
Calcium Channel
Calcium channels are membrane proteins that regulate the flow of calcium ions into and out of cells, which is essential for various cellular functions, including muscle contraction, neurotransmitter release, and gene expression. Dysregulation of calcium channel activity is associated with conditions such as hypertension, cardiac arrhythmias, and neurological disorders. At CymitQuimica, we provide a wide selection of calcium channel modulators to support your research in cardiovascular health, neurobiology, and signal transduction.
Found 493 products of "Calcium Channel"
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Cis-22a
CAS:<p>Cis-22a: selective TRPV6 inhibitor (IC50=0.32μM), halts T47D breast cancer cell growth.</p>Formula:C24H30F3N3O2Purity:99.07%Color and Shape:SolidMolecular weight:449.51EMD57033
CAS:<p>EMD57033 activates cardiac troponin C, enhances Ca2+ sensitivity to boost heart contraction.</p>Formula:C22H23N3O4SPurity:99.72% - >99.99%Color and Shape:SolidMolecular weight:425.5Reldesemtiv
CAS:<p>Reldesemtiv (CK-2127107) boosts exercise capacity, targeting fast muscle troponin, EC50 3.4 μM.</p>Formula:C19H18F2N6OPurity:97.27%Color and Shape:SolidMolecular weight:384.38Calcium channel-modulator-1
CAS:<p>Calcium channel-modulator-1 is a calcium channel-modulator (IC50:0.8 μM) with specialisation to block aortic constriction.</p>Formula:C26H24Cl2N2O7SPurity:99.95%Color and Shape:SolidMolecular weight:579.45AY 77
CAS:<p>AY 77: Potent, selective PAR2 agonist, favors Ca2+ (ec50=40nM) & ERK1/2 (ec50=2μM), boosts breast cancer cell migration.</p>Formula:C21H32N4O4Purity:99.7%Color and Shape:SolidMolecular weight:404.5Fluspirilene
CAS:<p>Fluspirilene is a long-acting antipsychotic for schizophrenia, inhibiting L-type calcium channels (IC50: 0.03 μM).</p>Formula:C29H31F2N3OPurity:99.59%Color and Shape:SolidMolecular weight:475.57Bupivacaine hydrochloride monohydrate
CAS:<p>Bupivacaine hydrochloride monohydrate is an NMDA receptor inhibitor that inhibits SCN5A channels and is commonly used in the study of chronic pain.</p>Formula:C18H31ClN2O2Purity:99.91%Color and Shape:SolidMolecular weight:342.9SR 33805 oxalate
CAS:<p>Ca2+ channel antagonist</p>Formula:C34H42N2O9SPurity:98%Color and Shape:SolidMolecular weight:654.77IAA65
CAS:<p>IAA65 is a potent inhibitor of T-type calcium channels, exhibiting an IC50 value of 18.9 μM, and holds potential for use in epilepsy research [1].</p>Formula:C16H13F6NO2Color and Shape:SolidMolecular weight:365.27CCR4 antagonist 2
CAS:<p>CCR4 antagonist 2 (Compound 31) is a novel potent, orally bioavailable small molecule antagonists of CC chemokine receptor 4 (CCR4) that inhibits Treg</p>Formula:C26H28Cl2N6OPurity:98%Color and Shape:SolidMolecular weight:511.45Cav 2.2/3.2 blocker 1
<p>Compound 9e is a Cav 2.2/3.2 blocker; IC50: 1.22 μM & 80 μM, respectively; penetrates CNS.</p>Formula:C28H30N2O3Color and Shape:SolidMolecular weight:442.55(rel)-Mirogabalin
CAS:<p>(rel)-Mirogabalin ((rel)-DS5565) is an inhibitor of voltage-dependent calcium channels, specifically targeting the α2δ-1 subunit.</p>Formula:C12H19NO2Color and Shape:SolidMolecular weight:209.28NNC 55-0396
CAS:<p>NNC 55-0396: Selective T-type calcium channel blocker, IC50 6.8 μM, inhibits human ovarian cancer cell growth.</p>Formula:C30H40Cl2FN3O2Purity:99.00%Color and Shape:SolidMolecular weight:564.56SB-423557
CAS:<p>SB-423557 is an orally active antagonist of calcium-sensing receptor (CaR) with IC50 of 520 nM</p>Formula:C28H36N2O4Purity:98%Color and Shape:SolidMolecular weight:464.60Mibefradil
CAS:<p>Mibefradil is a calcium channel blocker with moderate selectivity for T-type Ca2+ channels (IC50s: 2.7 μM and 18.6 μM for T-type and L-type currents).</p>Formula:C29H38FN3O3Purity:98%Color and Shape:SolidMolecular weight:495.63Sesamodil
CAS:<p>Sesamodil (SD 3211) is a novel calcium antagonist that can be used to study hypertension.</p>Formula:C29H32N2O6SPurity:98.58% - 99.01%Color and Shape:SolidMolecular weight:536.64Cav 3.2 inhibitor 1
<p>Cav 3.2 inhibitor 1 targets T-type calcium channels, weakly binds D2 receptors, and aids physical and visceral pain research.</p>Formula:C32H39N3OColor and Shape:SolidMolecular weight:481.67MP-010
CAS:<p>MP-010 is an FKBP12 ligand that regulates cytosolic calcium by stabilizing RyR channel activity. It facilitates functional improvement in SOD1G93A mice with amyotrophic lateral sclerosis (ALS), evidenced by enhanced motor coordination, increased integrity of neuromuscular junctions, and significantly higher spinal motor neuron survival rates. MP-010 is applicable for research in the field of neurological disorders.</p>Formula:C14H20N4O2SColor and Shape:SolidMolecular weight:308.399Cav 3.2 inhibitor 3
<p>Cav 3.2 inhibitor 3 is a potent inhibitor of the Cav3.2 T-type Ca2+channel (IC50: 0.1534 μM) and has a low binding affinity for D2 receptors.</p>Formula:C32H37N3O2Color and Shape:SolidMolecular weight:495.66PD-217014
CAS:<p>PD-217014 is an α2δ ligand that exhibits visceral analgesic activity and can suppress visceral hypersensitivity. Its antihyperalgesic effects are dose-dependent.</p>Formula:C10H17NO2Color and Shape:SolidMolecular weight:183.25

