Adrenergic Receptor
Adrenergic receptors are GPCRs that are activated by catecholamines, such as adrenaline and noradrenaline. These receptors are classified into alpha and beta subtypes, each of which plays a key role in the regulation of heart rate, blood pressure, and the fight-or-flight response. Adrenergic receptor modulators are essential in the treatment of cardiovascular diseases, asthma, and anxiety disorders. At CymitQuimica, we offer a wide range of high-quality adrenergic receptor modulators to support your research in endocrinology, cardiovascular pharmacology, and stress response.
Subcategories of "Adrenergic Receptor"
Found 645 products of "Adrenergic Receptor"
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Romifidine hydrochloride
CAS:<p>Romifidine hydrochloride, an α2 adrenergic receptor agonist, induces sedation effects in vivo.</p>Formula:C9H10BrClFN3Color and Shape:SolidMolecular weight:294.55Norepinephrine bitartrate salt
CAS:<p>Norepinephrine bitartrate salt is an adrenergic neurotransmitter.</p>Formula:C12H17NO9Purity:97.32% - 99.97%Color and Shape:SolidMolecular weight:319.27Norepinephrine
CAS:<p>Norepinephrine (Levophed) can stimulate apoptosis in adult rat ventricular myocytes by activation of the β-adrenergic pathway.</p>Formula:C8H11NO3Purity:99.43% - 99.84%Color and Shape:Colorless Microcrystals SolidMolecular weight:169.18Bunazosin
CAS:<p>Bunazosin is a potent and selective α1-adrenoceptor antagonist that can be used for antihypertensive and ocular hypotensive research [1].</p>Formula:C19H27N5O3Color and Shape:SolidMolecular weight:373.45Nifenalol
CAS:<p>Nifenalol is an adrenergic beta-blocker with good antiarrhythmic properties. It tends to lower blood pressure and provide protection against angina.</p>Formula:C11H16N2O3Purity:98%Color and Shape:SolidMolecular weight:224.26Reboxetine mesylate
CAS:<p>Reboxetine mesylate (FCE20124 mesylate) is a norepinephrine reuptake inhibitor (Ki: 8.2 nM).</p>Formula:C19H23NO3·CH4O3SPurity:99.18% - 99.87%Color and Shape:Tan Or Off-White Cyrstalline SolidMolecular weight:409.5Piribedil hydrochloride
CAS:<p>Piribedil HCl treats Parkinson's, circulatory issues, aids cancer research; inhibits MLL1; D2/D3 agonist; α2-antagonist. EC50: 0.18 μM.</p>Formula:C16H19ClN4O2Color and Shape:SolidMolecular weight:334.8Apraclonidine
CAS:<p>Apraclonidine (ALO 2145), an α2/weak α1 agonist, lowers IOP; used as eye drops.</p>Formula:C9H10Cl2N4Color and Shape:SolidMolecular weight:245.11Napitane Mesylate
CAS:<p>Napitane Mesylate inhibits norepinephrine transporter and blocks CNS CA uptake as an alpha 2-adrenoceptor antagonist.</p>Formula:C23H29NO5SPurity:98%Color and Shape:SolidMolecular weight:431.55Xamoterol
CAS:<p>Xamoterol is a cardiac stimulant.</p>Formula:C16H25N3O5Color and Shape:SolidMolecular weight:339.39Methyldopa hydrate
CAS:<p>Methyldopa hydrate (MK-351 hydrate) is a DOPA decarboxylase inhibitor and indirect α2-adrenergic receptor agonist used to treat hypertension.</p>Formula:C10H13NO4H2OPurity:99.67%Color and Shape:White SolidMolecular weight:238.24Pimozide
CAS:<p>Pimozide: antipsychotic that blocks type 2 dopamine, alpha-adrenergic, and 5-HT2 receptors, reducing tics and delusions.</p>Formula:C28H29F2N3OPurity:99.63% - >99.99%Color and Shape:SolidMolecular weight:461.55Desipramine
CAS:<p>Desipramine: tricyclic antidepressant that blocks norepinephrine reuptake and helps reduce sleep-related pharyngeal collapsibility.</p>Formula:C18H22N2Color and Shape:SolidMolecular weight:266.38Medetomidine hydrochloride
CAS:<p>Medetomidine hydrochloride (MPV785) is a selective α2-adrenoceptor agonist, with Ki of 1.08 nM, exhibts 1620-fold selectivity over α1-adrenoceptor.</p>Formula:C13H16N2·HClPurity:99.96%Color and Shape:White Or Off White Crystalline PowderMolecular weight:236.74Scopine
CAS:<p>Scopine (6,7-Epoxytropine), the metabolite of anisodine, is an α1-adrenergic receptor agonist used in the therapy of acute circulatory shock.</p>Formula:C8H13NO2Purity:99.79% - >99.99%Color and Shape:SolidMolecular weight:155.19Bevantolol
CAS:<p>Bevantolol, a selective β-1 adrenoceptor antagonist, is utilized for the investigation of angina pectoris and hypertension [1].</p>Formula:C20H27NO4Color and Shape:SolidMolecular weight:345.43Eformoterol Hemifumarate
CAS:<p>Formoterol fumarate (Eformoterol Hemifumarate), an effective, specific and long-acting β2-adrenoceptor agonist, is utilized in the treatment of COPD and asthma</p>Formula:C19H24N2O4C4H4O4Purity:99.86% - >99.99%Color and Shape:White PowderMolecular weight:402.4Dexmedetomidine
CAS:<p>Dexmedetomidine: a central alpha-2 adrenergic agonist for general anesthesia.</p>Formula:C13H16N2Purity:99% - >99.99%Color and Shape:SolidMolecular weight:200.28nifenalol.HCl
CAS:<p>Nifenalol.HCl(INPEA) is a antagonist of β-adrenergic receptor.</p>Formula:C11H17ClN2O3Purity:99.96%Color and Shape:SolidMolecular weight:260.72Phenylephrine
CAS:<p>Phenylephrine ((R)-(-)-Phenylephrine) is a selective α1-adrenoceptor agonist ( pKi: 5.86, 4.87 and 4.70 for α1D, α1B, and α1A receptors respectively).</p>Formula:C9H13NO2Purity:99.5% - 99.89%Color and Shape:SolidMolecular weight:167.21Talinolol
CAS:<p>(±)-Talinolol is a selective β1 adrenoceptor antagonist well known for its cardioprotective and antihypertensive activity.</p>Formula:C20H33N3O3Purity:98.8%Color and Shape:SolidMolecular weight:363.49Isoetharine mesylate salt
CAS:<p>Isoetharine mesylate salt (Isoetarine mesilate) is a β-adrenergic receptor agonist.</p>Formula:C14H25NO6SPurity:99.35% - 99.75%Color and Shape:SolidMolecular weight:335.42Betaxolol
CAS:<p>Betaxolol (Kerlone) is a selective beta1 adrenergic receptor blocker used in the treatment of hypertension and glaucoma.</p>Formula:C18H29NO3Purity:99.01%Color and Shape:White Crystalline SolidMolecular weight:307.43Droxidopa
CAS:<p>Droxidopa (L-DOPS), an oral prodrug, treats symptomatic orthostatic hypotension from neurogenic autonomic failure.</p>Formula:C9H11NO5Purity:97.27% - 99.88%Color and Shape:SolidMolecular weight:213.19Higenamine hydrochloride
CAS:<p>Higenamine HCl is a β2 adrenoreceptor agonist active in fat and muscle tissue.</p>Formula:C16H18ClNO3Purity:99.44% - 99.80%Color and Shape:White PowderMolecular weight:307.772Amezinium methylsulfate
CAS:<p>Amezinium methylsulfate (Lu-1631) has multiple mechanisms, including stimulation of α and β-1 receptors and inhibition of noradrenaline and tyramine uptake.</p>Formula:C12H15N3O5SPurity:99.64%Color and Shape:SolidMolecular weight:313.33Levobetaxolol hydrochloride
CAS:<p>Levobetaxolol hydrochloride ((S)-Betaxolol hydrochloride) is a beta blocker, used to lower the pressure in the eye in treating conditions such as glaucoma.</p>Formula:C18H29NO3·HClPurity:98.80% - 99.69%Color and Shape:SolidMolecular weight:343.89Meranzin
CAS:<p>Meranzin, a bioactive from TCM CSS, targets alpha 2-adrenoceptor, affects AMPA-ERK1/2–BDNF pathway, and may prevent atherosclerosis and depression.</p>Formula:C15H16O4Purity:95.08% - 99.3%Color and Shape:SolidMolecular weight:260.29(R)-Propranolol hydrochloride
CAS:<p>(R)-Propranolol hydrochloride (Dexpropranolol hydrochloride) is the less active enantiomer of the anti-adrenoceptor (β-adrenoceptor) antagonist propranolol.</p>Formula:C16H22ClNO2Purity:98.63% - 99.01%Color and Shape:SolidMolecular weight:295.8Medetomidine
CAS:<p>Medetomidine (MPV785 free base) is a selective α2-adrenoceptor agonist, with sedative and analgesic and vasoconstrictive hypoxic , in small animal anesthesia.</p>Formula:C13H16N2Purity:99.88%Color and Shape:SolidMolecular weight:200.28CGP 20712 A
CAS:<p>CGP 20712 A (CGP 20712 mesylate) is a β1-adrenergic receptor antagonist with antihypertensive activity that reverses RKT-induced gastric relaxation.</p>Formula:C24H29F3N4O8SPurity:99.37%Color and Shape:SolidMolecular weight:590.57Tamsulosin
CAS:<p>Tamsulosin: an alpha1A blocker for easing urination in BPH by relaxing prostate and bladder muscles.</p>Formula:C20H28N2O5SPurity:99.93%Color and Shape:White CrystalsMolecular weight:408.51Atipamezole
CAS:<p>Atipamezole (Antisedan) is a synthetic α2 adrenergic receptor antagonist. It has also been researched in humans as a potential anti-Parkinsonian drug.</p>Formula:C14H16N2Purity:99.88%Color and Shape:Off-White To Light Yellow Crystal PowderMolecular weight:212.29Alfuzosin
CAS:<p>Alfuzosin (SL 77499) is an alpha-1 adrenergic antagonist used to treat benign prostatic hypertrophy and urethral dysfunction.</p>Formula:C19H27N5O4Purity:99.64%Color and Shape:White Crystaline PowderMolecular weight:389.45Bucindolol
CAS:<p>Bucindolol (BMY 13105) is a novel and potent β1-adrenergic receptor blocker that mediates vasodilation and can be used to study chronic heart failure.</p>Formula:C22H25N3O2Purity:99.9%Color and Shape:SolidMolecular weight:363.45Latrepirdine dihydrochloride
CAS:<p>Latrepirdine dihydrochloride (Dimebolin dihydrochloride) is an orally active, and neuroactive antagonist of multiple drug targets.</p>Formula:C21H25N3·2HClPurity:98.45%Color and Shape:SolidMolecular weight:392.37Fenoterol hydrobromide
CAS:<p>Fenoterol hydrobromide is a beta2-adrenergic receptor agonist and bronchodilator used in the study of cardiovascular diseases such as asthma and bronchitis.</p>Formula:C17H22BrNO4Purity:99.88%Color and Shape:SolidMolecular weight:384.27SR59230A hydrochloride
CAS:<p>SR59230A hydrochloride (SR59230A HCl) is a beta3-adrenergic receptor antagonist that inhibits ultradian brown adipose tissue thermogenesis.</p>Formula:C21H28ClNO2Purity:99.49%Color and Shape:SolidMolecular weight:361.91DL-Phenylephrine HCl
CAS:<p>DL-Phenylephrine HCl is a selective agonist of the alpha1-adrenergic receptor.</p>Formula:C9H14ClNO2Purity:98%Color and Shape:SolidMolecular weight:203.67Tulobuterol
CAS:<p>Tulobuterol is mainly used for the prevention and treatment of bronchial asthma, asthmatic bronchitis and chronic bronchitis. Research shows that it could inhibit rhinovirus infection in primary cultures of human tracheal epithelial cells.</p>Formula:C12H18ClNOColor and Shape:Crystalline SolidMolecular weight:227.73PF-610355
CAS:<p>PF-610355 is a long-acting and potent β2-adrenergic receptor agonist (EC50: 0.26 nM).PF-610355 can be used to study asthma and COPD.</p>Formula:C34H39N3O6SPurity:99.73%Color and Shape:SolidMolecular weight:617.76Buflomedil
CAS:<p>Buflomedil is a vasoactive compound. Buflomedil has been used for peripheral arterial diseases.</p>Formula:C17H25NO4Purity:98%Color and Shape:SolidMolecular weight:307.38Pardoprunox
CAS:<p>Pardoprunox (SLV-308) is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties.</p>Formula:C12H15N3O2Purity:98%Color and Shape:SolidMolecular weight:233.27Penbutolol sulfate
CAS:<p>Penbutolol sulfate ((-)-Terbuclomine) is able to bind to both β2-adrenergic receptor and β1-adrenergic receptor, thus making it a non-selective β blocker.</p>Formula:C18H29NO2H2O4SPurity:98.55%Color and Shape:SolidMolecular weight:340.47Esmolol hydrochloride
CAS:<p>Esmolol is a cardioselective beta-blocker used in parenteral forms in the treatment of arrhythmias and severe hypertension.</p>Formula:C16H25NO4·HClPurity:98.72% - 99.48%Color and Shape:White SolidMolecular weight:331.15Norreticuline
CAS:<p>Norreticuline is a potential adrenoceptor-α/β agonist and CYP2D6 and D2 receptor inhibitor for the study of neurodegenerative diseases.</p>Formula:C18H21NO4Color and Shape:SolidMolecular weight:315.36Isoproterenol sulfate anhydrous
CAS:<p>Isoproterenol sulfate anhydrous is a useful alkaloid. It is used for biological research.</p>Formula:C22H36N2O10SPurity:98%Color and Shape:CoaMolecular weight:520.59Ridazolol HCl
CAS:<p>Ridazolol HCl (CAS 413) is a novel β-adrenoceptor (β-AR) blocker with α-adrenerolytic activity.</p>Formula:C15H19Cl3N4O3Purity:99.48%Color and Shape:SoildMolecular weight:409.7(RS)-ICI-118551 Hydrochloride
CAS:<p>ICI-118551 Hydrochloride (ICI-118,551) is a highly selective β2-adrenergic receptor antagonist with Ki values of 0.7, 49.5 and 611 nM for β2, β1 and β3</p>Formula:C17H27NO2·HClPurity:98.02%Color and Shape:SolidMolecular weight:313.86Atenolol Hydrochloride
CAS:<p>Atenolol Hydrochloride is a selective antagonist of ß1 receptor.</p>Formula:C14H23ClN2O3Purity:98%Color and Shape:SolidMolecular weight:302.80
