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NMDAR

NMDAR

N-Methyl-D-Aspartate Receptor (NMDAR) inhibitors are compounds that block the activity of NMDARs, a subtype of glutamate receptors that play a critical role in synaptic plasticity, learning, and memory. Overactivation of NMDARs is implicated in excitotoxicity, which can lead to neuronal damage and is associated with conditions such as stroke, traumatic brain injury, and neurodegenerative diseases. NMDAR inhibitors are essential tools for studying excitotoxicity and for developing neuroprotective therapies. At CymitQuimica, we offer a range of NMDAR inhibitors to support your research in synaptic function, neuroprotection, and cognitive disorders.

Found 28 products of "NMDAR"

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  • Mephenesin
    Targetmol
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    Mephenesin

    CAS:
    <p>Mephenesin (Cresoxydiol) is a centrally acting muscle relaxant with a short duration of action.</p>
    Formula:C10H14O3
    Purity:99.49%
    Color and Shape:Solid
    Molecular weight:182.22

    Ref: TM-T0015

  • SDZ 220-040 ammonium
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    SDZ 220-040 ammonium

    <p>SDZ 220-040 ammonium is a competitive glutamate ionotropic receptor NMDA antagonist used in the study of neurological disorders.</p>
    Formula:C16H19Cl2N2O6P
    Purity:98.47%
    Color and Shape:Solid
    Molecular weight:437.21

    Ref: TM-T23344L

  • L-689560
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    L-689560

    CAS:
    <p>L-689560, a radiolabeled ligand, studies NMDA receptors, is an antagonist at GluN1 glycine site.</p>
    Formula:C17H15Cl2N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:380.23

    Ref: TM-T15684

  • S1R agonist 2
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    S1R agonist 2

    CAS:
    <p>S1R agonist 2 is a selective S1R agonist with a Ki of 88 nM for S2R and 1.1 nM for S1R and is protective against ROS and NMDA-induced neurotoxicity.</p>
    Formula:C21H27NO
    Purity:98.85%
    Color and Shape:Solid
    Molecular weight:309.45

    Ref: TM-T72059

  • GluN2B receptor modulator-1
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    GluN2B receptor modulator-1

    CAS:
    <p>GluN2B receptor modulator-1 is a selective negative allosteric modulator of NMDA receptor GluN2B subunits (IC50 31 nM), valuable for neuropharmacology studies.</p>
    Formula:C17H15F3N4O2S
    Purity:99.56%
    Color and Shape:Solid
    Molecular weight:396.39

    Ref: TM-T39694

  • QNZ46
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    QNZ46

    CAS:
    <p>QNZ46 is a NR2C/NR2D-selective NMDA receptor non-competitive antagonist.</p>
    Formula:C24H17N3O6
    Purity:99.65%
    Color and Shape:Solid
    Molecular weight:443.41

    Ref: TM-T2362

  • Flutriafol
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    Flutriafol

    CAS:
    <p>Flutriafol is a pesticide, demethylation inhibitor, and NMDA receptor agonist</p>
    Formula:C16H13F2N3O
    Purity:98.75%
    Color and Shape:Solid
    Molecular weight:301.29

    Ref: TM-T7867

  • DNQX disodium salt
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    DNQX disodium salt

    CAS:
    <p>DNQX disodium salt is a water-soluble form of selective antagonist of non-NMDA receptor</p>
    Formula:C8H2N4Na2O6
    Purity:98.93%
    Color and Shape:Solid
    Molecular weight:296.1

    Ref: TM-T8459

  • Dizocilpine Maleate
    Targetmol
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    Dizocilpine Maleate

    CAS:
    <p>Dizocilpine Maleate (MK 801) is a potent noncompetitive antagonist of the NMDA receptor with Kd of 37.2 nM in rat brain membranes.</p>
    Formula:C20H19NO4
    Purity:99% - 99.96%
    Color and Shape:White Solid
    Molecular weight:337.38

    Ref: TM-T3320

  • Rapastinel Trifluoroacetate
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    Rapastinel Trifluoroacetate

    CAS:
    <p>Rapastinel Trifluoroacetate (GLYX-13 Trifluoroacetate) is an NMDA receptor modulator with glycine-site partial agonist properties.</p>
    Formula:C20H32F3N5O8
    Purity:99.01% - 99.77%
    Color and Shape:Solid
    Molecular weight:527.49

    Ref: TM-T5819

  • ZL006
    Targetmol
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    ZL006

    CAS:
    <p>ZL006 is an effective inhibitor of nNOS/PSD-95 interaction. ZL006 also inhibits NMDA receptor-mediated NO synthesis.</p>
    Formula:C14H11Cl2NO4
    Purity:98.29%
    Color and Shape:Solid
    Molecular weight:328.15

    Ref: TM-T17293

  • Traxoprodil
    Targetmol
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    Traxoprodil

    CAS:
    <p>Traxoprodil (CP101606) is a selective NMDA antagonist and protects hippocampal neurons (IC50: 10 nM).</p>
    Formula:C20H25NO3
    Purity:99.89%
    Color and Shape:Solid
    Molecular weight:327.42

    Ref: TM-TQ0233

  • (-)-Dizocilpine maleate
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    (-)-Dizocilpine maleate

    CAS:
    <p>(-)-Dizocilpine maleate ((-)-MK 801 (Maleate)) is a potent, selective and non-competitive NMDA receptor antagonist with Kd of 37.2 nM in rat brain membranes.</p>
    Formula:C20H19NO4
    Purity:>99.99%
    Color and Shape:White Solid
    Molecular weight:337.37

    Ref: TM-T6352

  • Acamprosate
    Targetmol
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    Acamprosate

    CAS:
    <p>Acamprosate, alcohol dependence treatment. Affordable Excellence: Reliable Quality You Can Trust</p>
    Formula:C5H11NO4S
    Purity:98.30%
    Color and Shape:Solid
    Molecular weight:181.21

    Ref: TM-T73059

  • Glypromate acetate(32302-76-4 free base)
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    Glypromate acetate(32302-76-4 free base)

    <p>Glypromate acetate is a neuroprotective agent, is a weak NMDA receptor agonist.</p>
    Formula:C14H23N3O8
    Purity:99.94%
    Color and Shape:Solid
    Molecular weight:361.35

    Ref: TM-T7778L

  • Flupirtine maleate
    Targetmol
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    Flupirtine maleate

    CAS:
    <p>Flupirtine maleate (Katadolon maleate), a centrally acting non-opioid analgesia, is the salt form of Flupirtine. Flupirtine is an NMDA receptor antagonist.</p>
    Formula:C15H17FN4O2·C4H4O4
    Purity:99.5% - 99.9%
    Color and Shape:Off-White Crystalline Powder
    Molecular weight:420.39

    Ref: TM-T6504

  • L-701324
    Targetmol
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    L-701324

    CAS:
    <p>L-701324 is an NMDA receptor with high affinity and selectivity for the glycine site, used as an orally active and long-acting anticonvulsant.</p>
    Formula:C21H14ClNO3
    Purity:98.63% - >99.99%
    Color and Shape:Solid
    Molecular weight:363.79

    Ref: TM-T1909

  • TCN 201
    Targetmol
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    TCN 201

    CAS:
    <p>TCN 201 is a selective antagonist of NMDA receptors containing the NR2A subunit.</p>
    Formula:C21H17ClFN3O4S
    Purity:98.5%
    Color and Shape:Solid
    Molecular weight:461.89

    Ref: TM-T7870

  • Eliprodil
    Targetmol
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    Eliprodil

    CAS:
    <p>Eliprodil (SL-820715), NR2B-NMDA receptor blocker (IC50: 1 uM), less potent on NR2A/NR2C (IC50&gt;100 uM), explored for Parkinson's and movement issues.</p>
    Formula:C20H23ClFNO
    Purity:99.53% - 99.77%
    Color and Shape:Solid
    Molecular weight:347.85

    Ref: TM-T1751

  • Radiprodil
    Targetmol
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    Radiprodil

    CAS:
    <p>Radiprodil (RGH-896) is an oral NMDA NR2B antagonist for potential DPNP neuropathic pain treatment.</p>
    Formula:C21H20FN3O4
    Purity:99.74%
    Color and Shape:Solid
    Molecular weight:397.4

    Ref: TM-T5385