PYK2
AZ7550
CAS:1421373-99-0
AZ7550, an active metabolite of AZD9291, inhibits the activity of IGF1R (IC50: 1.6 μM).
Formula:
C27H31N7O2
Purity:
97.07%
Color and Shape:
Solid
Molecular weight:
485.58
Ref: TM-T13564
1mg | 129.00 € | |
5mg | 282.00 € | |
10mg | 417.00 € | |
25mg | 689.00 € | |
50mg | 920.00 € | |
100mg | 1,287.00 € |
Estimated delivery in United States, on Thursday 9 May 2024
PF-431396
CAS:717906-29-1
PF-431396 is a dual PYK2/FAK inhibitor (IC50: 11/2 nM).
Formula:
C22H21F3N6O3S
Purity:
99.82%
Color and Shape:
Solid
Molecular weight:
506.5
Ref: TM-T2314
5mg | 59.00 € | |
10mg | 85.00 € | |
25mg | 148.00 € | |
50mg | 249.00 € | |
100mg | 420.00 € | |
200mg | 617.00 € | |
1ml*10 (DMSO) | 64.00 € |
Estimated delivery in United States, on Thursday 9 May 2024
PF-562271 besylate
CAS:939791-38-5
PF-562271 besylate (PF-00562271 Besylate) is a potent, ATP-competitive, reversible inhibitor of FAK with IC50 of …
Formula:
C21H20F3N7O3S·C6H6O3S
Purity:
99.5%
Color and Shape:
Solid
Molecular weight:
665.66
Ref: TM-T6177
1mg | 58.00 € | |
2mg | 80.00 € | |
5mg | 116.00 € | |
10mg | 145.00 € | |
25mg | 232.00 € | |
50mg | 343.00 € | |
100mg | 513.00 € | |
1ml*10 (DMSO) | 155.00 € |
Estimated delivery in United States, on Thursday 9 May 2024
NVP-TAE 226
CAS:761437-28-9
NVP-TAE 226 (TAE226) is an effective FAK inhibitor (IC50: 5.5 nM) and most effective to …
Formula:
C23H25ClN6O3
Purity:
99.17%
Color and Shape:
Solid
Molecular weight:
468.94
Ref: TM-T1918
1mg | 48.00 € | |
2mg | 62.00 € | |
5mg | 99.00 € | |
10mg | 160.00 € | |
25mg | 258.00 € | |
50mg | 369.00 € | |
100mg | 555.00 € | |
1ml*10 (DMSO) | 99.00 € |
Estimated delivery in United States, on Thursday 9 May 2024
PF-562271 hydrochloride
CAS:939791-41-0
PF-562271 hydrochloride (PF-562271 HCl) is a potent, ATP-competitive, reversible inhibitor of FAK with IC50 of …
Formula:
C21H20F3N7O3SHCl
Purity:
98.52%
Color and Shape:
Solid
Molecular weight:
543.95
Ref: TM-T21768
5mg | 77.00 € | |
10mg | 95.00 € | |
25mg | 149.00 € | |
50mg | 209.00 € | |
100mg | 309.00 € |
Estimated delivery in United States, on Thursday 9 May 2024
PF-562271
CAS:717907-75-0
PF-562271 is an effective ATP-competitive, reversible inhibitor of FAK(IC50=1.5 nM) and Pyk2 kinase(IC50=13 nM).
Formula:
C21H20F3N7O3S
Purity:
100%
Color and Shape:
Solid
Molecular weight:
507.49
Ref: TM-T2465
1mg | 58.00 € | |
5mg | 125.00 € | |
10mg | 156.00 € | |
25mg | 255.00 € | |
50mg | 370.00 € | |
100mg | 555.00 € | |
500mg | 1,163.00 € | |
1ml*10 (DMSO) | 138.00 € |
Estimated delivery in United States, on Thursday 9 May 2024
Conteltinib
CAS:1384860-29-0
Conteltinib (CT-707) is an enzyme inhibitor with antitumor activity targeting FAK, ALK, and Pyk2.Conteltinib exhibits …
Formula:
C32H45N9O3S
Purity:
99.54%
Color and Shape:
Solid
Molecular weight:
635.82
Ref: TM-T14997
25mg | 711.00 € | |
50mg | 933.00 € | |
100mg | 1,460.00 € |
Estimated delivery in United States, on Thursday 20 Jun 2024