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Other Inhibitors

Other Inhibitors

This category encompasses a wide variety of inhibitors that do not fit into the standard classifications but are still critical for various biochemical and pharmacological research. These inhibitors may target unique or less-studied pathways, enzymes, and molecular interactions, providing valuable tools for specialized research areas. At CymitQuimica, we offer a diverse selection of high-quality inhibitors across multiple biological targets and research disciplines, enabling you to explore novel therapeutic avenues and deepen your understanding of complex biological processes.

Found 37931 products of "Other Inhibitors"

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  • Defucogilvocarcin V

    CAS:
    <p>Defucogilvocarcin V is an antibiotic with activity against Gram-positive bacteria.</p>
    Formula:C21H16O5
    Color and Shape:Solid
    Molecular weight:348.349
  • SPR7


    <p>SPR7 is a potent and selective rhodesain inhibitor (Ki: 0.51 nM). SPR7 exhibited antiparasitic effects against T. b. brucei (EC50: 1.65 μM).</p>
    Formula:C30H32ClN3O3
    Color and Shape:Solid
    Molecular weight:518.05
  • Pulvilloric acid

    CAS:
    <p>Pulvilloric acid is an antifungal antibiotic produced by the organism Pen. pulvillorum 504.</p>
    Formula:C15H18O5
    Color and Shape:Solid
    Molecular weight:278.30
  • Manumycin E

    CAS:
    <p>Manumycin E exhibits activity against Gram-positive bacteria and Escherichia coli, but has limited effect on other Gram-negative bacteria and none on fungi. It inhibits RAS farnesyltransferase and demonstrates modest cytotoxic activity against the human colorectal cancer cell line [HCT-116].</p>
    Formula:C30H34N2O7
    Color and Shape:Solid
    Molecular weight:534.6
  • ONO-DI-004

    CAS:
    <p>ONO-DI-004 is a selective EP1 Prostanoid receptor agonist.</p>
    Formula:C24H38O6
    Color and Shape:Solid
    Molecular weight:422.55
  • 5-Hydroxymethyltubercidin

    CAS:
    <p>5-Hydroxymethyltubercidin is a semisynthetic antibiotic derived from tubercidin-5-carboxylic acid.</p>
    Formula:C12H16N4O5
    Color and Shape:Solid
    Molecular weight:296.279
  • Phoslactomycin C

    CAS:
    <p>Phoslactomycin C exhibits relatively weak activity against Gram-positive bacteria, but demonstrates stronger antifungal effects.</p>
    Formula:C30H48NO10P
    Color and Shape:Solid
    Molecular weight:613.677
  • Macquarimicin B

    CAS:
    <p>Macquarimicin B is an antibiotic.</p>
    Formula:C22H28O6
    Color and Shape:Solid
    Molecular weight:388.454
  • Endophenazine D

    CAS:
    <p>Endophenazine D is a phenazine-class antibiotic.</p>
    Formula:C15H12N2O4
    Color and Shape:Solid
    Molecular weight:284.27
  • Saframycin D

    CAS:
    <p>Saframycin D exhibits activity against Gram-positive bacteria and shows weaker potency against mycobacteria.</p>
    Formula:C28H31N3O9
    Color and Shape:Solid
    Molecular weight:553.56
  • Espinomycin A3

    CAS:
    <p>Espinomycin A3 is a 16-membered macrolide antibiotic (antibiotic) that exhibits activity against Gram-positive bacteria.</p>
    Formula:C40H65NO15
    Color and Shape:Solid
    Molecular weight:799.942
  • Benadrostin

    CAS:
    <p>Benadrostin is a Poly(ADP-ribose) synthetase inhibitor with an IC50 of 35μM.</p>
    Formula:C8H5NO4
    Color and Shape:Solid
    Molecular weight:179.13
  • Carpetimycin C

    CAS:
    <p>Carpetimycin C exhibits strong activity against both Gram-positive and Gram-negative bacteria, including those that produce β-lactamase. It also has a powerful inhibitory effect on β-lactamase .</p>
    Formula:C14H20N2O6S
    Color and Shape:Solid
    Molecular weight:344.383
  • Mycelianamide

    CAS:
    <p>Mycelianamide is an antibiotic effective against Gram-positive bacteria.</p>
    Formula:C22H28N2O5
    Color and Shape:Solid
    Molecular weight:400.468
  • BI-207524

    CAS:
    <p>BI-207524 is a novel NS5B Thumb Pocket 1 Inhibitor with Improved Potency for the Potential Treatment of Chronic Hepatitis C Virus Infection.</p>
    Formula:C35H36ClN5O5
    Color and Shape:Solid
    Molecular weight:642.14
  • Anti-ToCV agent 1


    <p>Anti-ToCV agent 1 can be used as a potential anti-ToCV drug.</p>
    Formula:C22H19FN2O5S
    Color and Shape:Solid
    Molecular weight:442.46
  • Lividomycin B

    CAS:
    <p>Lividomycin B is an aminoglycoside antibiotic with broad-spectrum activity against bacteria and mycobacteria. It does not exhibit cross-resistance with Streptomyces or Penicillium. Additionally, it offers protective effects in mice infected with Staphylococcus aureus and Pseudomonas aeruginosa.</p>
    Formula:C23H45N5O13
    Color and Shape:Solid
    Molecular weight:599.629
  • Griseorhodin C

    CAS:
    <p>Griseorhodin C is a quinone antibiotic primarily active against both Gram-positive and Gram-negative bacteria.</p>
    Formula:C25H18O13
    Color and Shape:Solid
    Molecular weight:526.40
  • AZ0108

    CAS:
    <p>AZ0108, an oral PARP1,2,6 inhibitor, selectively blocks centrosome clustering, is viable for in vivo studies, and doesn't inhibit PARP3/TNKS1.</p>
    Formula:C24H20F4N6O2
    Color and Shape:Solid
    Molecular weight:500.45
  • Octacosamicin B

    CAS:
    <p>Octacosamicin B exhibits activity against bacteria, yeast, and filamentous fungi, although its antibacterial effectiveness is relatively weak.</p>
    Formula:C32H54N4O9
    Color and Shape:Solid
    Molecular weight:638.793
  • Pluracidomycin D

    CAS:
    <p>Pluracidomycin D, a type of carbapenem antibiotic, exhibits activity against both Gram-positive and Gram-negative bacteria.</p>
    Formula:C9H11NO7S
    Color and Shape:Solid
    Molecular weight:277.25
  • Epithienamycin B

    CAS:
    <p>Epithienamycin B is a natural product isolated from Streptomyces flavoviridis.</p>
    Formula:C13H16N2O5S
    Color and Shape:Solid
    Molecular weight:312.34
  • Rimegepant sulfate hydrate

    CAS:
    <p>Rimegepant (BMS-927711/BHV-3000): oral CGRP blocker for migraines, effective without vasoconstriction, beats placebo, well-tolerated.</p>
    Formula:C56H64F4N12O13S
    Color and Shape:Solid
    Molecular weight:1221.2526
  • PTP1B-IN-18


    <p>PTP1B-IN-18 is an orally active, fully mixed protein tyrosine phosphatase 1B (PTP1B) inhibitor (Ki: 35.2 μM).PTP1B-IN-18 can be used to study type 2 diabetes.</p>
    Formula:C26H19N3O4S
    Color and Shape:Solid
    Molecular weight:469.51
  • Purine phosphoribosyltransferase-IN-1


    <p>Compound (S,R)-48 inhibits Pf, Pv, &amp; Tbr PRT with Ki of 50, 20, 2 nM.</p>
    Formula:C11H15N5Na4O10P2
    Color and Shape:Solid
    Molecular weight:531.17
  • RXR antagonist 1


    <p>RXR antagonist 1 is a Retinoid X Receptor (RXR) modulator that exhibits high RXR antagonism (pA2: 8.06). RXR antagonist 1 can be used to study type 2 diabetes.</p>
    Formula:C28H33F3N2O3
    Color and Shape:Solid
    Molecular weight:502.57
  • BAY-693

    CAS:
    <p>BAY-693 is a ERK5 negative control agent with IC50 (ERK5) = 6400 nM. Its analog, BAY-885, is a potent and selective ERK5 (MAPK7) inhibitor with IC50 of 40 nM</p>
    Formula:C26H30F3N7O2
    Color and Shape:Solid
    Molecular weight:529.56
  • PTP1B-IN-3 diammonium


    <p>PTP1B-IN-3 diammonium, an oral enzyme inhibitor, has potent antidiabetic and anticancer effects, with a 120 nM IC50.</p>
    Formula:C12H13BrF2N3O3P
    Color and Shape:Solid
    Molecular weight:396.12
  • VU0463271 quarterhydrate


    <p>VU0463271 quarterhydrate is a potent KCC2 antagonist, with an IC 50 of 61 nM [1].</p>
    Formula:C19H20N4O2S2
    Color and Shape:Solid
    Molecular weight:387
  • Oleuroside

    CAS:
    <p>Oleuroside can protect against mitochondrial dysfunction in models of early Alzheimer's disease and brain ageing.</p>
    Formula:C25H32O13
    Purity:98%
    Color and Shape:Solid
    Molecular weight:540.51
  • MRS2179 tetrasodium hydrate


    <p>MRS2179 blocks turkey P2Y1 receptor (Kb 102 nM, pA2 6.99), affects platelet aggregation, and has varying IC50s on P2 receptors.</p>
    Formula:C11H15N5Na4O10P2
    Color and Shape:Solid
    Molecular weight:576.21
  • Orvepitant

    CAS:
    <p>Orvepitant is a potent and selective NK1 antagonist, which may be potentially useful for patients with major depressive disorder (MDD), anxiety and insomnia.</p>
    Formula:C31H35F7N4O2
    Color and Shape:Solid
    Molecular weight:628.62
  • Damavaricin D

    CAS:
    <p>Damavaricin D exhibits activity against Gram-positive bacteria, Gram-negative bacteria, and fungi.</p>
    Formula:C38H49NO12
    Color and Shape:Solid
    Molecular weight:711.795
  • PD-1/PD-L1-IN-15


    <p>PD-1/PD-L1-IN-15 is a potent inhibitor of PD-1/PD-L1 (IC50: 60.1 nM) and has shown investigational potential for tumor immunotherapy.</p>
    Formula:C32H30N4O3
    Color and Shape:Solid
    Molecular weight:518.61
  • ABCA1 inducer 1

    CAS:
    <p>ABCA1 inducer 1, a non-lipid inducer of ABCA1, enhances ABCA1 expression in E3/4FAD mice expressing human APOE 3/4, augments the lipidation of apolipoprotein (APOE), and reverses various Alzheimer's disease (AD) phenotypes without increasing triglycerides.</p>
    Formula:C24H24Cl2N2O7S2
    Color and Shape:Solid
    Molecular weight:587.49
  • Bagremycin B

    CAS:
    <p>Bagremycin B is produced by the bacterium Streptomyces strain Tu 4128. It exhibits weak activity against Gram-positive bacteria, Saccharomyces cerevisiae, and Candida albicans.</p>
    Formula:C17H15NO4
    Color and Shape:Solid
    Molecular weight:297.305
  • Ezomycin A1

    CAS:
    <p>Ezomycin A1 is an antifungal antibiotic effective primarily against plant pathogens such as Sclerotinia and Botrytis. It is used to prevent and control diseases like Sclerotinia rot, gray mold, and candidiasis in crops.</p>
    Formula:C26H38N8O15S
    Color and Shape:Solid
    Molecular weight:734.69
  • Hydroxyakalone

    CAS:
    <p>Hydroxyakalone is an inhibitor of the enzyme xanthine oxidase (XOD, EC 1.2.3.2) and has an IC50 of 4.6 μM for XOD.</p>
    Formula:C5H5N5O2
    Color and Shape:Solid
    Molecular weight:167.126
  • Unoprostone isopropyl

    CAS:
    <p>Unoprostone isopropyl, a prostanoid and synthetic docosanoid, is approved for the treatment of ocular hypertension and open-angle glaucoma.</p>
    Formula:C25H44O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:424.61
  • 1-Hydroxy-2-nonyn-4-one

    CAS:
    <p>1-Hydroxy-2-nonyn-4-one is an antibiotic with activity against yeasts, filamentous fungi, tumors, and shows weak efficacy against both Gram-positive and Gram-negative bacteria.</p>
    Formula:C9H14O2
    Color and Shape:Solid
    Molecular weight:154.206
  • AH22921

    CAS:
    <p>AH22921 is an EP4 prostaglandin receptor antagonist with the ability to antagonize the activation of adenylyl cyclase by prostaglandins in CHO cells. It induces a rightward shift in the PGE? concentration-response curve in these cells, functioning as a non-competitive antagonist. AH22921 is selective for the EP4 receptor, inhibiting its activity in CHO cells without affecting the PGE? concentration-response curve in NPE cells that contain the EP2 receptor.</p>
    Formula:C29H35NO5
    Color and Shape:Solid
    Molecular weight:477.59
  • TIY-7


    <p>TIY-7 is a selective, orally active inhibitor of the promyosin receptor kinase (TRK) enzyme. TIY-7 exhibited anti-tumour effects in a mouse xenograft model.</p>
    Color and Shape:Solid
  • Sdz 210-096

    CAS:
    <p>Sdz 210-096: a 14 beta-benzyl morphinan, mu/kappa opiate receptor antagonist, stimulates LH secretion in rats.</p>
    Formula:C27H31NO2
    Color and Shape:Solid
    Molecular weight:401.54
  • WS-898


    <p>WS-898 boosts paclitaxel efficacy in resistant cells by inhibiting ABCB1; IC50: SW620/Ad300 - 5.0 nM, KB-C2 - 3.67 nM, HEK293/ABCB1 - 3.68 nM.</p>
    Formula:C33H25N7OS
    Color and Shape:Solid
    Molecular weight:567.66
  • SARS-CoV-2-IN-99

    CAS:
    <p>SARS-CoV-2-IN-99 (compound 58) is an inhibitor of the main protease of SARS-CoV-2.</p>
    Formula:C20H16Br2NO4P
    Color and Shape:Solid
    Molecular weight:525.13
  • MRS4865

    CAS:
    <p>MRS4865 (compound 7a) serves as a chimeric antagonist for the P2Y14 receptor and an agonist for UDP-glucose, offering protection against neuropathic pain.</p>
    Formula:C39H39F3N4O7
    Color and Shape:Solid
    Molecular weight:732.74
  • Calphostin D

    CAS:
    <p>Calphostins, PKC inhibitors from Cladosporium cladosporioides, include A, B, C, D, I; C is most potent.</p>
    Formula:C30H30O10
    Color and Shape:Solid
    Molecular weight:550.55
  • Oral antiplatelet agent 1

    CAS:
    <p>Oral antiplatelet agent 1 is a potent antiplatelet agent with an IC50 of 2.94 μM in vitro.</p>
    Formula:C23H24N4O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:468.53
  • Fujianmycin A

    CAS:
    <p>Fujianmycin A exhibits activity against Bacillus subtilis (hay bacillus).</p>
    Formula:C19H14O5
    Color and Shape:Solid
    Molecular weight:322.311
  • hTrkA-IN-2


    <p>hTrkA-IN-2 is a selective hTrkA metamorphosis inhibitor (IC50: 3.9 nM).</p>
    Formula:C24H22F3N5O3
    Color and Shape:Solid
    Molecular weight:485.46
  • PEN-866

    CAS:
    <p>PEN-866, a conjugate of HSP90i and SN-38, may control early NSCLC tumor growth.</p>
    Formula:C49H49N7O9
    Color and Shape:Solid
    Molecular weight:879.95
  • Griseusin B

    CAS:
    <p>Griseusin B is a quinone antibiotic primarily effective against Gram-positive bacteria.</p>
    Formula:C22H22O10
    Color and Shape:Solid
    Molecular weight:446.404
  • Epoxyquinomicin C

    CAS:
    <p>Epoxyquinomicin C is an antibiotic that can be isolated from Amycolatopsis sp. It exhibits anti-inflammatory properties against collagen-induced arthritis and is also utilized in the synthesis of the NF-κB inhibitor DHMEQ.</p>
    Formula:C14H13NO6
    Color and Shape:Solid
    Molecular weight:291.256
  • Metocurine chloride

    CAS:
    <p>Metocurine: a muscle relaxant, not for kidney failure patients as it's kidney-excreted.</p>
    Formula:C40H48Cl2N2O6
    Color and Shape:Solid
    Molecular weight:723.72
  • Acetoxycycloheximide

    CAS:
    <p>Acetoxycycloheximide triggers TNF receptor 1, prompts apoptosis, and cytochrome c release by activating c-Jun N-terminal kinase.</p>
    Formula:C17H25NO6
    Color and Shape:Solid
    Molecular weight:339.38
  • (R)-NVS-ZP7-4

    CAS:
    <p>(R)-NVS-ZP7-4, an R-isomer, inhibits ZIP7 to study ER zinc impact &amp; Notch pathway.</p>
    Formula:C28H28FN5OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:501.62
  • (±)-ANAP hydrochloride (1185251-08-4 free base)


    <p>(±)-ANAP hydrochloride is the amino acid analog of prodan. It can be used as a fluorescent probes and enhance environmental sensitivity.</p>
    Formula:C15H17ClN2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:308.76
  • DDCPPB-Glu

    CAS:
    <p>DDCPPB-Glu is a 6-5 fused ring heterocycle antifolate that shows antitumor activity.</p>
    Formula:C22H27N5O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:441.48
  • Ceclazepide

    CAS:
    <p>Ceclazepide is an antagonist of cholecystokinin receptor.</p>
    Formula:C30H32N6O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:556.61
  • DMP 728

    CAS:
    <p>DMP 728 is an antagonist of Glycoprotein IIb-IIIa.</p>
    Formula:C26H40N8O10S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:656.71
  • SORT1-IN-3

    CAS:
    <p>SORT1-IN-3 (compound 5) is a SORT1 inhibitor characterized by its ability to permeate the blood-brain barrier.</p>
    Formula:C16H26ClNO3
    Color and Shape:Solid
    Molecular weight:315.84
  • PD 113271

    CAS:
    <p>PD 113,271 is an analog of the fermentation products fostriecin with antitumor activity in vitro and in vivo.</p>
    Formula:C19H27O10P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:446.39
  • Adecypenol

    CAS:
    <p>Adecypenol is a unique adenosine deaminase inhibitor. It shows effective inhibitory activity against calf intestinal adenosine deaminase.</p>
    Formula:C12H16N4O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:280.28
  • MDK-3298

    CAS:
    <p>MDK-3298 is a reversible covalent inhibitor of Mcl-1, a target of protein-protein interaction (PPI).</p>
    Formula:C35H32BN3O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:617.46
  • PF-06462894

    CAS:
    <p>PF-06462894: morpholinopyrimidone, mGlu5 antagonist (Ki=6nM), no immune activation in mouse model.</p>
    Formula:C18H23N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:329.39
  • L 671776

    CAS:
    <p>L 671776 is an inositol monophosphatase inhibitor.</p>
    Formula:C23H32O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:388.5
  • L-Tyrosyl-L-glutamic acid

    CAS:
    <p>L-Tyrosyl-L-glutamic acid acts as an inhibitor of the amino acid permease GAP1.</p>
    Formula:C14H18N2O6
    Color and Shape:Solid
    Molecular weight:310.3
  • BRD-9526

    CAS:
    <p>BRD-9526 is a potent and selective inhibitor of Sonic Hedgehog (Shh).</p>
    Formula:C26H31Cl2N3O6S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:584.51
  • L 767679

    CAS:
    <p>L 767679 is an antagonist of the fibrinogen receptors.</p>
    Formula:C20H24N4O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:384.43
  • Azicemicin A

    CAS:
    <p>Azicemicin A exhibits mild antibacterial activity and shows no acute toxicity when administered via intraperitoneal injection to mice at a dosage of 150 mg/kg.</p>
    Formula:C23H25NO9
    Color and Shape:Solid
    Molecular weight:459.446
  • SSR-182289A (Free)

    CAS:
    <p>SSR-182289A (Free) is a thrombin inhibitor.</p>
    Formula:C30H33F2N5O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:597.68
  • Dinordrin

    CAS:
    <p>Dinordrin is an implantation inhibitor and hormone.</p>
    Formula:C27H36O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:424.57
  • Polyoxin K

    CAS:
    <p>Polyoxin K is a nucleoside antifungal antibiotic that exhibits significant effectiveness against rice sheath blight.</p>
    Formula:C22H30N6O13
    Molecular weight:586.51
  • Retelliptine

    CAS:
    <p>Retelliptine, a DNA topoisomerase II inhibitor, is used potentially for the treatment of cancer.</p>
    Formula:C25H32N4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:404.55
  • L 739749

    CAS:
    <p>L 739749 is a CAAX peptidomimetic. It is also an inhibitor of farnesyl-protein transferase.</p>
    Formula:C24H41N3O6S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:531.73
  • Naltalimide

    CAS:
    <p>Naltalimide: µ-opioid receptor partial agonist, improves bladder storage by affecting spinal cord reflex.</p>
    Formula:C28H28N2O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:472.53
  • Pamiparib maleate

    CAS:
    <p>Pamiparib (BGB-290) is a selective PARP inhibitor that blocks DNA repair and promotes apoptosis.</p>
    Formula:C44H42F2N8O14
    Purity:98%
    Color and Shape:Solid
    Molecular weight:944.859
  • Ambelline

    CAS:
    <p>Ambelline has antitumor activity.</p>
    Formula:C18H21NO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:331.36
  • MCTR1

    CAS:
    <p>MCTR1, a pro-resolving mediator derived from DHA, promotes tissue repair and reduces inflammation by enhancing phagocytosis and decreasing eicosanoids.</p>
    Formula:C32H47N3O9S
    Color and Shape:Solid
    Molecular weight:649.8
  • G-9791

    CAS:
    <p>G-9791 is an effective and selective inhibitor of group-I PAK.</p>
    Formula:C26H26ClFN6O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:508.98
  • LY 190388

    CAS:
    <p>LY 190388 is a penicillamine-containing enkephalin analog used as an mu receptor agonist with analgesia activity.</p>
    Formula:C30H41N5O7S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:615.74
  • Emd 52297

    CAS:
    <p>Emd 52297 is an inhibitor of renin.</p>
    Formula:C39H59N11O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:793.96
  • UTPγS trisodium salt

    CAS:
    <p>P2Y2 and P2Y4 receptor agonist</p>
    Formula:C9H12N2Na3O14P3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:566.15
  • AFP-07 free acid

    CAS:
    <p>AFP 07 free acid is a 7,7-difluoroprostacyclin derivative. It also acts as a selective and highly potent agonist for the IP receptor.</p>
    Formula:C22H30F2O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:412.47
  • Bagremycin A

    CAS:
    <p>Bagremycin A is identified in the actinobacterium strain Streptomyces (Streptomyces) Tu 4128. It exhibits weak antimicrobial activity against Gram-positive bacteria, Saccharomyces cerevisiae, and Candida albicans.</p>
    Formula:C15H13NO3
    Color and Shape:Solid
    Molecular weight:255.269
  • KT5926

    CAS:
    <p>KT5926 selectively inhibits myosin light chain kinase and NGF-dependent neurite growth; it's a K-252a analogue.</p>
    Formula:C30H27N3O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:525.55
  • NPEC-caged-(S)-3,4-DCPG

    CAS:
    <p>mGlu8a agonist</p>
    Formula:C19H16N2O10
    Purity:98%
    Color and Shape:Solid
    Molecular weight:432.34
  • KDOAM-25 trihydrochloride (2230731-99-2 free base)


    <p>KDOAM-25 trihydrochloride, a selective KDM5 inhibitor (IC50: 19-71 nM), boosts H3K4 methylation and hinders MM1S cell growth.</p>
    Formula:C15H28Cl3N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:416.77
  • AFP-07

    CAS:
    <p>AFP-07 is a highly selective and potent agonist. It was used for the prostacyclin receptor.</p>
    Formula:C22H29F2NaO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:434.45
  • L 731735

    CAS:
    <p>L 731735 is a farnesyltransferase inhibitor.</p>
    Formula:C19H40N4O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:420.61
  • Pralatrexate, (R)-

    CAS:
    <p>Pralatrexate is a high-affinity DHFR inhibitor targeting RFC-1, used in cancer treatment and immunosuppression.</p>
    Formula:C23H23N7O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:477.47
  • Antiproliferative agent-3


    <p>Antiproliferative agent-3 (comp 4) exhibits potent growth inhibitory effects against MCF-7 cells with IC 50 of 0.19 nM [1].</p>
    Formula:C11H12N2O5S
    Color and Shape:Solid
    Molecular weight:284.29
  • ROPA

    CAS:
    <p>ROPA, a potent PKCalpha and PKCgamma activator, promotes tumor growth through PKC-activation.</p>
    Formula:C28H32O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:464.55
  • AT1R antagonist 2


    <p>AT1R antagonist 2 is a potent AT1R selective ligand with good AT1R affinity (Ki: 26 nM).</p>
    Formula:C29H37N5O4S2
    Color and Shape:Solid
    Molecular weight:583.77
  • Squalestatin 2

    CAS:
    <p>Squalestatin 2 is an inhibitor of squalene synthase.</p>
    Formula:C33H44O13
    Purity:98%
    Color and Shape:Solid
    Molecular weight:648.69
  • PrCP-7414

    CAS:
    <p>PrCP-7414 is a potent PrCP inhibitor, CAS# 1252037-41-4, named after the CAS number's last four digits.</p>
    Formula:C31H33Cl2N5O2
    Color and Shape:Solid
    Molecular weight:578.53
  • MI-1851

    CAS:
    <p>MI-1851 is a potent peptidomimetic inhibitor. MI-1851could prevent proteolytic processing of the S protein from SARSCoV-2 by endogenous furin in HEK293 cells.</p>
    Formula:C34H53N15O6
    Color and Shape:Solid
    Molecular weight:767.88
  • Cryptopleurine

    CAS:
    <p>Cryptopleurine is an inhibitor of gene products associated with cell proliferation, survival, invasion and angiogenesis. It acts by targeting the NF-κB pathway.</p>
    Formula:C24H27NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:377.48
  • BMS-751324

    CAS:
    <p>BMS-751324: p38α MAPK inhibitor with carbamyl-methyl, esters, phosphate from HPA. Reduces rat arthritis swelling and TNFα.</p>
    Formula:C32H35N6O10P
    Color and Shape:Solid
    Molecular weight:694.63
  • VEGFR-2-IN-10


    <p>VEGFR-2-IN-10 has enhanced antiangiogenic potency against VEGFR2 phosphorylation induced by VEGF with an IC50 value of 0.7 μM and no cytotoxic effects.</p>
    Formula:C20H21N3O2
    Color and Shape:Solid
    Molecular weight:335.4
  • ATR-IN-7

    CAS:
    <p>ATR-IN-7 is a potent inhibitor of ATR.</p>
    Formula:C21H22FN7O
    Color and Shape:Solid
    Molecular weight:407.44
  • TEI-9063

    CAS:
    <p>TEI-9063 is a stable and highly specific prostacyclin analogue of prostacyclin receptor in mast cell tumor p-815 cells.</p>
    Formula:C23H38O4
    Color and Shape:Solid
    Molecular weight:378.55
  • Enpp-1-IN-12


    <p>ENPP1-IN-12 is a potent, oral ENPP1 inhibitor with a Ki of 41 nM and anti-tumor properties.</p>
    Formula:C17H19N5O3S
    Color and Shape:Solid
    Molecular weight:373.43
  • PAD-IN-2

    CAS:
    <p>PAD-IN-2, potent PAD4 inhibitor, IC50 &lt;1 μM; targets autoimmune/cancer disorders.</p>
    Formula:C27H28ClN5O2
    Color and Shape:Solid
    Molecular weight:490
  • FPR2 agonist 2


    <p>Potent FPR2 agonist, crosses blood-brain barrier, EC50: 0.13 nM; reduces inflammation and mitochondrial dysfunction, inhibits caspase-3.</p>
    Formula:C25H20F2N4O2
    Color and Shape:Solid
    Molecular weight:446.45
  • PD-1/PD-L1-IN-16


    <p>PD-1/PD-L1-IN-16 is a potent inhibitor of PD-1/PD-L1 (IC50: 53.2 nM) and has shown research potential for tumour immunotherapy.</p>
    Formula:C34H30N4O4
    Color and Shape:Solid
    Molecular weight:558.63
  • Basroparib

    CAS:
    <p>Basroparib is an inhibitor of ribose polymerase (PARP) and has shown antitumour effects.</p>
    Formula:C18H21F2N7O3
    Color and Shape:Solid
    Molecular weight:421.4
  • EP4 receptor antagonist 2

    CAS:
    <p>EP4 receptor antagonist 2 (compound 2-13) is a potent agonist of the EP4 receptor (IC50: 7.8 nM) and has antitumour effects.</p>
    Formula:C27H29N3O5
    Color and Shape:Solid
    Molecular weight:475.54
  • Sapintoxin D

    CAS:
    <p>Sapintoxin D is a fluorescent phorbol ester and selective activator of protein kinase C.</p>
    Formula:C30H37NO8
    Color and Shape:Solid
    Molecular weight:539.62
  • Anti-TSWV agent 1


    <p>Anti-TSWV agent 1 is a highly effective inactivator (EC50:144 μg/mL) of tomato spotted wilt virus (TSWV).</p>
    Formula:C22H27ClN4OS3
    Color and Shape:Solid
    Molecular weight:495.12
  • ONO-AE1-259 lysine

    CAS:
    <p>ONO-AE1-259 is a highly selective agonist of prostaglandin e2 receptor (ep2)</p>
    Formula:C28H49ClN2O6
    Color and Shape:Solid
    Molecular weight:545.15
  • Enpp-1-IN-11


    <p>Enpp-1-IN-11 inhibits ENPP1 with a 45 nM Ki, is plasma stable, and has low clearance in human/mouse livers, potentially aiding cancer research.</p>
    Formula:C15H15N5O3S
    Color and Shape:Solid
    Molecular weight:345.38
  • Ranakinin

    CAS:
    <p>Ranakinin is a novel tachykinin receptor agonist; from the brain of frog, Rana ridibunda.</p>
    Formula:C62H95N17O15S
    Color and Shape:Solid
    Molecular weight:1350.59
  • Iroxanadine hydrobromide

    CAS:
    <p>Iroxanadine hydrobromide is a MAPK p38 inhibitor potentially for the treatment of atherosclerosis.</p>
    Formula:C14H21BrN4O
    Color and Shape:Solid
    Molecular weight:341.25
  • NB-216

    CAS:
    <p>NB-216 is a macrocyclic peptidic BACE-1 inhibitor.</p>
    Formula:C35H45N3O4
    Color and Shape:Solid
    Molecular weight:571.75
  • M-89 MLL inhibitor

    CAS:
    <p>M-89, a potent Menin-MLL blocker: Kd 1.4 nM, IC50 25 nM for MV4;11 cells, 55 nM for MOLM-13, &gt;100x selective over HL-60.</p>
    Formula:C37H47N5O4S
    Color and Shape:Solid
    Molecular weight:657.87
  • Flusoxolol

    CAS:
    <p>Flusoxolol is a beta-adrenoceptor partial agonist.</p>
    Formula:C22H30FNO4
    Color and Shape:Solid
    Molecular weight:391.48
  • Cilengitide hydrochloride

    CAS:
    <p>Cilengitide hydrochloride is a salt that may combat cancer by blocking specific integrins, disrupting cell interactions and angiogenesis.</p>
    Formula:C27H41ClN8O7
    Color and Shape:Solid
    Molecular weight:625.12
  • PDE4B/7A-IN-1

    CAS:
    <p>5-HT1A antagonist; Ki=8nM, Kb=0.04nM. PDE4B IC50=80.4μM; PDE7A IC50=151.3μM. Good biofilm penetration, stable, anticognitive, antidepressant.</p>
    Formula:C25H35N3O3
    Color and Shape:Solid
    Molecular weight:425.56
  • Topoisomerase II inhibitor 6


    <p>Topoisomerase II inhibitor 6, a potent tryptanthrin derivative, blocks G2 phase in CCRF-CEM cells, induces DNA breaks, and may be used for cancer research.</p>
    Formula:C19H18N4O2
    Color and Shape:Solid
    Molecular weight:334.37
  • Antitumor agent-47


    <p>Antitumor agent-47, a silibinin derivative, shows cytotoxicity in NCI-H1299 (IC50: 8.07µM) and HT29 (IC50: 6.27µM) cells.</p>
    Formula:C30H27NO11
    Color and Shape:Solid
    Molecular weight:577.54
  • Brostallicin HCl

    CAS:
    <p>Brostallicin, a synthetic MGB, inhibits DNA replication in cancer cells, inducing cell death, effective against MMR-defective tumors.</p>
    Formula:C30H36BrClN12O5
    Color and Shape:Solid
    Molecular weight:760.04
  • MRS2279 diammonium

    CAS:
    <p>MRS2279 diammonium, a P2Y1 antagonist with K i 2.5 nM, IC 50 51.6 nM, blocks ADP-induced platelet aggregation, pK b 8.05.</p>
    Formula:C13H24ClN7O8P2
    Color and Shape:Solid
    Molecular weight:503.77
  • Xylarianaphthol-1

    CAS:
    <p>Xylarianaphthol-1 is an activator of p21 promoter in a p53-independent manner.</p>
    Formula:C16H20BrFN2O2
    Color and Shape:Solid
    Molecular weight:371.24
  • FTI-2628

    CAS:
    <p>FTI-2628 is a novel inhibitor of protein farnesyltransferase (FT), inhibiting the growth of P. falciparum in red blood cells and suppressing parasitemia.</p>
    Formula:C31H34N4O3S
    Color and Shape:Solid
    Molecular weight:542.69
  • B-3852

    CAS:
    <p>B-3852 is a Bradykinin inhibitor.</p>
    Formula:C55H74F3N15O11
    Color and Shape:Solid
    Molecular weight:1178.27
  • LY3325656

    CAS:
    <p>LY3325656, a GPR142 agonist with anti-diabetic properties, progresses to phase 1 trials for Type 2 diabetes.</p>
    Formula:C21H23F3N6O2
    Color and Shape:Solid
    Molecular weight:448.44
  • 7(Z),11(Z)-Nonacosadiene

    CAS:
    <p>7(Z),11(Z)-Nonacosadiene, a female fly pheromone, spurs male courtship; it's a C29 diene made by a female-specific elongase.</p>
    Formula:C29H56
    Color and Shape:Solid
    Molecular weight:404.75
  • VEGFR-2-IN-26

    CAS:
    <p>VEGFR-2-IN-26 inhibits VEGFR-2 (IC50: 15.5 nM), combating various cancers' cell growth.</p>
    Formula:C24H19F3N6O2
    Color and Shape:Solid
    Molecular weight:480.44
  • Antitumor agent-51


    <p>Antitumor agent-51 targets osteosarcoma with 21.9 nM IC50, high selectivity, and low toxicity.</p>
    Formula:C23H25N5O2S
    Color and Shape:Solid
    Molecular weight:435.54
  • Polyozellin

    CAS:
    <p>Polyozellin is a prolyl endopeptidase inhibitor with properties effective against inflammation, cancer, and diseases related to oxidative stress.</p>
    Formula:C22H14O10
    Color and Shape:Solid
    Molecular weight:438.341
  • SK&amp;F 108361

    CAS:
    <p>SK&amp;F 108361 is a symmetric diol that binds HIV-1 protease symmetrically.</p>
    Formula:C24H48N6O6
    Color and Shape:Solid
    Molecular weight:516.67
  • MV061194

    CAS:
    <p>MV061194 is a potent and selective cathepsin K (Cat K) inhibitor.</p>
    Formula:C28H37N5O4S
    Color and Shape:Solid
    Molecular weight:539.69
  • CXCR4 probe 1

    CAS:
    <p>CXCR4 probe 1, a specific PET tracer, targets CXCR4 with antagonist TN14003 (IC50: 6.9 nM), aiding in imaging CXCR4-related diseases and tumors.</p>
    Formula:C24H30FN5O4S
    Color and Shape:Solid
    Molecular weight:502.59
  • OPN expression inhibitor 1

    CAS:
    <p>OPN expression inhibitor 1 is an osteopontin expression inhibitor used in the study of breast cancer metastasis.</p>
    Formula:C25H33N3O5
    Purity:99.78%
    Color and Shape:Solid
    Molecular weight:455.55
  • Difeterol

    CAS:
    <p>Difeterol is a biochemical.</p>
    Formula:C25H29NO2
    Color and Shape:Solid
    Molecular weight:375.50
  • Chitinase-IN-5


    <p>Chitinase-IN-5 (8i) blocks OfChi-h (IC50: 0.051 μM), has insecticidal qualities, useful for eco-friendly pest control.</p>
    Formula:C20H21ClFN7
    Color and Shape:Solid
    Molecular weight:413.88
  • Fluperolone acetate

    CAS:
    <p>Fluperolone acetate is a Glucocorticoid/Adrenal Cortex Hormone.</p>
    Formula:C24H31FO6
    Color and Shape:Solid
    Molecular weight:434.50
  • Diatretyne Ⅰ

    CAS:
    <p>Diatretyne I (Diatretyne amide) exhibits mild activity against Gram-positive bacteria.</p>
    Formula:C8H5NO3
    Color and Shape:Solid
    Molecular weight:163.13
  • Steroid sulfatase/17β-HSD1-IN-1


    <p>Steroid sulfatase/17β-HSD1-IN-1 is a highly effective inhibitor of both steroid sulfatase and 17β-hydroxysteroid dehydrogenase type 1 (17β-HSD1) activities,</p>
    Formula:C19H18N2O5S
    Color and Shape:Solid
    Molecular weight:386.42
  • TLN-232

    CAS:
    <p>TLN-232, a synthetic heptapeptide, may inhibit cancer by targeting M2PK to disrupt tumor cell energy production.</p>
    Formula:C36H49N9O7S2
    Color and Shape:Solid
    Molecular weight:783.96
  • Dermostatin A

    CAS:
    <p>Dermostatin A is a polyene antibiotic with antifungal properties suitable for studying fungal infections.</p>
    Formula:C40H64O11
    Color and Shape:Solid
    Molecular weight:720.93
  • AY 17,605

    CAS:
    <p>AY 17,605 is an inhibitor of bovine heart and rat brain nucleoside-3',5'- monophosphate phosphodiesterase.</p>
    Formula:C25H36O5
    Color and Shape:Solid
    Molecular weight:416.55
  • Epiderstatin

    CAS:
    <p>Epiderstatin is isolated from Streptomyces pulveraceus subsp. epiderstagenes; inhibits mitogenic activity of epidermal growth factor.</p>
    Formula:C15H20N2O4
    Color and Shape:Solid
    Molecular weight:292.33
  • Antcin B

    CAS:
    <p>Antcin B is an inhibitor of SARS-CoV-2 3-chymotrypsin-like protease (3CL Pro). It interacts with several crucial amino acid residues of 3CL Pro, including Leu141, Asn142, Glu166, and His163, through hydrogen bonding, salt bridges, and hydrophobic interactions, thereby inhibiting its activity. This inhibition blocks the cleavage of viral polyproteins and suppresses the replication of the SARS-CoV-2 virus within host cells. Antcin B shows potential for research in the context of COVID-19.</p>
    Formula:C29H40O5
    Color and Shape:Solid
    Molecular weight:468.625
  • [R-(Z)]-4-Amino-3-chloro-2-pen-tenedioicacid

    CAS:
    <p>[R-(Z)]-4-Amino-3-chloro-2-pentenedioic acid inhibits Micrococcus luteus.</p>
    Formula:C5H6ClNO4
    Color and Shape:Solid
    Molecular weight:179.56
  • Enpp-1-IN-7


    <p>Enpp-1-IN-7: potent enpp-1 inhibitor, broad specificity, potential in cancer/infectious disease research. (WO2021203772A1)</p>
    Formula:C18H19N7O4S
    Color and Shape:Solid
    Molecular weight:429.45
  • LLS30

    CAS:
    <p>LLS30 inhibits Gal-1, reduces its binding affinity, and may help treat advanced prostate cancer.</p>
    Formula:C34H33Cl4N5O3
    Color and Shape:Solid
    Molecular weight:701.47
  • Porothramycin B

    CAS:
    <p>Porothramycin B is an antibiotic with activity against Gram-positive bacteria and anaerobes.</p>
    Formula:C19H23N3O4
    Color and Shape:Solid
    Molecular weight:357.404
  • MRS-2339

    CAS:
    <p>MRS-2339 is a P2X receptor activator.</p>
    Formula:C12H15ClN5O6P
    Color and Shape:Solid
    Molecular weight:391.70
  • 6"'-Deamino-6"'-hydroxyneomycin B

    CAS:
    <p>6"'-Deamino-6"'-hydroxyneomycin B is an aminoglycoside antibiotic produced by [Streptomyces fradiaeUC 75]. It is effective against both Gram-positive and Gram-negative bacteria and serves as an intermediate in the biosynthesis of neomycin.</p>
    Formula:C23H45N5O14
    Color and Shape:Solid
    Molecular weight:615.628
  • SHR0687

    CAS:
    <p>SHR0687: potent KOR agonist, selective, favorable PK, effective in rat pain model, minimal BBB penetration, less CNS side effects.</p>
    Formula:C39H60N8O5
    Color and Shape:Solid
    Molecular weight:720.94
  • STING agonist-7


    <p>STING agonist-7 is an agonist of non-nucleotide STING that binds selectively to mouse STING but not human STING [1].</p>
    Formula:C17H12N4O4
    Color and Shape:Solid
    Molecular weight:336.3
  • Granaticin B

    CAS:
    <p>Granaticin B inhibits the initial phase of RNA biosynthesis and exhibits activity against Gram-positive bacteria, mycobacteria (weak), and Trichomonas vaginalis, along with the ability to suppress tumor cells.</p>
    Formula:C28H30O12
    Color and Shape:Solid
    Molecular weight:558.531
  • AX15910


    <p>AX15910 is a potent inhibitor of BRD4 and ERK5.</p>
    Formula:C32H38N6O3
    Color and Shape:Solid
    Molecular weight:554.7
  • Haliangicin B

    CAS:
    <p>Haliangicin B exhibits activity against filamentous fungi and is also effective against oomycetes, but it does not possess any antibacterial properties.</p>
    Formula:C22H32O5
    Color and Shape:Solid
    Molecular weight:376.49
  • Epelmycin D

    CAS:
    <p>Epelmycin D exhibits activity against both Gram-positive and Gram-negative bacteria, as well as Candida albicans, and demonstrates efficacy against leukemia (L1210).</p>
    Formula:C30H35NO11
    Color and Shape:Solid
    Molecular weight:585.599
  • Kaitocephalin

    CAS:
    <p>Kaitocephalin: naturally occurring, non-selective antagonist blocking glutamate receptors, made by Eupenicillium shearii fungus.</p>
    Formula:C18H21Cl2N3O9
    Color and Shape:Solid
    Molecular weight:494.28
  • MK-1220

    CAS:
    <p>MK-1220 is a novel Macrocyclic Inhibitor of Hepatitis C Virus NS3/4A Protease with Improved Preclinical Plasma Exposure.</p>
    Formula:C40H53N5O9S
    Color and Shape:Solid
    Molecular weight:779.94
  • Pluracidomycin C2

    CAS:
    <p>Pluracidomycin C2 is a carbapenem antibiotic with activity against both Gram-positive and Gram-negative bacteria.</p>
    Formula:C11H15NO9S2
    Color and Shape:Solid
    Molecular weight:369.37
  • LAF-153

    CAS:
    <p>LAF-153 is a reversible Methionine Aminopeptidase‑2 (MetAP-2) Inhibitor.</p>
    Formula:C18H32N2O7
    Color and Shape:Solid
    Molecular weight:388.46
  • STA 2

    CAS:
    <p>STA 2 is an analogue of TXA2, a thromboxane receptor in the colonic epithelium.</p>
    Formula:C21H34O3S
    Color and Shape:Solid
    Molecular weight:366.56
  • Plagiochilin A

    CAS:
    <p>Plagiochilin A Inhibits Cytokinetic Abscission and Induces Cell Death</p>
    Formula:C15H14O7
    Color and Shape:Solid
    Molecular weight:306.27
  • RDN2150

    CAS:
    <p>RDN2150 (Compound 25), a ZAP-70 inhibitor with an IC50 of 14.6 nM, covalently binds to the C346 residue of ZAP-70, suppressing the expression of CD25 and CD69</p>
    Formula:C28H29ClN8O4
    Color and Shape:Solid
    Molecular weight:577.03
  • EBOV-GP-IN-1


    <p>EBOV-GP-IN-1 (Compound 28) is a potent inhibitor of Ebola entry, acting on the Ebola virus envelope glycoprotein (EBOV-GP) (IC50: 0.05 μM).</p>
    Formula:C25H40ClN3O2
    Color and Shape:Solid
    Molecular weight:450.06
  • BMS-961955

    CAS:
    <p>BMS-961955 is an allosteric inhibitor of the hepatitis C virus NS5B polymerase.</p>
    Formula:C37H43FN4O4S
    Color and Shape:Solid
    Molecular weight:658.83
  • AN-12-H5

    CAS:
    <p>AN-12-H5 is an anti-enteroviral compound that targets the replication process of PV and EV71 viruses.</p>
    Formula:C24H23N3O4S3
    Color and Shape:Solid
    Molecular weight:513.65
  • Ac-ATS010-KE

    CAS:
    <p>Ac-ATS010-KE is a novel Selective, irreversible, and Rapid Cell-Permeable Inhibitor of Human Caspase-3.</p>
    Formula:C43H41F5N6O12S
    Color and Shape:Solid
    Molecular weight:960.88
  • 11-Demethyltomaymycin

    CAS:
    <p>11-Demethyltomaymycin is an antibiotic that exhibits antiviral activity against Escherichia coli T1 and T3 bacteriophages, along with antibacterial properties against Gram-positive bacteria. Furthermore, it shows cytotoxic effects on leukemia L1210 cells.</p>
    Formula:C15H18N2O4
    Color and Shape:Solid
    Molecular weight:290.314
  • 17β-HSD1-IN-1


    <p>17β-HSD1-IN-1 (Compound 1) can be used in the non-small cell lung cancer (NSCLC) research.</p>
    Formula:C21H21NO3
    Color and Shape:Solid
    Molecular weight:335.4
  • LASSBio-1632


    <p>LASSBio-1632: Novel anti-asthmatic, blocks PDE4A/D, reduces AHR &amp; lung TNF-α, crosses BBB.</p>
    Formula:C18H20N2O6S
    Color and Shape:Solid
    Molecular weight:392.43
  • Antitumor agent-48


    <p>Antitumor agent-48, a 2,3-dehydrosilybin derivative, exhibits cytotoxicity on MCF-7, NCI-H1299, HepG2, HT29 cells; IC50 ranging 8.06-16.51 µM.</p>
    Formula:C35H34N2O14
    Color and Shape:Solid
    Molecular weight:706.65
  • Henagliflozin

    CAS:
    <p>Henagliflozin (SHR3824): an oral, selective SGLT2 inhibitor, weak on SGLT1.</p>
    Formula:C22H24ClFO7
    Color and Shape:Solid
    Molecular weight:454.87
  • TP-030-2

    CAS:
    <p>TP-030-2 is a RIPK1 inhibitor (human K i =0.43 nM ; mouse IC 50 =100 nM) .</p>
    Formula:C23H21BrN4O3
    Color and Shape:Solid
    Molecular weight:481.34
  • ZIKV-IN-5


    <p>ZIKV-IN-5 is an acid-stable, low cytotoxic anti-ZIKV agent with an EC50 value of 0.71 μM. ZIKV-IN-5 showed effective inhibition of ZIKV NS5 MTase activity.</p>
    Formula:C36H45NO4Si
    Color and Shape:Solid
    Molecular weight:583.83
  • Chitinovorin C

    CAS:
    <p>Chitinovorin C is a β-lactam class antibiotic (antibiotic) that exhibits weak inhibitory activity against Gram-negative bacteria.</p>
    Formula:C15H20N4O8S
    Color and Shape:Solid
    Molecular weight:416.406
  • O-Demethylpaulomycin A

    CAS:
    <p>O-Demethylpaulomycin A is an antibiotic known for its antibacterial properties. It is particularly effective against Gram-positive bacteria, including Staphylococcus aureus.</p>
    Formula:C33H44N2O17S
    Color and Shape:Solid
    Molecular weight:772.771
  • NS2B/NS3-IN-5


    <p>Compound 25b inhibits DENV2/ZIKV NS2B/NS3 proteases; IC50: ZIKV 0.67μM, DENV2 4.38μM.</p>
    Formula:C14H9IN2O3S
    Color and Shape:Solid
    Molecular weight:412.2
  • Coleon-U-quinone

    CAS:
    <p>Coleon-U-quinone, a P-gp inhibitor, reduces cancer cell viability and enhances Doxorubicin sensitivity in resistant cells.</p>
    Formula:C20H24O5
    Color and Shape:Solid
    Molecular weight:344.4
  • Canosimibe

    CAS:
    <p>Canosimibe is a cholesterol absorption inhibitor</p>
    Formula:C44H60FN3O10
    Color and Shape:Solid
    Molecular weight:809.96
  • Scytalol A

    CAS:
    <p>Scytalol A selectively inhibits the biosynthesis of dihydroxynaphthalene melanin in Lachnellula sp. A32-89, while not affecting the growth of the strain.</p>
    Formula:C15H18O6
    Color and Shape:Solid
    Molecular weight:294.3
  • PI4KIIIbeta-IN-11

    CAS:
    <p>PI4KIIIbeta-IN-11 is a PI4KIIIβ inhibitor (mean pIC50=9.1) that can be used to study diseases caused by RNA viruses and Plasmodium falciparum.</p>
    Formula:C33H39N7O3
    Color and Shape:Solid
    Molecular weight:581.71
  • DNDI-8219

    CAS:
    <p>DNDI-8219 is an antitubercular agent. It has potent antileishmanial effects.</p>
    Formula:C13H10F3N3O5
    Color and Shape:Solid
    Molecular weight:345.23
  • DMGF

    CAS:
    <p>DMGF, a biflavonoid from Taxus, induces apoptosis, autophagy, and inhibits B16F10 cell motility and MMP-2 expression, hindering melanoma metastasis.</p>
    Formula:C32H22O10
    Color and Shape:Solid
    Molecular weight:566.51
  • CGC 11144

    CAS:
    <p>CGC 11144 is a Polyamine analogue inhibit tumor growth in vitro and in vivo.</p>
    Formula:C40H100Cl10N10
    Color and Shape:Solid
    Molecular weight:1075.82
  • Anticancer agent 16


    <p>Anticancer agent 16 showed good cytotoxic effects on HCT-116 cell line (IC50: 8.55 μM), NCI-H460 cell line (IC50: 5.41 μM) and SKOV3 cell line (IC50: 6.4 μM).</p>
    Formula:C27H33N5O6
    Color and Shape:Solid
    Molecular weight:523.58
  • Napyradiomycin C2

    CAS:
    <p>Napyradiomycin C2 is an antibiotic with activity against Gram-positive bacteria and mycobacteria.</p>
    Formula:C25H27Cl3O5
    Color and Shape:Solid
    Molecular weight:513.838
  • Pradimicin T2

    CAS:
    <p>Pradimicin T2 is an antibiotic with activity against filamentous fungi and yeast-like fungi.</p>
    Formula:C37H37NO19
    Color and Shape:Solid
    Molecular weight:799.685
  • Anticancer agent 26


    <p>Anticancer agent 26 is a promising candidate for cancer therapy and deserves further development.</p>
    Formula:C28H33NO5
    Color and Shape:Solid
    Molecular weight:463.57
  • NRX-2663

    CAS:
    <p>NRX-2663 boosts β-catenin binding to E3 ligase SCFβ-TrCP (Kd: 54.8 nM, EC50: 22.9 nM).</p>
    Formula:C20H13F3N2O5
    Color and Shape:Solid
    Molecular weight:418.32
  • WAY-855

    CAS:
    <p>WAY-855 is an EAAT2-preferring, nonsubstrate inhibitor of high-affinity glutamate uptake.</p>
    Formula:C9H11NO4
    Color and Shape:Solid
    Molecular weight:197.19
  • Ascofuranone

    CAS:
    <p>Ascofuranone is an inhibitor of the ubiquinol oxidase activity of Trypanosoma brucei mitochondrial alternative oxidase (TAO), as well as an inhibitor of HsDHODH</p>
    Formula:C23H29ClO5
    Color and Shape:Solid
    Molecular weight:420.93
  • TLR7/8 agonist 7

    CAS:
    <p>TLR7/8 agonist 7 activates immune cells, useful in ISAC synthesis and immunity research.</p>
    Formula:C26H37N7O2
    Color and Shape:Solid
    Molecular weight:479.62
  • AZ12971554


    <p>AZ12971554: Human thrombin inhibitor, Ki=0.3nM; APTT IC50=0.68µM; ECT IC50=0.16µM.</p>
    Formula:C20H17ClFN7O3
    Color and Shape:Solid
    Molecular weight:457.85
  • PS-519

    CAS:
    <p>PS-519 is a human tissue plasminogen activator and proteasome inhibitor.</p>
    Formula:C12H19NO4
    Color and Shape:Solid
    Molecular weight:241.28
  • AMG-222 tosylate

    CAS:
    <p>AMG-222 tosylate is a DPP-IV inhibitor in clinical development for type II diabetes.</p>
    Formula:C39H47N9O6S
    Color and Shape:Solid
    Molecular weight:769.91
  • Seldomycin factor 1

    CAS:
    <p>Seldomycin factor 1 (XK 88-1) is an aminoglycoside antibiotic known for its broad-spectrum antibacterial activity.</p>
    Formula:C17H34N4O10
    Color and Shape:Solid
    Molecular weight:454.473
  • GW-597901 cinnamate

    CAS:
    <p>GW-597901 cinnamate is a long-acting beta(2)-agonist.</p>
    Formula:C34H46N2O8S
    Color and Shape:Solid
    Molecular weight:642.80
  • Kigamicin A

    CAS:
    <p>Kigamicin A exhibits activity against Gram-positive bacteria, including methicillin-resistant Staphylococcus aureus (MRSA), with a minimum inhibitory concentration (MIC) ranging from 0.025 to 0.78 μg/mL.</p>
    Formula:C34H35NO13
    Color and Shape:Solid
    Molecular weight:665.64
  • Mutalomycin

    CAS:
    <p>Mutalomycin is a polyether antibiotic with activity against Gram-positive bacteria, mycoplasma, and coccidia.</p>
    Formula:C41H70O12
    Color and Shape:Solid
    Molecular weight:754.987