NMDAR
N-Methyl-D-Aspartate Receptor (NMDAR) inhibitors are compounds that block the activity of NMDARs, a subtype of glutamate receptors that play a critical role in synaptic plasticity, learning, and memory. Overactivation of NMDARs is implicated in excitotoxicity, which can lead to neuronal damage and is associated with conditions such as stroke, traumatic brain injury, and neurodegenerative diseases. NMDAR inhibitors are essential tools for studying excitotoxicity and for developing neuroprotective therapies. At CymitQuimica, we offer a range of NMDAR inhibitors to support your research in synaptic function, neuroprotection, and cognitive disorders.
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MRZ 2-514
CAS:202808-11-5
MRZ 2-514 (8-bromo-4,5-dihydroxypyridazino[4,5-b]quinolin-1-one) is a strychnine-insensitive modulatory site of the NMDA receptor (glycineB)antagonist with Ki
Formula:
C11H6BrN3O3
Purity:
98.13%
Color and Shape:
Solid
Molecular weight:
308.09
Ref: TM-T12110
| 1mg | 93.00 € | ||
| 5mg | 195.00 € | ||
| 10mg | 318.00 € | ||
| 25mg | 631.00 € | ||
| 50mg | 1,062.00 € | ||
| 100mg | 1,428.00 € | ||
| 1mL*10mM (DMSO) | 216.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
6-Methoxy-2-naphthoic acid
CAS:2471-70-7
6-Methoxy-2-naphthoic acid (6-Methoxy-2-naphthalenecarboxylic acid) is an modulator of NMDAR.
Formula:
C12H10O3
Purity:
99.03%
Color and Shape:
White To Off-White Powder Crystals Crystalline Powder And/Or Chunks
Molecular weight:
202.21
Ref: TM-T0556
| 100mg | 35.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
D-AP5
CAS:79055-68-8
D-AP5 (D-APV) is a NMDA receptor antagonist.
Formula:
C5H12NO5P
Purity:
100% - 98%
Color and Shape:
White Fine Crystalline Powder
Molecular weight:
197.13
Ref: TM-T10930
| 1mg | 35.00 € | ||
| 2mg | 47.00 € | ||
| 5mg | 69.00 € | ||
| 10mg | 109.00 € | ||
| 25mg | 222.00 € | ||
| 50mg | 443.00 € | ||
| 1mL*10mM (DMSO) | 68.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
CIQ
CAS:486427-17-2
CIQ is a subunit-selective potentiator of NMDA receptors containing the NR2C or NR2D subunit. EC50 …
Formula:
C26H26ClNO5
Purity:
99.50%
Color and Shape:
Solid
Molecular weight:
467.94
Ref: TM-T14971
| 2mg | 34.00 € | ||
| 5mg | 49.00 € | ||
| 10mg | 81.00 € | ||
| 25mg | 141.00 € | ||
| 50mg | 203.00 € | ||
| 100mg | 299.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
NMDA-IN-1
CAS:700878-19-9
NMDA-IN-1 is a potent and NR2B-selective antagonist of NMDA(NMDA Ki of 0.85 nM; NR2B Ca2+ …
Formula:
C20H23ClFN3O
Purity:
97.01%
Color and Shape:
Solid
Molecular weight:
375.87
Ref: TM-T12234
| 1mg | 69.00 € | ||
| 5mg | 130.00 € | ||
| 10mg | 218.00 € | ||
| 25mg | 358.00 € | ||
| 50mg | 502.00 € | ||
| 100mg | 676.00 € | ||
| 200mg | 909.00 € | ||
| 1mL*10mM (DMSO) | 144.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Mephenesin
CAS:59-47-2
Mephenesin (Cresoxydiol) is a centrally acting muscle relaxant with a short duration of action.
Formula:
C10H14O3
Purity:
99.52%
Color and Shape:
Solid
Molecular weight:
182.22
Ref: TM-T0015
| 1g | 38.00 € | ||
| 5g | 80.00 € | ||
| 10g | 103.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
BDBM50597431
CAS:1629853-49-1
BDBM50597431 is an NMDA receptor modulator that may have can be used to study Alzheimer's …
Formula:
C27H43F3O2
Purity:
98.64% - 99.28%
Color and Shape:
Soild
Molecular weight:
456.62
Ref: TM-T28367L1
| 1mg | 182.00 € | ||
| 5mg | 400.00 € | ||
| 10mg | 591.00 € | ||
| 25mg | 920.00 € | ||
| 50mg | 1,268.00 € | ||
| 100mg | 1,723.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
SDZ 220-040 ammonium
SDZ 220-040 ammonium is a competitive glutamate ionotropic receptor NMDA antagonist used in the study …
Formula:
C16H19Cl2N2O6P
Purity:
97.31%
Color and Shape:
Liquid
Molecular weight:
437.21
Ref: TM-T23344L
| 1mg | 263.00 € | ||
| 5mg | 629.00 € | ||
| 10mg | 980.00 € | ||
| 25mg | 1,479.00 € | ||
| 50mg | 1,904.00 € | ||
| 100mg | 2,644.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
L-689560
CAS:139051-78-8
L-689560, a radiolabeled ligand, studies NMDA receptors, is an antagonist at GluN1 glycine site.
Formula:
C17H15Cl2N3O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
380.23
Ref: TM-T15684
| 10mg | 634.00 € | ||
| 50mg | 2,646.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Cycloleucine
CAS:52-52-8
Cycloleucine is an antagonist of NMDA receptor associated glycine receptor with a Ki of 600 …
Formula:
C6H11NO2
Purity:
98.13%
Color and Shape:
Liquid
Molecular weight:
129.16
Ref: TM-T9626
| 25mg | 46.00 € | ||
| 50mg | 59.00 € | ||
| 100mg | 86.00 € | ||
| 200mg | 114.00 € | ||
| 500mg | 183.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
ALDH3A1-IN-1
CAS:1039855-56-5
ALDH3A1-IN-1 (Compound 18) is a potent inhibitor of ALDH3A1 with IC50 of 1.61 μM, outperforms …
Formula:
C13H18N2O3
Purity:
99.86%
Color and Shape:
Liquid
Molecular weight:
250.29
Ref: TM-T60372
| 2mg | 44.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
N-Methyl-DL-aspartic acid
CAS:17833-53-3
N-Methyl-DL-aspartic acid, a glutamate analogue and NMDA receptor agonist, is utilized in neurological disease research.
Formula:
C5H9NO4
Purity:
99.62%
Color and Shape:
Liquid
Molecular weight:
147.13
Ref: TM-T64344
| 1g | 34.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Ro 25-6981 Maleate
CAS:1312991-76-6
Ro 25-6981 Maleate is an NMDA receptor antagonist used in the study of neurological disorders …
Formula:
C26H33NO6
Purity:
99.42%
Color and Shape:
Solid
Molecular weight:
455.54
Ref: TM-T12758L
| 1mg | 40.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 165.00 € | ||
| 1mL*10mM (DMSO) | 94.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Lanicemine dihydrochloride
CAS:153322-06-6
Lanicemine dihydrochloride (AZD-6765 dihydrochloride) is an NMDA channel blocker with antidepressant activity and can be …
Formula:
C13H16Cl2N2
Purity:
99.43%
Color and Shape:
Liquid
Molecular weight:
271.19
Ref: TM-T60471
| 2mg | 35.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 90.00 € | ||
| 25mg | 169.00 € | ||
| 50mg | 271.00 € | ||
| 100mg | 414.00 € | ||
| 500mg | 898.00 € | ||
| 1mL*10mM (DMSO) | 45.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
NKH477
CAS:138605-00-2
NKH477, a water-soluble forskolin derivative, enhances cardiac function, has antiproliferative properties, and boosts cAMP levels.
Formula:
C27H44ClNO8
Purity:
98%
Color and Shape:
Solid
Molecular weight:
546.09
Ref: TM-T16332
| 2mg | 66.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Rapastinel
CAS:117928-94-6
Rapastinel (TPPT-amide) (GLYX-13) is an N-methyl-D-aspartate receptor (NMDAR) modulator.
Formula:
C18H31N5O6
Purity:
98%
Color and Shape:
Solid
Molecular weight:
413.47
Ref: TM-T3407
| 1mg | 47.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 114.00 € | ||
| 25mg | 226.00 € | ||
| 50mg | 336.00 € | ||
| 1mL*10mM (DMSO) | 90.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
DNQX disodium salt
CAS:1312992-24-7
DNQX disodium salt is a water-soluble form of selective antagonist of non-NMDA receptor
Formula:
C8H2N4Na2O6
Purity:
100%
Color and Shape:
Solid
Molecular weight:
296.1
Ref: TM-T8459
| 1mg | 85.00 € | ||
| 5mg | 170.00 € | ||
| 10mg | 250.00 € | ||
| 25mg | 411.00 € | ||
| 50mg | 577.00 € | ||
| 100mg | 781.00 € | ||
| 200mg | 1,035.00 € | ||
| 1mL*10mM (DMSO) | 169.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Traxoprodil
CAS:134234-12-1
Traxoprodil (CP101606) is a selective NMDA antagonist and protects hippocampal neurons (IC50: 10 nM).
Formula:
C20H25NO3
Purity:
99.86%
Color and Shape:
Solid
Molecular weight:
327.42
Ref: TM-TQ0233
| 5mg | 56.00 € | ||
| 10mg | 74.00 € | ||
| 25mg | To inquire | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
ZL006
CAS:1181226-02-7
ZL006 is an effective inhibitor of nNOS/PSD-95 interaction. ZL006 also inhibits NMDA receptor-mediated NO synthesis.
Formula:
C14H11Cl2NO4
Purity:
98.29%
Color and Shape:
Solid
Molecular weight:
328.15
Ref: TM-T17293
| 1mg | 38.00 € | ||
| 2mg | 49.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 98.00 € | ||
| 25mg | 186.00 € | ||
| 50mg | 296.00 € | ||
| 100mg | 506.00 € | ||
| 200mg | 730.00 € | ||
| 500mg | 1,095.00 € | ||
| 1mL*10mM (DMSO) | 88.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Dizocilpine Maleate
CAS:77086-22-7
Dizocilpine Maleate (MK 801) is a potent noncompetitive antagonist of the NMDA receptor with Kd …
Formula:
C20H19NO4
Purity:
99% - 99.96%
Color and Shape:
White Solid
Molecular weight:
337.38
Ref: TM-T3320
| 5mg | 38.00 € | ||
| 10mg | 54.00 € | ||
| 25mg | 89.00 € | ||
| 50mg | 143.00 € | ||
| 100mg | 251.00 € | ||
| 200mg | 412.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
