purity:
100.00%
Color and Shape:
Solid
Molecular weight:
425.46
Estimated delivery in United States, on Monday 7 Feb 2022
Itacitinib
CAS:1334298-90-6
Itacitinib is an orally bioavailable inhibitor of Janus-associated kinase 1 (JAK1) with potential antineoplastic activity.
Formula:
C26H23F4N9O
Purity:
97.57%
Color and Shape:
solid
Molecular weight:
553.53
Estimated delivery in United States, on Monday 7 Feb 2022
FLLL32
CAS:1226895-15-3
FLLL32 is an effective JAK2/STAT3 inhibitor (IC50 of <5 μM).
Formula:
C28H32O6
Purity:
96.39%
Color and Shape:
solid
Molecular weight:
464.55
Estimated delivery in United States, on Monday 7 Feb 2022
PF-06700841 (P-Tosylate)
CAS:2140301-96-6
PF-06700841 P-Tosylate is a potent dual inhibitor of Janus kinase 1 (JAK1) and TYK2 (IC50s …
Formula:
C25H29F2N7O4S
Purity:
99.82%
Color and Shape:
Solid
Molecular weight:
561.60
Estimated delivery in United States, on Monday 7 Feb 2022
Abrocitinib
CAS:1622902-68-4
Abrocitinib (PF-04965842) is a potent, specific and orally-active JAK1 inhibitor (IC50s: 29/803 nM for JAK1/2).
Formula:
C14H20N5O2S
Purity:
99.91%
Color and Shape:
Solid，White To Beige
Molecular weight:
323.41
Estimated delivery in United States, on Monday 7 Feb 2022
Peficitinib
CAS:944118-01-8
Peficitinib (ASP015K, JNJ-54781532) is an orally bioavailable JAK inhibitor. Phase 3.
Formula:
C18H22N4O2
Purity:
98.0%
Molecular weight:
326.39
Estimated delivery in United States, on Monday 7 Feb 2022
ZM 39923 HCl
CAS:1021868-92-7
ZM 39923 HCl is an JAK1/3 inhibitor with pIC50 of 4.4/7.1, almost no activity to …
Formula:
C23H25NO·HCl
Purity:
98.05%
Color and Shape:
solid
Molecular weight:
367.91
Estimated delivery in United States, on Monday 7 Feb 2022
SC99
CAS:882290-02-0
SC99 is a selective inhibitor of JAK2-STAT3 activation. SC99 downregulates the expression of STAT3-modulated genes.SC99 …
Formula:
C15H8Cl2FN3O
Molecular weight:
336.15
Estimated delivery in United States, on Monday 7 Feb 2022
PF-06651600
CAS:1792180-81-4
PF-06651600 is a potent JAK3-selective inhibitor (IC50: 33.1 nM).
Formula:
C15H19N5O
Purity:
99.10%
Color and Shape:
Solid
Molecular weight:
285.34
Estimated delivery in United States, on Monday 7 Feb 2022
ITK inhibitor 2
CAS:1309784-09-5
ITK inhibitor 2 is a interleukin-2-inducible T-cell kinase (ITK) inhibitor , with an IC50 of …
Formula:
C25H33N5O2
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
435.56
Estimated delivery in United States, on Monday 7 Feb 2022
JAK-IN-11
CAS:916742-11-5
JAK-IN-11 is a potent and selective inhibitor of JAK, has the potential for the skin …
Formula:
C23H22FN5O4S
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
483.52
Estimated delivery in United States, on Monday 7 Feb 2022
SAR20347
CAS:1450881-55-6
SAR-20347 is an inhibitor of TYK2, JAK1/2/3 (IC50: 0.6/23/26/41 nM).
Formula:
C21H18ClFN4O4
Purity:
99.35%
Color and Shape:
Solid
Molecular weight:
444.85
Estimated delivery in United States, on Monday 7 Feb 2022
Momelotinib Mesylate
CAS:1056636-07-7
Momelotinib Mesylate is an ATP-competitive JAK1/JAK2 inhibitor (IC50: 11 nM/18 nM). It has 10-fold selectivity …
Formula:
C24H26N6O5S
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
510.57
Estimated delivery in United States, on Monday 7 Feb 2022
JDTic dihydrochloride
CAS:785835-79-2
JDTic is a potent antagonist of kappa-opioid receptors (KOR), blocking the -agonist U50, 488-induced antinociception.
Formula:
C28H41Cl2N3O3
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
538.55
Estimated delivery in United States, on Monday 7 Feb 2022
Decernotinib
CAS:944842-54-0
Decernotinib(VX-509; VRT-831509) is a potent and selective Janus kinase 3 (JAK3) inhibitor with Ki of …
Formula:
C18H19F3N6O
Purity:
99.45%
Color and Shape:
solid
Molecular weight:
392.38
Estimated delivery in United States, on Monday 7 Feb 2022
BD750
CAS:892686-59-8
BD750 is an effective immunosuppressant and a JAK3/STAT5 inhibitor, inhibits IL-2-induced JAK3/STAT5-dependent T cell proliferation(IC50 …
Formula:
C14H13N3OS
Purity:
99.76%
Color and Shape:
Solid
Molecular weight:
271.34
Estimated delivery in United States, on Monday 7 Feb 2022
Fedratinib hydrochloride hydrate
CAS:1374744-69-0
Fedratinib hydrochloride hydrate is a potent, selective, ATP-competitive and orally active JAK2 inhibitor.
Formula:
C27H40Cl2N6O4S
Purity:
98.96%
Molecular weight:
615.61
Estimated delivery in United States, on Monday 7 Feb 2022
NVP-BSK805
CAS:1092499-93-8
NVP-BSK805 is an ATP-competitive JAK2 inhibitor.
Formula:
C27H28F2N6O
Purity:
98.75%
Color and Shape:
solid
Molecular weight:
490.54
Estimated delivery in United States, on Monday 7 Feb 2022
JAK2 inhibitor G5-7
CAS:939681-36-4
JAK2 inhibitor G5-7 is an orally active JAK2 inhibitor, selectively inhibits JAK2mediated phosphorylation and activation …
Formula:
C24H23F2NO3
Molecular weight:
411.4
Estimated delivery in United States, on Monday 7 Feb 2022
CHZ868
CAS:1895895-38-1
CHZ868 is a type II JAK2 inhibitor (IC50: 0.17 μM in EPOR JAK2 WT Ba/F3 …
Formula:
C22H19F2N5O2
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
423.42
Estimated delivery in United States, on Monday 7 Feb 2022
Ganoderic acid B
CAS:81907-61-1
Ganoderic acid B is a chemical marker in quality control of G. lucidum and related …
Formula:
C30H44O7
Purity:
98.00%
Color and Shape:
solid
Molecular weight:
516.67
Estimated delivery in United States, on Monday 7 Feb 2022
WDR5-0103 hydrochloride[890190-22-4(free base)]
WDR5-0103 is an effective and specific WD repeat-containing protein 5 (WDR5) antagonist (Kd: 450 nM).
Formula:
C21H26ClN3O4
Purity:
99.81%
Color and Shape:
solid
Molecular weight:
419.9
Estimated delivery in United States, on Monday 7 Feb 2022
PF-06700841
CAS:1883299-62-4
PF-06700841 is a potent dual JAK1/TYK2 inhibitor (IC50s: 17 nM/23 nM). It also inhibits JAK2/3 …
Formula:
C18H21F2N7O
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
389.4
Estimated delivery in United States, on Monday 7 Feb 2022
GLPG0634 analogue
CAS:1206101-20-3
GLPG0634 (analog) is a specific JAK1 inhibitor with IC50 of 10/28/810/116 nM for JAK1/2/3 and …
Formula:
C21H23N5O3S
Purity:
100.00%
Color and Shape:
solid
Molecular weight:
425.5
Estimated delivery in United States, on Monday 7 Feb 2022
WHI-P97
CAS:211555-05-4
WHI-P97 is a rationally designed potent inhibitor of JAK-3. IC50 value: Target: JAK3 Treatment of …
Formula:
C16H13Br2N3O3
Purity:
99.02%
Color and Shape:
solid
Molecular weight:
455.1
Estimated delivery in United States, on Monday 7 Feb 2022
WHI-P258
CAS:21561-09-1
WHI-P258 is a dimethoxyquinazoline inhibitor of JAK3. This compound binds JAK3 weakly and may be …
Formula:
C16H15N3O2
Purity:
99.59%
Color and Shape:
solid
Molecular weight:
281.31
Estimated delivery in United States, on Monday 7 Feb 2022
