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Opioid Receptor

Opioid Receptor

Opioid receptors are a group of G protein-coupled receptors that mediate the effects of endogenous and exogenous opioids. These receptors play a central role in pain modulation, mood regulation, and addictive behaviors. Opioid receptor agonists and antagonists are extensively used in pain management and addiction treatment, as well as in research on neurological and psychiatric disorders. At CymitQuimica, we provide a comprehensive selection of high-quality opioid receptor modulators to support your research in neurobiology, pain management, and addiction therapy.

Found 296 products of "Opioid Receptor"

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  • BMS-986121
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    BMS-986121

    CAS:
    <p>BMS-986121 is a selective positive allosteric modulator (PAM) of the μ opioid receptor with analgesic effects.</p>
    Formula:C15H9Cl2N3O2S
    Purity:99.67%
    Color and Shape:Solid
    Molecular weight:366.22

    Ref: TM-T40392

  • Asimadoline
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    Asimadoline

    CAS:
    <p>Asimadoline (EMD-61753) is a proprietary small molecule therapeutic, originally discovered by Merck KGaA of Darmstadt, Germany.</p>
    Formula:C27H30N2O2
    Color and Shape:Solid
    Molecular weight:414.54

    Ref: TM-T4633

  • LY2940094 tartrate
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    LY2940094 tartrate

    CAS:
    <p>LY-2940094, a nociceptin receptor antagonist, is used potentially for the treatment of major depressive disorder and alcoholism.</p>
    Formula:C26H29ClF2N4O8S
    Color and Shape:Solid
    Molecular weight:631.04

    Ref: TM-T27939

  • Naloxegol (NKTR-118)
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    Naloxegol (NKTR-118)

    CAS:
    <p>Naloxegol (NKTR-118; AZ-13337019) is an opioid-receptor antagonist[1].</p>
    Formula:C34H53NO11
    Color and Shape:Solid
    Molecular weight:651.78

    Ref: TM-T36374

  • b-Casomorphin (1-3) Acetate
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    b-Casomorphin (1-3) Acetate

    <p>b-Casomorphin (1-3) Acetate is a tri-peptide with an opioid effect.</p>
    Formula:C25H31N3O7
    Purity:98.99%
    Color and Shape:Solid
    Molecular weight:485.53

    Ref: TM-T21660L

  • BMS986187
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    BMS986187

    CAS:
    <p>BMS986187 is a novel Potent and Selective Positive Allosteric Modulators of the delta-Opioid Receptor.</p>
    Formula:C31H34O4
    Purity:99.09%
    Color and Shape:Solid
    Molecular weight:470.6

    Ref: TM-T8991

  • N-terminally acetylated Leu-enkephalin
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    N-terminally acetylated Leu-enkephalin

    <p>Leu-enkephalin, an endogenous 5-amino acid peptide, activates opioid receptors; its acetylated form exists.</p>
    Formula:C30H39N5O8
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:597.66

    Ref: TM-T8557

  • Ac-RYYRWK-NH2 acetate
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    Ac-RYYRWK-NH2 acetate

    <p>Ac-RYYRWK-NH2 acetate is a potent partial agonist of the nociceptin receptor(NOP), which is the endogenous ORL1 receptor agonist.</p>
    Formula:C51H73N15O11
    Purity:98.59%
    Color and Shape:Solid
    Molecular weight:1072.22

    Ref: TM-TP1941L1

  • Nalmefene hydrochloride
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    Nalmefene hydrochloride

    CAS:
    <p>Nalmefene antagonizes the effects of opioids by competing for the opioid receptors in the CNS.</p>
    Formula:C21H26ClNO3
    Purity:98% - 99.85%
    Color and Shape:Solid
    Molecular weight:375.89

    Ref: TM-T6221

  • Sinomenine
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    Sinomenine

    CAS:
    <p>Sinomenine (Kukoline) is a pure alkaloid isolated from the Sinomenium acutum, is utilized in the treatment of rheumatism and arthritis.</p>
    Formula:C19H23NO4
    Purity:99.02% - 99.73%
    Color and Shape:White Powder
    Molecular weight:329.39

    Ref: TM-T2726

  • Hemorphin-7 acetate(152685-85-3 free base)
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    Hemorphin-7 acetate(152685-85-3 free base)

    <p>Hemorphin-7 acetate is a hemorphin peptide, an endogenous opioid peptide derived from the β-chain of hemoglobin.</p>
    Formula:C51H68N12O13
    Purity:99.66%
    Color and Shape:Solid
    Molecular weight:1057.16

    Ref: TM-TP1404L

  • Leuphasyl TFA
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    Leuphasyl TFA

    CAS:
    <p>Leuphasyl TFA: a long-lasting, degradation-resistant peptide &amp; δ-opioid receptor agonist for signaling research.</p>
    Formula:C31H40F3N5O9
    Purity:98.79%
    Color and Shape:Solid
    Molecular weight:683.67

    Ref: TM-T20435L

  • EST73502 hydrochloride
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    EST73502 hydrochloride

    CAS:
    <p>EST73502 HCl is an oral dual MOR agonist/σ1R antagonist, BBB-penetrant, Ki: 64 nM (MOR), 118 nM (σ1R), with antinociceptive properties.</p>
    Formula:C19H27ClF2N2O2
    Color and Shape:Solid
    Molecular weight:388.88

    Ref: TM-T9669

  • Naloxegol oxalate
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    Naloxegol oxalate

    CAS:
    <p>Naloxegol oxalate (NKTR-118) is a peripherally-selective opioid antagonist for the treatment of opioid-induced constipation.</p>
    Formula:C36H55NO15
    Purity:99.67% - >99.99%
    Color and Shape:Solid
    Molecular weight:741.83

    Ref: TM-T3355

  • Corydaline
    Targetmol
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    Corydaline

    CAS:
    <p>Corydaline: an isoquinoline alkaloid that aids digestion, has anti-inflammatory and pain relief properties, and inhibits CYP2C19 and CYP2C9.</p>
    Formula:C22H27NO4
    Purity:98.97% - 99.86%
    Color and Shape:Solid
    Molecular weight:369.45

    Ref: TM-T5S2360

  • GR 89696 free base
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    GR 89696 free base

    CAS:
    <p>GR 89696 free base is a potent κ2 opioid receptor agonist with a high selectivity, offering potential benefits in pruritus prevention.</p>
    Formula:C19H25Cl2N3O3
    Color and Shape:Solid
    Molecular weight:414.33

    Ref: TM-T72520

  • Sec-O-Glucosylhamaudol
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    Sec-O-Glucosylhamaudol

    CAS:
    <p>Sec-O-Glucosylhamaudol has anti-inflammatory and strong antinociceptive properties, acting on p38 MAPK and opioid receptors.</p>
    Formula:C21H26O10
    Purity:99.79%
    Color and Shape:Solid
    Molecular weight:438.43

    Ref: TM-T5S0581

  • Nociceptin
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    Nociceptin

    CAS:
    <p>Nociceptin (Orphanin FQ) is a 17-amino-acid polypeptide that is structurally related to the opioid peptide dynorphin A.</p>
    Formula:C79H129N27O22
    Purity:99.35%
    Color and Shape:Solid
    Molecular weight:1809.04

    Ref: TM-TP1071

  • Nociceptin (1-13) amide TFA
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    Nociceptin (1-13) amide TFA

    <p>Nociceptin (1-13), amide: ORL1 receptor agonist, pEC50 7.9 (mouse vas deferens), Ki 0.75 nM (rat forebrain binding).</p>
    Formula:C63H101F3N22O17
    Purity:97.64%
    Color and Shape:Solid
    Molecular weight:1495.61

    Ref: TM-TP1793L

  • MCOPPB
    Targetmol
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    MCOPPB

    CAS:
    <p>MCOPPB: potent, selective nociceptin receptor agonist, pKi 10.07, minor opioid activity, anxiolytic in animals, non-sedative.</p>
    Formula:C26H40N4
    Color and Shape:Solid
    Molecular weight:408.62

    Ref: TM-T21345