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Adenosine Receptor

Adenosine Receptor

Adenosine receptors are a class of GPCRs that respond to the endogenous nucleoside adenosine. These receptors are involved in regulating various physiological processes, including cardiovascular function, sleep-wake cycles, and immune responses. Adenosine receptor modulators have therapeutic potential in treating conditions such as cardiac arrhythmias, inflammation, and neurodegenerative diseases. At CymitQuimica, we provide a selection of high-quality adenosine receptor modulators to support your research in cardiovascular biology, neuroscience, and immunology.

Found 242 products of "Adenosine Receptor"

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  • VUF8507
    Targetmol
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    VUF8507

    CAS:
    <p>Vuf8507 is an allosteric regulator of adenosine receptor.</p>
    Formula:C21H15N3O
    Color and Shape:Solid
    Molecular weight:325.36

    Ref: TM-T35086

  • PD 81723
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    PD 81723

    CAS:
    <p>Allosteric potentiator at the adenosine A1 receptor</p>
    Formula:C14H12F3NOS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:299.31

    Ref: TM-T23130

  • Sipagladenant
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    Sipagladenant

    CAS:
    <p>Sipagladenant: oral inverse agonist for A2A adenosine receptor, may aid frontal lobe dysfunction research.</p>
    Formula:C20H19N3O4S
    Color and Shape:Solid
    Molecular weight:397.45

    Ref: TM-T61876

  • SCH-202676 HBr
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    SCH-202676 HBr

    CAS:
    <p>SCH-202676 HBr is an allosteric agonist. It also an GPCR antagonist.</p>
    Formula:C15H13N3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:267.35

    Ref: TM-T24770

  • A3AR antagonist 2
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    A3AR antagonist 2

    CAS:
    <p>A3AR antagonist 2 is a potent antagonist of the human A3 adenosine receptor, exhibiting a Ki value of 4.54 nM.</p>
    Formula:C22H16N6O3
    Color and Shape:Solid
    Molecular weight:412.4

    Ref: TM-T72588

  • TH-162
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    TH-162

    CAS:
    <p>TH-162 (R)-PIA is an A1 adenosine receptor agonist with ~100× higher affinity than its (+)-isomer.</p>
    Formula:C19H23N5O4
    Color and Shape:Solid
    Molecular weight:385.42

    Ref: TM-T26266

  • PQ-69
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    PQ-69

    CAS:
    <p>PQ-69 is a selective adenosine A1 receptor antagonist with inverse agonist activity.</p>
    Formula:C20H19FN4O
    Color and Shape:Solid
    Molecular weight:350.39

    Ref: TM-T28446

  • MRS 1523
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    MRS 1523

    CAS:
    <p>MRS 1523: selective adenosine A3 antagonist, Ki 18.9/113 nM (human/rat), blocks N-type Ca channels &amp; inhibits action potentials in rat DRG neurons.</p>
    Formula:C23H29NO3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:399.55

    Ref: TM-T16135

  • Inupadenant
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    Inupadenant

    CAS:
    <p>Inupadenant is an orally active, highly selective A2A receptor antagonist. Inupadenant is not brain-penetrant. Inupadenant has potent anti-tumor activity[1].</p>
    Formula:C25H26F2N8O4S2
    Color and Shape:Solid
    Molecular weight:604.65

    Ref: TM-T37014

  • CAY10680
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    CAY10680

    CAS:
    <p>CAY10680 inhibits MAO-B (IC50=34.9 nM) &amp; A2A receptors (Ki=39.5 nM), sparing other adenosine types &amp; MAO-A, may treat Parkinson's.</p>
    Formula:C18H16N2O2S
    Color and Shape:Solid
    Molecular weight:324.4

    Ref: TM-T37354

  • FR-194921
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    FR-194921

    CAS:
    <p>FR-194921: potent oral adenosine A1 antagonist, improves cognition, reduces anxiety, similar efficacy in humans, rats, mice.</p>
    Formula:C23H23N5O
    Color and Shape:Solid
    Molecular weight:385.46

    Ref: TM-T27379

  • CVT-2759
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    CVT-2759

    CAS:
    <p>CVT-2759, potential A(1)-ADOR partial agonist, could slow ventricular rate without severe cardiac side effects.</p>
    Formula:C17H24N6O6
    Color and Shape:Solid
    Molecular weight:408.41

    Ref: TM-T31119

  • Adenosine receptor inhibitor 2
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    Adenosine receptor inhibitor 2

    CAS:
    <p>Compound 14b is a potent AR inhibitor with dual affinity, stronger for A1 (Ki = 52.2 nM) than A2A (Ki = 167 nM) ARs.</p>
    Formula:C17H20BrN5O2
    Color and Shape:Solid
    Molecular weight:406.28

    Ref: TM-T62018

  • Acefylline piperazine
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    Acefylline piperazine

    CAS:
    <p>Acefylline piperazine, a less toxic theophylline derivative, treats asthma and bronchitis by bronchodilation, stimulating respiration and CNS.</p>
    Formula:C9H10N4O4·xC4H10N2
    Color and Shape:Solid
    Molecular weight:562.54

    Ref: TM-T70097

  • JNJ-40255293
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    JNJ-40255293

    CAS:
    <p>JNJ-40255293 is an antagonist of adenosine A2A/A1.</p>
    Formula:C23H22N4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:402.45

    Ref: TM-T24209

  • AK-IN-1
    Targetmol
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    AK-IN-1

    CAS:
    <p>AK-IN-1: competitive adenosine inhibitor, not ATP; inhibits AK 86-89% at 2-10 µM; promising for ischaemia, inflammation, seizure research.</p>
    Formula:C22H21N3O4
    Color and Shape:Solid
    Molecular weight:391.42

    Ref: TM-T73436

  • ATL-801
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    ATL-801

    CAS:
    <p>ATL-801 is anselective antagonist of A2B receptor with herapeutic activity for colitis.</p>
    Formula:C24H25N7O3
    Color and Shape:Solid
    Molecular weight:459.5

    Ref: TM-T26680

  • Kira8 Hydrochloride
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    Kira8 Hydrochloride

    CAS:
    <p>Kira8 Hydrochloride is a mono-selective IRE1α inhibitor that allosterically attenuates IRE1α RNase activity with an IC50 of 5.9 nM.</p>
    Formula:C31H30Cl2N6O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:637.58

    Ref: TM-T11762

  • A2AAR/HDAC-IN-2
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    A2AAR/HDAC-IN-2

    CAS:
    <p>A2AAR/HDAC-IN-2: potent dual A2AAR/HDAC inhib., Ki 10.3 nM, IC50 18.5 nM, anti-tumor potential.</p>
    Formula:C23H26N6O4
    Color and Shape:Solid
    Molecular weight:450.49

    Ref: TM-T62717

  • Theophylline sodium glycinate
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    Theophylline sodium glycinate

    CAS:
    <p>Theophylline sodium glycinate inhibits PDE3, treats asthma/COPD, blocks adenosine receptors, activates HDAC, reduces inflammation and induces apoptosis.</p>
    Formula:C9H12N5NaO4
    Color and Shape:Solid
    Molecular weight:277.216

    Ref: TM-T60511