CymitQuimica logo
5-HT Receptor

5-HT Receptor

5-HT receptors, also known as serotonin receptors, are a group of G protein-coupled receptors (GPCRs) that mediate the effects of serotonin, a neurotransmitter involved in mood regulation, anxiety, sleep, appetite, and other physiological processes. These receptors are divided into several subtypes, each with distinct functions and pharmacological properties. 5-HT receptor modulators are widely studied for their roles in treating depression, anxiety disorders, and other neuropsychiatric conditions. At CymitQuimica, we offer a range of high-quality 5-HT receptor modulators to support your research in neuropharmacology, mood disorders, and GPCR signaling.

Found 940 products of "5-HT Receptor"

Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
products per page.
  • LY320954
    Targetmol
    + Info

    LY320954

    CAS:
    <p>LY320954 is an antagonist of 5-HT2A receptor.</p>
    Formula:C21H26N4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:382.46

    Ref: TM-T27945

  • (S)-Bexicaserin
    Targetmol
    + Info

    (S)-Bexicaserin

    CAS:
    <p>(S)-Bexcaserin (compound 2) serves as a 5-HT2C receptor agonist, presenting research possibilities in obesity and psychiatric disorders [1].</p>
    Formula:C15H19F2N3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:295.33

    Ref: TM-T79838

  • Befiradol
    Targetmol
    + Info

    Befiradol

    CAS:
    <p>Befiradol (NLX-112) is an agonist of 5-HT1A receptor.</p>
    Formula:C20H22ClF2N3O
    Color and Shape:Solid
    Molecular weight:393.86

    Ref: TM-T10495L

  • Frovatriptan
    Targetmol
    + Info

    Frovatriptan

    CAS:
    <p>Frovatriptan, potent 5-HT 1B/D agonist, shows high cerebroselectivity and efficacy for migraine with aura.</p>
    Formula:C14H17N3O
    Color and Shape:Solid
    Molecular weight:243.3

    Ref: TM-T60345

  • LY108742
    Targetmol
    + Info

    LY108742

    CAS:
    <p>LY108742 is an antagonist of 5-HT2.</p>
    Formula:C21H28N2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:356.46

    Ref: TM-T27929

  • Dothiepin
    Targetmol
    + Info

    Dothiepin

    CAS:
    <p>Dothiepin (Dosulepin; Dothep), an antidepressant with sedative/anxiolytic properties, preferentially inhibits noradrenaline over serotonin uptake, enhancing</p>
    Formula:C19H21NS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:295.44

    Ref: TM-T78126

  • 5-HT2C agonist-3 free base
    Targetmol
    + Info

    5-HT2C agonist-3 free base

    CAS:
    <p>5-HT2C agonist-3 ((+)-19) free base, a selective 5-HT2C agonist (EC50: 24 nM, Ki: 78 nM), exhibits antipsychotic drug-like activity and inhibits Amphetamine-</p>
    Formula:C19H22FNO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:315.38

    Ref: TM-T79803

  • Brilaroxazine
    Targetmol
    + Info

    Brilaroxazine

    CAS:
    <p>Brilaroxazine (RP5063): multimodal dopamine/5-HT modulator, partial agonist at D2/D3/D4, 5-HT1A/2A, and antagonist at 5-HT2B/7.</p>
    Formula:C22H25Cl2N3O3
    Purity:99.36%
    Color and Shape:Solid
    Molecular weight:450.36

    Ref: TM-T14782

  • Robalzotan
    Targetmol
    + Info

    Robalzotan

    CAS:
    <p>Robalzotan is a selective 5-HT1A receptor antagonist.</p>
    Formula:C18H23FN2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:318.39

    Ref: TM-T24721

  • Gentisein
    Targetmol
    + Info

    Gentisein

    CAS:
    <p>Gentisein (NSC-329491), a primary metabolite of Mangiferin, exhibits significant inhibition of serotonin uptake, demonstrating potency with an IC50 value of 4.7</p>
    Formula:C13H8O5
    Purity:96.89%
    Color and Shape:Solid
    Molecular weight:244.2

    Ref: TM-T19931

  • (±)-Fabesetron hydrochloride
    Targetmol
    + Info

    (±)-Fabesetron hydrochloride

    CAS:
    <p>FK1052 hydrochloride is a potent 5-HT3 and 5-HT4 receptor dual antagonist.</p>
    Formula:C18H20ClN3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:329.82

    Ref: TM-T11293

  • 5-HT3-In-1
    Targetmol
    + Info

    5-HT3-In-1

    CAS:
    <p>5-HT3-In-1 (compound example 8) exhabits with 5-HT3 inhibition activity.</p>
    Formula:C16H21ClN4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:352.82

    Ref: TM-T10006

  • Velusetrag
    Targetmol
    + Info

    Velusetrag

    CAS:
    <p>Velusetrag(TD-5108), a potent 5-HT4 agonist, is in development for gastroparesis, constipation, and IBS.</p>
    Formula:C25H36N4O5S
    Color and Shape:Solid
    Molecular weight:504.64

    Ref: TM-T35046

  • GR-127935
    Targetmol
    + Info

    GR-127935

    CAS:
    <p>GR-127935 is a potent and selective 5-HT1B/1D receptor antagonist.</p>
    Formula:C29H31N5O3
    Color and Shape:Solid
    Molecular weight:497.59

    Ref: TM-T70559

  • 5-HT2 agonist-1 free base
    Targetmol
    + Info

    5-HT2 agonist-1 free base

    CAS:
    <p>Compound 24 (5-HT2 agonist-1 free base) is a potent agonist for 5-HT2A, 5-HT2B, and 5-HT2C receptors, exhibiting IC50 values of 10 nM, 8.3 nM, and 1.6 nM,</p>
    Formula:C19H22N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:310.39

    Ref: TM-T79805

  • Indeloxazine hydrochloride
    Targetmol
    + Info

    Indeloxazine hydrochloride

    CAS:
    <p>Indeloxazine HCl: Serotonin releaser, NE reuptake inhibitor, NMDA antagonist; antidepressant that boosts acetylcholine in rats.</p>
    Formula:C14H18ClNO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:267.75

    Ref: TM-T19629

  • Mesembrine
    Targetmol
    + Info

    Mesembrine

    CAS:
    <p>Mesembrine is an alkaloid, a 5-HT transporter inhibitor (K i 1.4 nM), and inhibits PDE4B (IC50 7.8 μM).</p>
    Formula:C17H23NO3
    Color and Shape:Solid
    Molecular weight:289.37

    Ref: TM-T73857

  • CP-122288
    Targetmol
    + Info

    CP-122288

    CAS:
    <p>CP-122288: potent, selective 5-HT1B/D/F agonist; inhibits plasma protein extravasation, neurogenic inflammation.</p>
    Formula:C16H23N3O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:321.44

    Ref: TM-T27059

  • SB 258719
    Targetmol
    + Info

    SB 258719

    CAS:
    <p>SB 258719 is a selective antagonist of 5-HT7 receptor with pKi of 7.5.</p>
    Formula:C18H30N2O2S
    Purity:99.73%
    Color and Shape:Solid
    Molecular weight:338.51

    Ref: TM-T12855

  • Cyanopindolol fumarate
    Targetmol
    + Info

    Cyanopindolol fumarate

    CAS:
    <p>Cyanopindolol fumarate is a 5-HT receptor antagonist [1].</p>
    Formula:C16H21N3O2C4H4O4
    Color and Shape:Solid
    Molecular weight:345.4

    Ref: TM-T84896