Histamine Receptor
Histamine receptors are GPCRs that mediate the effects of histamine, a biogenic amine involved in immune responses, gastric acid secretion, and neurotransmission. There are four subtypes of histamine receptors (H1, H2, H3, and H4), each playing distinct roles in allergic reactions, gastric function, and central nervous system activity. Histamine receptor antagonists are widely used in the treatment of allergies, peptic ulcers, and motion sickness. At CymitQuimica, we provide a comprehensive selection of high-quality histamine receptor modulators to support your research in immunology, gastroenterology, and neuropharmacology.
Found 358 products of "Histamine Receptor"
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Niperotidine
CAS:<p>Niperotidine is an antagonist of histamine H2-receptor.</p>Formula:C20H26N4O5SPurity:98%Color and Shape:SolidMolecular weight:434.51Iodophenpropit dihydrobromide
CAS:<p>Iodophenpropit dihydrobromide: selective histamine H3 antagonist, reversible binding, high affinity (KD: 0.32 nM).</p>Formula:C15H20BrIN4SPurity:98%Color and Shape:SolidMolecular weight:495.22PF-03654746 Tosylate
CAS:<p>PF-03654746 Tosylate is selective antagonist of histamine H3 receptor with high brain penetration.</p>Formula:C25H32F2N2O4SPurity:98%Color and Shape:SolidMolecular weight:494.6JNJ-39220675
CAS:<p>JNJ-39220675, a selective histamine H3 receptor antagonist, reduces the abuse-related effects of alcohol in rats.</p>Formula:C21H24FN3O2Purity:98.13% - 99.89%Color and Shape:SolidMolecular weight:369.43JNJ-28610244
CAS:<p>JNJ-28610244 is a specific agonist of the H4 receptor. It acts by blocking Mac-1-dependent activation of p38 MAPK.</p>Formula:C16H21N3OPurity:98%Color and Shape:SolidMolecular weight:271.36Hetramine
CAS:<p>Hetramine is a synthetic pyrimidine agent that possesses antihistamine and anti anaphylactic effects.</p>Formula:C15H20N4Purity:98%Color and Shape:SolidMolecular weight:256.35Fenethazine
CAS:<p>Fenethazine is an effective antihistamine used as an antiallergic drug.</p>Formula:C16H18N2SColor and Shape:SolidMolecular weight:270.39HSR-609
CAS:<p>HSR-609, a histamine H1 receptor antagonist, is used potentially for the treatment of allergic rhinitis.</p>Formula:C21H21FN2O3Purity:98%Color and Shape:SolidMolecular weight:368.4Setastine
CAS:<p>Setastine, a highly selective H1 receptor antagonist, acts as a non-sedative antihistamine.</p>Formula:C22H28ClNOColor and Shape:SolidMolecular weight:357.92BMH-7
CAS:<p>BMH-7 (Histamine H4 receptor antagonist-2) is a p53 activator, demonstrating anti-cancer activity by activating the p53 pathway.</p>Formula:C20H21N5OPurity:99.71%Color and Shape:SolidMolecular weight:347.41Tei 6472
CAS:<p>Tei 6472 is a more hydrophilic form of TEI-1338 which is a novel, selective lipoxygenase inhibitor.</p>Formula:C32H39N3O5Purity:98%Color and Shape:SolidMolecular weight:545.67Nα-Methylhistamine dihydrochloride
CAS:<p>Nα-Methylhistamine dihydrochloride is a histamine H3 receptor agonist.</p>Formula:C6H13Cl2N3Purity:98%Color and Shape:SolidMolecular weight:198.094Embramine
CAS:<p>Embramine, used as an antihistamine and anticholinergic, is a monoethanolamine.</p>Formula:C18H22BrNOPurity:98%Color and Shape:SolidMolecular weight:348.28PF 03654746 FA
<p>PF 03654746 FA is a human histamine receptor H(3) antagonist that can be used to study cognitive impairment and Alzheimer's disease.</p>Formula:C19H26F2N2O3Purity:99.44%Color and Shape:SoildMolecular weight:368.42VUF 8430 dihydrobromide
CAS:<p>histamine H4 receptor full agonist</p>Formula:C4H12BrN5SPurity:98%Color and Shape:SolidMolecular weight:242.14Bavisant dihydrochloride
CAS:<p>Bavisant (JNJ-310010740) is an oral, selective H3 receptor antagonist enhancing wakefulness and cognition.</p>Formula:C19H29Cl2N3O2Purity:98%Color and Shape:SolidMolecular weight:402.36ICI 162,846
CAS:<p>ICI 162,846 is an orally active and potent H2 receptor antagonist that inhibits gastric secretion and may be used in the study of duodenal ulcers.</p>Formula:C11H17F3N6OPurity:97.45%Color and Shape:SolidMolecular weight:306.29Setastine HCl
CAS:<p>Setastine HCl is a potent antagonist of histamine H1-receptor mediated responses.</p>Formula:C22H29Cl2NOColor and Shape:SolidMolecular weight:394.38A 987306
CAS:<p>A-987306: Potent, oral histamine H4 antagonist; Ki: 3.4 nM (rat), 5.8 nM (human); reduces inflammation in mouse peritonitis.</p>Formula:C18H25N5OColor and Shape:SolidMolecular weight:327.42Azelastine
CAS:<p>Azelastine (Azelastinum) is a phthalazine derivative, and is an histamine antagonist and mast cell stabilizer.</p>Formula:C22H24ClN3OPurity:99.35%Color and Shape:White Crystal PowderMolecular weight:381.90Zaltidine
CAS:<p>Zaltidine is an antagonist of H2-receptor, and has the antisecretory action.</p>Formula:C8H10N6SPurity:98%Color and Shape:SolidMolecular weight:222.27JNJ-10191584
CAS:<p>JNJ-10191584, a potent and selective antagonist at the histamine H4 receptor, has antiinflammatory and analgesic effects in animal studies of acute inflammation</p>Formula:C13H15ClN4OColor and Shape:SolidMolecular weight:278.74Alimemazine
CAS:<p>Alimemazine, an antipruritic and HA-receptor antagonist, also partially activates H1R and other GPCRs.</p>Formula:C18H22N2SPurity:98%Color and Shape:Crystals SolidMolecular weight:298.45Aminopotentidine
CAS:<p>H2 antagonist</p>Formula:C26H35N7O2Purity:98%Color and Shape:SolidMolecular weight:477.6Zolantidine dimaleate
CAS:<p>H2 receptor antagonist</p>Formula:C26H31N3O5SPurity:98%Color and Shape:SolidMolecular weight:497.61BMY-25271
CAS:<p>BMY-25271 is an antagonist of histamine H2 receptor.</p>Formula:C12H19N5O2S2Purity:98%Color and Shape:SolidMolecular weight:329.44ABT-239
CAS:<p>ABT-239 is a novel, highly efficacious antagonist belonging to the non-imidazole class of histamine H3 receptor (H3R) antagonists.</p>Formula:C22H22N2OPurity:>99.99%Color and Shape:SolidMolecular weight:330.42(R)-Mequitazine
CAS:<p>(R)-Mequitazine, a muscarinic acetylcholine receptor (M-AChRs) antagonist, is used potentially for the treatment of asthma.</p>Formula:C20H22N2SColor and Shape:SolidMolecular weight:322.47A-304121
CAS:<p>A-304121 is a histamine H(3) receptor.</p>Formula:C20H29N3O3Color and Shape:SolidMolecular weight:359.46OUP-186
CAS:<p>OUP-186 is a selective H3 receptor antagonist that suppresses breast cancer cell growth with an IC50 of ~50 μM and induces apoptosis.</p>Formula:C19H30ClN3SColor and Shape:SolidMolecular weight:367.98JNJ 10181457 dihydrochloride
CAS:<p>JNJ 10181457 dihydrochloride is a Histamine H3 receptor antagonist.</p>Formula:C20H28N2OPurity:98%Color and Shape:SolidMolecular weight:312.45Mianserin
CAS:<p>Mianserin, an H1 receptor reverse agonist, is a psychoactive compound in the tetracyclic antidepressant (TeCA) treatment family.</p>Formula:C18H20N2Purity:99.85%Color and Shape:SolidMolecular weight:264.36Wy 49051
CAS:<p>Wy 49051 is an orally active antagonist of H1 receptor(IC50 of 44 nM).</p>Formula:C28H33N5O3Purity:99.89%Color and Shape:SolidMolecular weight:487.59ROS 234
CAS:<p>ROS 234 is a potent H3 antagonist with pKB 9.46 for Guinea-pig ileum and pKi 8.90 for Rat cortex; ED50 of 19.12 mg/kg in rats, but with limited central access.</p>Formula:C13H15N5Color and Shape:SolidMolecular weight:241.29PF-03654746
CAS:<p>PF-03654746: selective H3 antagonist, boosts cognition in Alzheimer's, may treat allergic rhinitis.</p>Formula:C18H24F2N2OPurity:98.85% - 99.57%Color and Shape:SolidMolecular weight:322.39AZD5213
CAS:<p>AZD5213: selective human H3 receptor antagonist, pKi 9.3, for sleep/cognition research.</p>Formula:C19H25N3O2Color and Shape:SolidMolecular weight:327.42Repirinast
CAS:<p>Repirinast is a mediator release inhibitor. It is used to treat asthma.</p>Formula:C20H21NO5Color and Shape:SolidMolecular weight:355.38Immepip
CAS:<p>Immepip, a H3 agonist, has been shown to attenuate cortical histamine release and is utilized in the research of neurological diseases.</p>Formula:C9H15N3Color and Shape:SolidMolecular weight:165.24Phenyltoloxamine
CAS:<p>Phenyltoloxamine (Bistrimin): antihistamine with sedative, analgesic properties, and Sigma-1 receptor affinity (Ki=160 nM).</p>Formula:C17H21NOColor and Shape:SolidMolecular weight:255.35Mizolastine dihydrochloride
CAS:<p>Mizolastine dihydrochloride is a histamine H1-receptor antagonist (IC50: 47 nM).</p>Formula:C24H27Cl2FN6OPurity:98%Color and Shape:SolidMolecular weight:505.42GSK 189254 HCl
CAS:<p>GSK 189254A: histamine H3 antagonist, treats narcolepsy, may improve cognition and help with dementia, neuropathic pain.</p>Formula:C21H26ClN3O2Purity:98%Color and Shape:SolidMolecular weight:387.9GSK334429
CAS:<p>GSK334429 is an antagonist of histamine H3 receptor.</p>Formula:C20H29F3N4OColor and Shape:SolidMolecular weight:398.47Sequifenadine
CAS:<p>Sequifenadine has the potential in researching of inflammatory eye disease with allergic symptoms that is a H1-antihistamine [1] [2].</p>Formula:C22H27NOColor and Shape:SolidMolecular weight:321.46A-940894
CAS:<p>A-940894: Potent H4 receptor antagonist, anti-inflammatory, binds well to human/rat H4, low affinity for H1/H2/H3, good pharmacokinetics.</p>Formula:C17H21N5Color and Shape:SolidMolecular weight:295.38Loratadine N-oxide
CAS:<p>Loratadine N-oxide is a metabolite of the histamine H1 receptor inverse agonist loratadine.</p>Formula:C22H23ClN2O3Color and Shape:SolidMolecular weight:398.88MK-0249
CAS:<p>MK-0249 is a potent antagonist of histamine H3 receptor (human H3, Ki : 1.7 nM).</p>Formula:C23H24F3N3O2Purity:99.90%Color and Shape:SolidMolecular weight:431.45N-Acetylhistamine
CAS:<p>N-Acetylhistamine (N-Omega-acetylhistamine) is a metabolite of histamine.</p>Formula:C7H11N3OPurity:99.51%Color and Shape:SolidMolecular weight:153.18Izuforant
CAS:<p>Izuforant (JW1601) has anti-inflammatory effects, binds h5-HT3R (IC50: 9.1 μM), and blocks H4R orally (IC50: 36 nM).</p>Formula:C12H12BrN7Color and Shape:SolidMolecular weight:334.17A-943931
CAS:<p>A-943931 is a selective histamine H4 receptor antagonist with human and rat Ki values of 4.6 and 3.8 nM respectively.inhibits the scratching response in mice.</p>Formula:C17H21N5Purity:99.79%Color and Shape:SolidMolecular weight:295.38Pitolisant oxalate
CAS:<p>Pitolisant oxalate is a potent and selective inverse agonist of nonimidazole at the recombinant human histamine H3 receptor with Ki of 0.16 nM.</p>Formula:C19H28ClNO5Purity:98%Color and Shape:SolidMolecular weight:385.88
