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Metabolism

Metabolism

Metabolism inhibitors are compounds that interfere with metabolic pathways, altering the production and utilization of energy within cells. These inhibitors are used to study the regulation of metabolism, the role of metabolic pathways in diseases like cancer and diabetes, and to develop new therapeutic strategies. Metabolism inhibitors can target various enzymes and processes involved in glycolysis, fatty acid oxidation, and other metabolic functions. At CymitQuimica, we offer a wide range of high-quality metabolism inhibitors to support your research in biochemistry, metabolic disorders, and drug development.

Subcategories of "Metabolism"

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Found 8597 products of "Metabolism"

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  • EMD638683 R-Form

    CAS:
    <p>EMD638683 is a highly selective SGK1 inhibitor with IC50 of 3 μM. EMD638683 R-Form is the R-form of EMD638683.</p>
    Formula:C18H18F2N2O4
    Color and Shape:Solid
    Molecular weight:364.34
  • L791943

    CAS:
    <p>L791943 is a selective, potent) inhibitor of Phosphodiesterase-4 (PDE4,IC50 of 4.2 nM).</p>
    Formula:C24H17F10NO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:573.38
  • RB 101

    CAS:
    <p>RB 101 suppresses enkephalinase and aminopeptidases; biologically cleaved at disulfide to produce inhibitors of both aminopeptidase N and neutral endopeptidase.</p>
    Formula:C31H38N2O3S3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:582.84
  • CL4H6

    CAS:
    <p>CL4H6, a pH-sensitive cationic lipid, serves as the primary constituent of lipid nanoparticles (LNPs). These LNPs are instrumental in targeting and delivering siRNA, leading to a potent gene-silencing response [1] [2].</p>
    Formula:C59H113NO5
    Color and Shape:Solid
    Molecular weight:916.53
  • Quizalofop

    CAS:
    <p>Quizalofop (Xylafop) is a reagent of biochemical.</p>
    Formula:C17H13ClN2O4
    Purity:97.14%
    Color and Shape:Solid
    Molecular weight:344.75
  • WAY-297848

    CAS:
    <p>WAY-297848 is a novel glucokinase activator for the prevention or treatment of hyperglycemia, diabetes mellitus, obesity, dyslipidemia, and metabolic syndrome.</p>
    Formula:C13H13ClN2O2S
    Purity:98.19%
    Color and Shape:Solid
    Molecular weight:296.77
  • Fluspirilene

    CAS:
    <p>Fluspirilene is a long-acting antipsychotic for schizophrenia, inhibiting L-type calcium channels (IC50: 0.03 μM).</p>
    Formula:C29H31F2N3O
    Purity:99.59%
    Color and Shape:Solid
    Molecular weight:475.57
  • RS 8359

    CAS:
    <p>RS 8359 is a selective MAO-A reversible inhibitor with a 2200:1 A:B ratio, exhibiting antidepressant effects.</p>
    Formula:C14H12N4O
    Purity:99.3%
    Color and Shape:Solid
    Molecular weight:252.27
  • NPAS3-IN-1

    CAS:
    <p>NPAS3-IN-1 is an NPAS3-ARNT heterodimerization inhibitor that regulates NPAS3 transcription by modulating the heterodimerization of NPAS3 with ARNT.</p>
    Formula:C10H5N3O2S3
    Purity:99.56%
    Color and Shape:Solid
    Molecular weight:295.36
  • OGT 2115

    CAS:
    <p>OGT 2115 blocks heparanase (IC50=0.4µM), cleaving heparan sulfate; antiangiogenic (IC50=1µM).</p>
    Formula:C24H16BrFN2O4
    Purity:97.17%
    Color and Shape:Solid
    Molecular weight:495.3
  • ER 50891

    CAS:
    <p>ER-50891 is a potent RARα antagonist, countering retinoic acid inhibition and aiding BMP2-induced osteoblast differentiation.</p>
    Formula:C29H24N2O2
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:432.51
  • Inolitazone

    CAS:
    <p>Inolitazone (RS5444) a high-affinity PPARγ agonist. Inolitazone exhibits IC50 for growth inhibition is ~0.8 nM in vitro.</p>
    Formula:C27H26N4O4S
    Purity:99.41% - 99.53%
    Color and Shape:Solid
    Molecular weight:502.58
  • Enpp-1-IN-16

    CAS:
    <p>Enpp-1-IN-16 is an ENPP1 inhibitor, yo anti-cancer activity.Enpp-1-IN-16 can be used to study insulin resistance and chondrocalcinosis.</p>
    Formula:C23H32N4O4
    Purity:99.87%
    Color and Shape:Solid
    Molecular weight:428.52
  • Mitiperstat

    CAS:
    <p>Mitiperstat, a strong MPO inhibitor, helps prevent heart failure and coronary artery disease.</p>
    Formula:C15H15ClN4OS
    Purity:98.36%
    Color and Shape:Solid
    Molecular weight:334.82
  • WAY-620147

    CAS:
    <p>WAY-620147 inhibits Monoamine Oxidase and can be used for the study of neurological disorders.</p>
    Formula:C12H16BrN3O2
    Purity:99.55%
    Color and Shape:Solid
    Molecular weight:314.18
  • h-NTPDase-IN-2

    CAS:
    <p>h-NTPDase-IN-2 is a broad-spectrum NTPDase inhibitor that inhibits multiple h-NTPDas isoforms.</p>
    Formula:C19H16N4S
    Purity:99.58%
    Color and Shape:Solid
    Molecular weight:332.42
  • CCT365623

    CAS:
    <p>CCT365623: oral Lysyl Oxidase inhibitor, potent, selective, good pharmacokinetics, anti-metastatic.</p>
    Formula:C18H17NO4S3
    Purity:97.299% - 99.49%
    Color and Shape:Solid
    Molecular weight:407.53
  • 7-BIA

    CAS:
    <p>7-BIA is a receptor-type protein tyrosine phosphatase D (PTPRD) inhibitor with anti-addictive properties and can be used in the study of neuropathic pain.</p>
    Formula:C15H18O6
    Purity:≥98% - ≥98%
    Color and Shape:Solid
    Molecular weight:294.3
  • TPN171

    CAS:
    <p>TPN171 is potent PDE5 inhibitor with subnanomolar potency for PDE5 and good selectivity over PDE6, which has the potential for the treatment of pulmonary</p>
    Formula:C24H35N5O3
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:441.57
  • Calcium channel-modulator-1

    CAS:
    <p>Calcium channel-modulator-1 is a calcium channel-modulator (IC50:0.8 μM) with specialisation to block aortic constriction.</p>
    Formula:C26H24Cl2N2O7S
    Purity:99.95%
    Color and Shape:Solid
    Molecular weight:579.45
  • Ecopladib

    CAS:
    <p>Ecopladib inhibits cPLA2α with IC50 of 0.15 μM (micelles) &amp; 0.11 μM (rat blood).</p>
    Formula:C39H33Cl3N2O5S
    Purity:95.15%
    Color and Shape:Solid
    Molecular weight:748.11
  • Cis-22a

    CAS:
    <p>Cis-22a: selective TRPV6 inhibitor (IC50=0.32μM), halts T47D breast cancer cell growth.</p>
    Formula:C24H30F3N3O2
    Purity:99.07%
    Color and Shape:Solid
    Molecular weight:449.51
  • Rilapladib

    CAS:
    <p>Rilapladib (SB 659032) is a selective inhibitor of Lipoprotein-Associated Phospholipase A2(Lp-PLA2, IC50 = 230 pM) and an antagonist of the platelet activating</p>
    Formula:C40H38F5N3O3S
    Purity:99.92%
    Color and Shape:Solid
    Molecular weight:735.8
  • 4A3-SC8

    CAS:
    <p>4A3-SC8 is a modular, degradable dendrimer facilitating the extension of survival in aggressive liver cancer models through the delivery of small RNAs [1].</p>
    Formula:C75H139N3O16S4
    Purity:99.87%
    Color and Shape:Solid
    Molecular weight:1467.18
  • HIF-2α agonist 2

    CAS:
    <p>HIF-2α agonist 2 is an HIF-2α agonist with an EC50 value of 1.68 μM for HIF-2α.</p>
    Formula:C13H8Br2N2O2S
    Purity:98.87%
    Color and Shape:Soild
    Molecular weight:416.09
  • ALDH2 modulator 1

    CAS:
    <p>ALDH2 modulator 1 is a potent and orally active modulator of acetaldehyde dehydrogenase-2 (ALDH2), which reduces blood alcohol levels in mice.</p>
    Formula:C18H18ClFN2O3
    Purity:99.68%
    Color and Shape:Soild
    Molecular weight:364.8
  • Dechloro Rivaroxaban

    CAS:
    <p>Dechloro Rivaroxaban is a Factor Xa inhibitor that inhibits free FXa and plasminogen and fibrin-associated FXa activity in humans.</p>
    Formula:C19H19N3O5S
    Purity:98.63%
    Color and Shape:Solid
    Molecular weight:401.44
  • KB-74935

    CAS:
    <p>KB-74935: enzyme inhibitor, mineralocorticoid blocker, treats cholesterol, hypolipidemia, neurological issues, Alzheimer's.</p>
    Formula:C19H18ClF4N3O3S
    Purity:99.4%
    Color and Shape:Solid
    Molecular weight:479.88
  • CB29

    CAS:
    <p>CB29 is a specific inhibitor of aldehyde dehydrogenase 3A1 (ALDH3A1).</p>
    Formula:C15H15N3O5S
    Purity:99.36%
    Color and Shape:Solid
    Molecular weight:349.36
  • p-Ethynylphenylalanine

    CAS:
    <p>p-Ethynylphenylalanine (4-Ethynyl-L-phenylalanine), a tryptophan hydroxylase (TPH) inhibitor, is competitive, effective, selective, and reversible, with a Ki of</p>
    Formula:C11H11NO2
    Purity:97.57%
    Color and Shape:Solid
    Molecular weight:189.21
  • AMG 579

    CAS:
    <p>AMG 579 is an efficacious and selective inhibitor of PDE10A (IC50 = 0.1 nM).</p>
    Formula:C25H23N5O3
    Purity:99.87%
    Color and Shape:Solid
    Molecular weight:441.48
  • PA452

    CAS:
    <p>PA452 is a selective antagonist of retinoic X receptor (RXR) and suppresses the effect of Retinoic acid on Th1/Th2 development.</p>
    Formula:C26H37N3O3
    Purity:97.14%
    Color and Shape:Solid
    Molecular weight:439.59
  • Setileuton

    CAS:
    <p>Setileuton (MK0633) is a specific 5-LOX inhibitor and can be used in research on asthma and atherosclerosis.</p>
    Formula:C22H17F4N3O4
    Purity:98.85% - 99.35%
    Color and Shape:Solid
    Molecular weight:463.38
  • BI-3231

    CAS:
    <p>BI-3231 is a hydroxysteroid 17ß-dehydrogenase 13 HSD17B13 inhibitor that inhibits hHSD17B13 .BI-3231 can be used to study cirrhosis.</p>
    Formula:C16H14F2N4O3S
    Purity:98.2%
    Color and Shape:Solid
    Molecular weight:380.37
  • NEP-IN-1

    CAS:
    <p>NEP-IN-1 is an inhibitor of neutral endopeptidase (NEP, IC50 = 2 nM) and can be used in studies about female sexual arousal disorders.</p>
    Formula:C21H30ClNO4
    Purity:99.69%
    Color and Shape:Solid
    Molecular weight:395.92
  • Xanthine oxidase-IN-1

    CAS:
    <p>Xanthine oxidase-IN-1 is an effective inhibitor of xanthine oxidase with an IC50 value of 6.5 nM.</p>
    Formula:C16H8F2N2O3
    Purity:97.36% - 99.22%
    Color and Shape:Solid
    Molecular weight:314.24
  • PDE9-IN-(S)-C33

    CAS:
    <p>PDE9-IN-(S)-C33: potent PDE9 inhibitor with 11 nM IC50, for CNS diseases and diabetes study.</p>
    Formula:C18H20ClN5O
    Purity:98.75%
    Color and Shape:Solid
    Molecular weight:357.84
  • PXS-6302 hydrochloride

    CAS:
    <p>PXS-6302 hydrochloride is a potent irreversible lysine oxidase (LOX) inhibitor, inhibiting Bovine LOX, rh LOXL1, rh LOXL2, rh LOXL3, and rh LOXL4 with IC50 of 3</p>
    Formula:C10H11ClF3NO2S
    Purity:99.89%
    Color and Shape:Soild
    Molecular weight:301.71
  • DGAT-1 inhibitor 2

    CAS:
    <p>DGAT-1 inhibitor 2: effective against obesity, targets enzyme in triglyceride synthesis for diabetes treatment.</p>
    Formula:C24H28N4O3
    Purity:98.36%
    Color and Shape:Solid
    Molecular weight:420.5
  • Ranirestat

    CAS:
    <p>Ranirestat (AS-3201) is an AR inhibitor with neuroprotective properties that improves peripheral nerve dysfunction in rats with advanced diabetic polyneuropathy</p>
    Formula:C17H11BrFN3O4
    Purity:98.83% - 99.44%
    Color and Shape:Solid
    Molecular weight:420.19
  • Cudetaxestat

    CAS:
    <p>Cudetaxestat (BLD-0409) is a potent inhibitor of orally active autotaxin.</p>
    Formula:C21H15Cl2F2N3O2S
    Purity:99.9%
    Color and Shape:Solid
    Molecular weight:482.33
  • Varespladib methyl

    CAS:
    <p>Varespladib methyl (LY333013), a bioavailable prodrug of Varespladib, is a selective group II secretory phospholipase A2 inhibitor.</p>
    Formula:C22H22N2O5
    Purity:99.42% - 99.97%
    Color and Shape:Solid
    Molecular weight:394.42
  • ML400

    CAS:
    <p>ML400 (CID73050863) is an allosteric inhibitor of LMPTP with an EC50 of 1μM. ML400 displays good cell-based activity and rodent pharmacokinetics.</p>
    Formula:C24H29N3O
    Purity:99.95%
    Color and Shape:Solid
    Molecular weight:375.51
  • TP-10

    CAS:
    <p>TP-10 is a selective inhibitor of PDE10A against other PDEs with IC50 of 0.8 nM.</p>
    Formula:C26H19F3N4O
    Purity:99.21%
    Color and Shape:Solid
    Molecular weight:460.45
  • Mutant IDH1-IN-2

    CAS:
    <p>Mutant IDH1-IN-2 is a inhibitor of mutant Isocitrate dehydrogenase (IDH) proteins, with IC50 of 16.6 nM in Fluorescence biochemical assay, IC50 of <22 nM in LS-</p>
    Formula:C24H31F2N5O2
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:459.53
  • D-2-Phosphoglyceric acid

    CAS:
    <p>D-2-Phosphoglyceric acid is a crucial metabolic intermediate known for its role in enhancing cellular energy metabolism and regulating biosynthesis. It plays a key role in both glycolysis and photosynthesis, which are essential for cellular energy supply. Additionally, D-2-Phosphoglyceric acid serves as a biomarker for monitoring metabolic states in various organisms.</p>
    Formula:C3H7O7P
    Color and Shape:Solid
    Molecular weight:186.06
  • CYP2C1/CYP2C19-IN-2


    <p>CYP2C1/CYP2C19-IN-2 is a potent inhibitor of CYP2C9/CYP2C19 without liver toxicity or genotoxicity and can be used to study Zika virus (ZIKV) infection.</p>
    Formula:C27H28N2O6S
    Color and Shape:Solid
    Molecular weight:508.59
  • PDE4-IN-12


    <p>PDE4-IN-12 is a potent and safe PDE4 ubiquitous inhibitor that acts on PDE4 (IC50: 3.5 nM, SI: 2.71) and PDE7 (IC50: 15 nM, SI: 4.27).</p>
    Formula:C34H35NO6
    Color and Shape:Solid
    Molecular weight:553.64
  • Clopidogrel-β-D-glucuronide

    CAS:
    <p>Clopidogrel-β-D-glucuronide is a metabolite of Clopidogrel. It directly interacts with the CYP2C8 enzyme and strongly inhibits the hepatic enzyme CYP2C8.</p>
    Formula:C21H22ClNO8S
    Color and Shape:Solid
    Molecular weight:483.919
  • α-Hydroxy alprazolam

    CAS:
    <p>α-Hydroxy alprazolam (U 40125), the primary metabolite of α-Hydroxy alprazolam, possesses pharmacological activity accounting for 60% of that of Alprazolam.</p>
    Formula:C17H13ClN4O
    Color and Shape:Solid
    Molecular weight:324.76