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Inhibitors

Inhibitors

Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.

Subcategories of "Inhibitors"

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Found 66627 products of "Inhibitors"

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  • MtTMPK-IN-5


    <p>MtTMPK-IN-5 inhibits Mtb TMPK with IC50 of 34 μM and fights tuberculosis with MIC of 12.5 μM, aiding TB research.</p>
    Formula:C21H23N5O2
    Color and Shape:Solid
    Molecular weight:377.44
  • Thiomuscimol hydrobromide

    CAS:
    <p>Thiomuscimol hydrobromide is an agonist of GABAA receptor.</p>
    Formula:C4H6N2OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:130.17
  • Calphostin I

    CAS:
    <p>Calphostins, from Cladosporium fungus, inhibit PKC. Notably, calphostin C is a potent biochemical tool.</p>
    Formula:C44H38O15
    Color and Shape:Solid
    Molecular weight:806.76
  • FPI-1465

    CAS:
    <p>FPI-1465: Dual serine-β-lactamase &amp; PBP inhibitor; IC50 PBP2=1.0 μg/mL; Kd CTX-M-15=0.011μM, OXA-48=5.3μM.</p>
    Formula:C11H18N4O7S
    Color and Shape:Solid
    Molecular weight:350.35
  • MRTX849 acid

    CAS:
    <p>MRTX849 acid, used to make PROTAC LC-2, effectively degrades KRAS G12C at 0.25-0.76 μM DC50.</p>
    Formula:C34H37ClFN7O4
    Color and Shape:Solid
    Molecular weight:662.16
  • MCB-3681

    CAS:
    <p>MCB-3681, active against gram-positive bacterium, is the antibacterial Oxaquin's active substance.</p>
    Formula:C31H32F2N4O8
    Color and Shape:Solid
    Molecular weight:626.6
  • Mesulergine

    CAS:
    <p>Mesulergine is metabolized into dopaminergic agonists.</p>
    Formula:C18H26N4O2S
    Color and Shape:Solid
    Molecular weight:362.49
  • KF 20274

    CAS:
    <p>KF 20274 is an adenosine A1 antagonist; purinergic receptor antagonist.</p>
    Formula:C21H29N5O
    Color and Shape:Solid
    Molecular weight:367.49
  • Dinordrin

    CAS:
    <p>Dinordrin is an implantation inhibitor and hormone.</p>
    Formula:C27H36O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:424.57
  • PARP10/15-IN-1


    <p>PARP10/15-IN-1 (compound 8l) is a dual PARP10 and PARP15 inhibitor with IC50s of 160 nM and 370 nM, respectively. It can be used in cancer research[1].</p>
    Formula:C13H10N2O3S
    Color and Shape:Solid
    Molecular weight:274.3
  • MAO-B-IN-10


    <p>MAO-B-IN-10: Potent, selective MAO-B inhibitor; crosses blood-brain barrier; IC50 5.3 μM; reduces Aβ aggregation 58.2%, disaggregates 43.3%.</p>
    Formula:C23H26N2O4
    Color and Shape:Solid
    Molecular weight:394.46
  • Demethoxyviridin

    CAS:
    <p>Demethoxyviridin inhibits mammalian Ptdlns 3-kinase (p110) and is antifungal.</p>
    Formula:C19H14O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:322.31
  • GSK3739936

    CAS:
    <p>GSK3739936 inhibits HIV-1 integrase (IC50: 11.1 nM, EC50: 1.7 nM), weak on CYP (IC50 &gt;24.3 μM), rapid absorption, moderate clearance, high oral availability.</p>
    Formula:C34H43FN2O4
    Color and Shape:Solid
    Molecular weight:562.71
  • LTD4 antagonist 1

    CAS:
    <p>LTD4 antagonist 1 is a potent and orally active antagonist of leukotriene D4 (LTD4; Ki: 0.57 nM).</p>
    Formula:C31H32F3N3O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:615.66
  • Kinamycin B

    CAS:
    <p>Kinamycin B is an antibacterial agent with anticancer activity.</p>
    Formula:C20H16N2O8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:412.35
  • Cap-dependent endonuclease-IN-10

    CAS:
    <p>Cap-dependent endonuclease-IN-10, with low toxicity &amp; good stability, effectively inhibits flu viruses and shows promise against A, B, C types.</p>
    Formula:C25H18F2N4O5S
    Color and Shape:Solid
    Molecular weight:524.50
  • NSC 828467


    <p>NSC 828467 is one of the top five CA-IX inhibitors with significant in vitro anticancer activity (IC50: 27.2 nM).</p>
    Formula:C21H19N9O2S
    Color and Shape:Solid
    Molecular weight:461.5
  • Neuraminidase-IN-7


    <p>Neuraminidase-IN-7, a thiophene, inhibits neuraminidase (IC50 0.03 μM), showing promise for flu research.</p>
    Formula:C21H20N2O6S
    Color and Shape:Solid
    Molecular weight:428.46
  • AS-1940477 hydrobromide

    CAS:
    <p>AS-1940477 hydrobromide is a p38 mitogen-activated protein kinase (MAPK) inhibitor.</p>
    Formula:C24H23BrFN5O2
    Color and Shape:Solid
    Molecular weight:512.38
  • PDE4-IN-5


    <p>PDE4-IN-5: potent PDE4 inhibitor, IC50 = 3.1 nM, superb skin penetration, anti-psoriasis effect.</p>
    Formula:C21H28N2O3
    Color and Shape:Solid
    Molecular weight:356.46
  • Antifungal agent 25


    <p>Antifungal agent 25: broad-spectrum, stable in vivo, effective against Candida albicans, including fluconazole-resistant strains.</p>
    Color and Shape:Solid
  • Py-MPB-amino-C3-PBD

    CAS:
    <p>Py-MPB-amino-C3-PBD is a cytotoxic agent comprised non-alkylating group,with antimicrobial activity.</p>
    Formula:C41H44N8O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:744.84
  • YKL-1-116

    CAS:
    <p>YKL-1-116 is an effective, selective, and covalent CDK7 inhibitor.</p>
    Formula:C34H38N8O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:606.72
  • ER272

    CAS:
    <p>ER272 is a natural PKC activator, inducing hippocampal neurogenesis.</p>
    Formula:C24H34O6
    Color and Shape:Solid
    Molecular weight:418.52
  • Retezorogant

    CAS:
    <p>Retezorogant is a retinoic acid receptor-related orphan receptor gamma (RORγ) antagonist.</p>
    Formula:C23H33ClN2O3
    Color and Shape:Solid
    Molecular weight:420.97
  • KRAS inhibitor-21

    CAS:
    <p>KRAS inhibitor-21 (22b) is a KRAS G12C inhibitor (IC50&lt;0.01 μM) that can be used in cancer research.</p>
    Formula:C33H41N5O3
    Color and Shape:Solid
    Molecular weight:555.71
  • Macbecin I

    CAS:
    <p>Hsp90 inhibitor</p>
    Formula:C30H42N2O8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:558.66
  • SDZ 220-040

    CAS:
    <p>SDZ 220-040 是一种选择性哺乳动物 NMDA 受体拮抗剂,可诱导根系生长的部分无重力模式 。</p>
    Formula:C16H16Cl2NO6P
    Purity:98.13%
    Color and Shape:Solid
    Molecular weight:420.18
  • CP-642931

    CAS:
    <p>CP-642931 (Sorbitol dehydrogenase-IN-1) is a sorbitol dehydrogenase inhibitor used in the study of diabetes mellitus and cardiovascular disease.</p>
    Formula:C17H25N7O
    Purity:99.67% - >99.99%
    Color and Shape:Solid
    Molecular weight:343.43
  • Zelasudil

    CAS:
    <p>Zelasudil (RXC007) is a Rho-related (ROCK) kinase inhibitor for the study of idiopathic pulmonary fibrosis and inflammation.</p>
    Formula:C22H21F2N7O
    Purity:99.15%
    Color and Shape:Solid
    Molecular weight:437.445
  • BMS-986141

    CAS:
    <p>BMS-986141(UDM-003183) is a selective and potent protease-activated receptor-4 (PAR-4) antagonist with oral activity and an IC50 value of 0.4 nM.BMS-98614</p>
    Formula:C27H23N5O5S2
    Purity:98.43% - 99.26%
    Color and Shape:Solid
    Molecular weight:561.63
  • AM103

    CAS:
    <p>AM103 is an effective and selective inhibitor of FLAP (IC50 = 4.2 nM).</p>
    Formula:C36H38N3NaO4S
    Purity:99.75%
    Color and Shape:Solid
    Molecular weight:631.76
  • (+)-Tetrabenazine

    CAS:
    <p>(+)-Tetrabenazine ((3R,11bR)-Tetrabenazine) is a reversible vesicular monoamine transporter 2 (VMAT-2) inhibitor, inhibits transport by VMAT2 with 10-fold</p>
    Formula:C19H27NO3
    Purity:98.31%
    Color and Shape:Solid
    Molecular weight:317.42
  • Emprumapimod

    CAS:
    <p>Emprumapimod, an oral p38α MAPK inhibitor, targets RPMI-8226 cells, curbs LPS-induced IL-6; IC50: 100 pM; for cardiomyopathy, acute pain.</p>
    Formula:C24H29F2N5O3
    Purity:99.21% - >99.99%
    Color and Shape:Solid
    Molecular weight:473.52
  • BAY-3827

    CAS:
    <p>BAY-3827 is an AMPK inhibitor with antiproliferative activity and antitumor activity. BAY-3827 inhibits the phosphorylation of acetyl CoA carboxylase 1.</p>
    Formula:C27H25FN6O
    Purity:99.90%
    Color and Shape:Solid
    Molecular weight:468.53
  • HOIPIN-8 sodium

    CAS:
    <p>HOIPIN-8 sodium is a LUBAC inhibitor for the study of inflammatory and immune diseases.</p>
    Formula:C23H15F2N4NaO3
    Purity:97.34%
    Color and Shape:Solid
    Molecular weight:456.38
  • HRO761

    CAS:
    <p>HRO761 is a potent Werne r syndrome RecQ DNA deconjugase (WRN) inhibitor that can be used to study cancers such as colon and stomach cancer.</p>
    Formula:C31H31ClF3N9O5
    Purity:98.74% - 99.62%
    Color and Shape:Solid
    Molecular weight:702.08
  • O-Propargyl-Puromycin

    CAS:
    <p>O-Propargyl-Puromycin (OP-puro) is a potent protein synthesis inhibitor, a puromycin acetylene analog.</p>
    Formula:C24H29N7O5
    Purity:97.83% - 99.70%
    Color and Shape:Solid
    Molecular weight:495.53
  • Dual FAAH/sEH-IN-1

    CAS:
    <p>Dual FAAH/sEH-IN-1 inhibits both sEH (IC50: 9.6 nM) and FAAH (IC50: 7 nM), offering potent anti-inflammatory effects.</p>
    Formula:C25H22ClN3O3S2
    Purity:99.89%
    Color and Shape:Solid
    Molecular weight:512.04
  • Tuvusertib

    CAS:
    <p>Tuvusertib (M1774), an oral ATR inhibitor (Ki&lt;1µM), selectively blocks CHK1 phosphorylation, disrupts DNA repair, and induces tumor cell apoptosis.</p>
    Formula:C16H12F2N8O
    Purity:98.44% - 99.66%
    Color and Shape:Solid
    Molecular weight:370.32
  • BODIPY FL prazosin

    CAS:
    <p>BODIPY FL prazosin is an α1-adrenergic antagonist that inhibits α1a-AR and α1b-AR.</p>
    Formula:C28H32BF2N7O3
    Purity:97.27%
    Color and Shape:Solid
    Molecular weight:563.41
  • SYM2206

    CAS:
    <p>SYM2206 is a low affinity non-competitive AMPA receptor antagonist with an IC50 value of 1.6 μM.SYM2206 exhibits anticancer activity by blocking Nav1.6-mediated</p>
    Formula:C20H22N4O3
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:366.41
  • NDI-034858

    CAS:
    <p>NDI-034858 (TAK-279) is a tyrosine kinase 2 (TYK2) inhibitor (Kd&lt;200 pM) that targets the JH2 structural domain of Tyk2 for the treatment of autoimmune diseases</p>
    Formula:C23H24N8O3
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:460.49
  • Simmitecan hydrochloride

    CAS:
    <p>Simmitecan hydrochloride is a camptothecin derivative, a topoisomerase I inhibitor with anticancer activity, which can be used to study is solid tumors.</p>
    Formula:C34H39ClN4O6
    Purity:98.20% - 98.93%
    Color and Shape:Solid
    Molecular weight:635.15
  • GLPG0974

    CAS:
    <p>GLPG0974 is an antagonist of FFA2/GPR43 with IC50 of 9 nM.</p>
    Formula:C25H25ClN2O4S
    Purity:99.8%
    Color and Shape:Solid
    Molecular weight:484.99
  • EZM0414

    CAS:
    <p>EZM0414 is a potent, selective, orally bioavailable inhibitor of SETD2 with IC50 of 18 nM in SETD2 biochemical assay and IC50 of 34 nM in a cellular assay.</p>
    Formula:C22H29FN4O2
    Purity:99.58%
    Color and Shape:Solid
    Molecular weight:400.49
  • INCB054329

    CAS:
    <p>INCB054329 is a BET inhibitor targeting BRD2/3/4 and BRDT with IC50s ranging from 1-119 nM.</p>
    Formula:C19H16N4O3
    Purity:99.52%
    Color and Shape:Solid
    Molecular weight:348.36
  • Eravacycline dihydrochloride

    CAS:
    <p>Eravacycline dihydrochloride (TP-434-046) is a potent and broad-spectrum antibacterial agent against six E. coli (MICs: 0.125-0.25 mg/L).</p>
    Formula:C27H33Cl2FN4O8
    Purity:94.59% - 95%
    Color and Shape:Solid
    Molecular weight:631.48
  • KI696

    CAS:
    <p>KI696 is a high-affinity probe that potently inhibits the interaction of Keap1 and NRF2.</p>
    Formula:C28H30N4O6S
    Purity:99.74%
    Color and Shape:Solid
    Molecular weight:550.63
  • Gepotidacin mesylate dihydrate

    CAS:
    <p>Gepotidacin mesylate dihydrate (GSK2140944 mesylate dihydrate) is an antibiotic and an inhibitor of bacterial type II topoisomerase.</p>
    Formula:C25H36N6O8S
    Purity:99.85%
    Color and Shape:Solid
    Molecular weight:580.65
  • Elacytarabine

    CAS:
    <p>Elacytarabine (M7594 0037), a lipid-conjugated derivative of the nucleoside analog cytarabine, is an antineoplastic drug. It has cytotoxicity in solid tumors.</p>
    Formula:C27H45N3O6
    Purity:97.69%
    Color and Shape:Solid
    Molecular weight:507.66
  • MAO-B-IN-17

    CAS:
    <p>MAO-B-IN-17 is a selective and potent monoamine oxidase B (MAO-B) inhibitor (IC50: 5.08 μM) for the study of central nervous system disorders like Parkinson's.</p>
    Formula:C17H17F2NO2
    Purity:99.41%
    Color and Shape:Soild
    Molecular weight:305.32
  • BCL6-IN-3

    CAS:
    <p>BCL6-IN-3: potent BCL6 inhibitor, 70 nM GI50 in SU-DHL4, affects cell functions, antitumor.</p>
    Formula:C24H31ClF2N6O2
    Purity:98.17%
    Color and Shape:Solid
    Molecular weight:508.99
  • STK-15

    CAS:
    <p>STK-15 is a candidate for use as a fatty acid binding protein 5 (FABP5) inhibitor.</p>
    Formula:C34H29NO5
    Purity:98.05%
    Color and Shape:Solid
    Molecular weight:531.6
  • NRX-103095

    CAS:
    <p>NRX-103095 increases β-catenin binding to SCFβ-TrCP E3 ligase; EC50 is 163 nM for pSer33/Ser37 affinity boost.</p>
    Formula:C22H16Cl2F3N3O3S
    Purity:99.58% - 99.95%
    Color and Shape:Solid
    Molecular weight:530.35
  • AKT Kinase Inhibitor

    CAS:
    <p>AKT Kinase Inhibitor is an Akt inhibitor with antitumor activity that selectively inhibits cell proliferation in a dose-dependent manner.Cost-effective and quality-assured.</p>
    Formula:C16H19N7O3
    Purity:97.83% - 99.13%
    Color and Shape:Solid
    Molecular weight:357.37
  • Obicetrapib

    CAS:
    <p>Obicetrapib (AMG-899) is an inhibitor of cholesteryl ester transfer protein.</p>
    Formula:C32H31F9N4O5
    Purity:99.26% - >99.99%
    Color and Shape:Solid
    Molecular weight:722.6
  • SB-423562

    CAS:
    <p>SB-423562 is a calcium-sensing receptor (CaSR) antagonist and can be used in studies about osteoporosis.</p>
    Formula:C26H32N2O4
    Purity:99.22%
    Color and Shape:Solid
    Molecular weight:436.54
  • KU-60019

    CAS:
    <p>KU-60019 is a specific inhibitor of ATM kinase (IC50: 6.3 nM).</p>
    Formula:C30H33N3O5S
    Purity:98.05% - 98.50%
    Color and Shape:Solid
    Molecular weight:547.67
  • BMS 299897

    CAS:
    <p>BMS 299897, a sulfonamide γ-secretase inhibitor, inhibits Aβ production with an IC50 of 7 nM in HEK293 cells overexpressing APP.</p>
    Formula:C24H21ClF3NO4S
    Purity:99.82%
    Color and Shape:Solid
    Molecular weight:511.94
  • Vecabrutinib

    CAS:
    <p>Vecabrutinib (SNS-062) is a potent and noncovalent BTK and ITK inhibitor (Kd: 0.3 nM and 2.2 nM, respectively). Vecabrutinib displays an IC50 of 24 nM for ITK.</p>
    Formula:C22H24ClF4N7O2
    Purity:99.74%
    Color and Shape:Solid
    Molecular weight:529.92
  • LLY-283

    CAS:
    <p>LLY-283, PRMT5 inhibitor, IC50 22 nM, Kd 6 nM, oral, selective, with antitumor effects.</p>
    Formula:C17H18N4O4
    Purity:99.49%
    Color and Shape:Solid
    Molecular weight:342.35
  • NRX-103094

    CAS:
    <p>NRX-103094 boosts β-catenin binding to SCFβ-TrCP ligase with EC50 62 nM and Kd 0.6 nM.</p>
    Formula:C20H11Cl2F3N2O4S
    Purity:99.13%
    Color and Shape:Solid
    Molecular weight:503.28
  • Lometrexol

    CAS:
    <p>Lometrexol (LY 264618) is an antifolate that inhibits GARFT, blocks purine synthesis, induces apoptosis, and has anticancer properties.</p>
    Formula:C21H25N5O6
    Purity:97.76% - 99.56%
    Color and Shape:Solid
    Molecular weight:443.45
  • NRX-1532


    <p>NRX-1532 is a small molecule β-catenin:β-TrCP interaction enhancer.</p>
    Formula:C16H11F3N4O2
    Purity:98.95% - 99.68%
    Color and Shape:Solid
    Molecular weight:348.28
  • Cort108297

    CAS:
    <p>Cort108297: selective GR modulator/antagonist, high GR affinity (Ki: 0.45nM), no other steroid receptor affinity.</p>
    Formula:C26H25F4N3O3S
    Purity:98.36% - 99.94%
    Color and Shape:Solid
    Molecular weight:535.55
  • SY-5609

    CAS:
    <p>SY-5609 (CDK7-IN-3) is a selective non-covalent CDK7 inhibitor, with weak inhibitory activity against CDK2, CDK9 and CDK12.Cost-effective and quality-assured.</p>
    Formula:C23H26F3N6OP
    Purity:99.34% - >99.99%
    Color and Shape:Solid
    Molecular weight:490.46
  • Aldometanib

    CAS:
    <p>Aldometanib (LXY-05-029) is an oral aldolase inhibitor that maintains metabolic balance by blocking FBP and activating lysosomal AMPK.</p>
    Formula:C27H43Cl2IN2
    Purity:99.32% - 99.55%
    Color and Shape:Solid
    Molecular weight:593.46
  • AZ12601011

    CAS:
    <p>AZ12601011 is a TGFBR1 kinase inhibitor that inhibits the growth of breast tumors.</p>
    Formula:C19H15N5
    Purity:98.81%
    Color and Shape:Solid
    Molecular weight:313.36
  • IDX184

    CAS:
    <p>IDX184 is a potent, orally active, targeted HCV polymerase inhibitor and nucleoside polymerase.IDX184 effectively inhibits HCV polymerase (IC50=0.31 μM, Ki=52.3</p>
    Formula:C25H35N6O9PS
    Purity:97.15%
    Color and Shape:Solid
    Molecular weight:626.62
  • Treprostinil diethanolamine

    CAS:
    <p>Treprostinil diethanolamine (UT-15C) is a potent agonist of EP2, DP1 and IP, with values of 3.6, 4.4, 32.1, 212, 826, 2505 and 4680 nM for EP2, DP1, IP, EP1,</p>
    Formula:C27H45NO7
    Purity:99.86%
    Color and Shape:Solid
    Molecular weight:495.65
  • VX-984

    CAS:
    <p>VX-984 (M9831) is an oral DNA-PK inhibitor, crossing the blood-brain barrier, targeting GBM and NSC-LC.</p>
    Formula:C23H21D2N7O
    Purity:97.65% - 99.98%
    Color and Shape:Solid
    Molecular weight:415.49
  • Picrotoxinin

    CAS:
    <p>Picrotoxinin blocks chloride channels, antagonizes GABAA noncompetitively (IC50: 1.15 μM, α1β2γ2L), and induces convulsions.</p>
    Formula:C15H16O6
    Purity:98.07%
    Color and Shape:Solid
    Molecular weight:292.28
  • Pocenbrodib

    CAS:
    <p>Pocenbrodib (FT-7051) is a potent inhibitor of the bromodomain of the CBP/p300 family with potential antitumour activity and is palatable for cancer research.</p>
    Formula:C28H32FN3O6
    Purity:98.48% - 99.54%
    Color and Shape:Solid
    Molecular weight:525.57
  • AChE-IN-26

    CAS:
    <p>AChE-IN-26 (compound 4a) is an AChE (acetylcholinesterase) inhibitor (IC50: 0.42 μM).</p>
    Formula:C21H21BrN2O3
    Purity:99.24% - 99.85%
    Color and Shape:Soild
    Molecular weight:429.31
  • Enbezotinib

    CAS:
    <p>Enbezotinib is an inhibitor of RET autophosphorylation and can be used in cancer research.</p>
    Formula:C21H21FN6O3
    Purity:99.84%
    Color and Shape:Solid
    Molecular weight:424.43
  • Cbl-b-IN-3

    CAS:
    <p>Cbl-b-IN-3 is a potent inhibitor of casitas b lineage lymphoma proto-oncogene-b (Cbl-b) (ic50 &lt; 1 nM).Cost-effective and quality-assured.</p>
    Formula:C30H34F3N5O
    Purity:99%
    Color and Shape:Solid
    Molecular weight:537.62
  • USP15-IN-1

    CAS:
    <p>USP15-IN-1 is a potent USP15 inhibitor (IC50 is 3.76 μM).</p>
    Formula:C22H23N3O3
    Purity:99.509% - 99.81%
    Color and Shape:Solid
    Molecular weight:377.44
  • GSK3368715 dihydrochloride

    CAS:
    <p>GSK3368715 dihydrochloride (EPZ019997 dihydrochloride) is a PRMTs inhibitor , with anticancer activity, for the study of advanced solid tumors.</p>
    Formula:C20H40Cl2N4O2
    Purity:99.66% - 99.66%
    Color and Shape:Solid
    Molecular weight:439.46
  • Vofopitant

    CAS:
    <p>Vofopitant (GR 205171) is a potent NK1 receptor antagonist with anxiolytic and antiemetic activity for the study of post-traumatic stress disorder (PTSD).</p>
    Formula:C21H23F3N6O
    Purity:97.86%
    Color and Shape:Solid
    Molecular weight:432.44
  • Milademetan

    CAS:
    <p>Milademetan (DS-3032), an MDM2 inhibitor, exhibits antitumor activity, induces G1 cell cycle arrest and apoptosis, and can be used to study solid tumors.</p>
    Formula:C30H34Cl2FN5O4
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:618.53
  • D75-4590

    CAS:
    <p>D75-4590, a β-1,6-Glucan synthetase inhibitor, combats fungal infections by targeting cell walls.</p>
    Formula:C21H27N5
    Purity:98.56% - 98.85%
    Color and Shape:Solid
    Molecular weight:349.47
  • Aleglitazar

    CAS:
    <p>Aleglitazar (R1439) (R1439) is a potent dual PPARα/γ agonist, with IC50s of 38 nM and 19 nM for human PPARa and PPARγ, respectively.</p>
    Formula:C24H23NO5S
    Purity:99.03%
    Color and Shape:Solid
    Molecular weight:437.51
  • AChE/BChE-IN-10

    CAS:
    <p>AChE/BChE-IN-10 inhibits AChE/BChE (IC50: 0.176/0.47 μM), crosses the blood-brain barrier, and prevents Aβ-aggregation.</p>
    Formula:C26H30N2O2
    Purity:99.55% - 99.88%
    Color and Shape:Soild
    Molecular weight:402.53
  • LY2979165

    CAS:
    <p>LY2979165 (mGlu2 agonist) is an orthosteric agonist of mGluR2 and can be used in studies about serving as an anti-depressant.</p>
    Formula:C13H22N6O6S
    Purity:98.41%
    Color and Shape:Solid
    Molecular weight:390.42
  • SB-224289 hydrochloride

    CAS:
    <p>SB-224289 hydrochloride (SB-224289A) is a selective antagonist of 5-HT1B receptor, with anxiolytic effect.</p>
    Formula:C32H33ClN4O3
    Purity:97.82% - 98.99%
    Color and Shape:Solid
    Molecular weight:557.08
  • ALOX15-IN-2

    CAS:
    <p>ALOX15-IN-2: Potent ALOX15 inhibitor. IC50: 1.55 μM for LA; 2.79 μM for AA. Stops linoleic/arachidonic acid oxidation.</p>
    Formula:C23H29N3O4S
    Purity:98.10%
    Color and Shape:Solid
    Molecular weight:443.56
  • BDZ-g

    CAS:
    <p>BDZ-g: potent, selective AMPA receptor antagonist; useful for researching neurological disorders.</p>
    Formula:C21H21N5O2S
    Purity:99.97%
    Color and Shape:Solid
    Molecular weight:407.49
  • Odevixibat

    CAS:
    <p>Odevixibat (A4250) is a selective oral inhibitor for ileal bile acid transport, potentially treating primary biliary cirrhosis.</p>
    Formula:C37H48N4O8S2
    Purity:99.53% - 99.83%
    Color and Shape:Solid
    Molecular weight:740.93
  • BMS453

    CAS:
    <p>BMS453 (BMS-189453), a synthetic retinoid, is a potent and selective agonist of RARβ and a potent testicular toxin.</p>
    Formula:C27H24O2
    Purity:99.93%
    Color and Shape:Solid
    Molecular weight:380.48
  • BQ-788

    CAS:
    <p>BQ-788 is an ETB receptor antagonist with potential hypertensive activity that inhibits exogenous ET-1-induced elevation of coronary perfusion pressure.</p>
    Formula:C34H51N5O7
    Purity:98.81%
    Color and Shape:Solid
    Molecular weight:641.8
  • Cap-dependent endonuclease-IN-1

    CAS:
    <p>Cap-dependent endonuclease-IN-1: potent, oral inhibitor with antiviral properties against influenza.</p>
    Formula:C27H22F2N2O6S
    Purity:98.88% - 99.09%
    Color and Shape:Solid
    Molecular weight:540.54
  • BLU2864

    CAS:
    <p>BLU2864: oral PRKACA inhibitor, IC50=0.3 nM, potential in cancer/poly. kidney disease research.</p>
    Formula:C24H19F3N4O2
    Purity:97.58% - 99.92%
    Color and Shape:Soild
    Molecular weight:452.43
  • DRF-1042

    CAS:
    <p>DRF-1042 is a camptothecin analog with anticancer and insecticidal activity and is used to study solid tumors such as prostate and colon cancer.</p>
    Formula:C22H20N2O6
    Purity:98.34%
    Color and Shape:Solid
    Molecular weight:408.4
  • Umibecestat

    CAS:
    <p>Umibecestat inhibits human and mouse BACE-1 (IC50: 11 nM &amp; 10 nM), potentially for Alzheimer's research.</p>
    Formula:C19H15ClF7N5O2
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:513.8
  • Darizmetinib

    CAS:
    <p>Darizmetinib (HRX215) is an MKK4 inhibitor.</p>
    Formula:C21H17F2N5O3S
    Purity:98.03% - 99.57%
    Color and Shape:Solid
    Molecular weight:457.45
  • WAY-213613 hydrochloride

    CAS:
    <p>WAY-213613 hydrochloride: potent, selective GLT-1/EAAT2 inhibitor (IC50 85 nM); weaker for EAAT1/3; inactive at glutamate receptors; research tool for CNS.</p>
    Formula:C16H13BrF2N2O4
    Purity:99.14% - 99.37%
    Color and Shape:Soild
    Molecular weight:415.19
  • NB-360

    CAS:
    <p>NB-360: potent, brain-penetrant BACE1/2 inhibitor; IC50s: 5-6 nM; high selectivity vs pepsin, cathepsin E/D.</p>
    Formula:C21H19F4N5O2
    Purity:99.72%
    Color and Shape:Solid
    Molecular weight:449.4
  • Dazostinag disodium

    CAS:
    <p>Dazostinag disodium (TAK-676) is a synthetic novel interferon gene (STING) agonist.Cost-effective and quality-assured.</p>
    Formula:C21H20F2N8Na2O10P2S2
    Purity:98.84% - 99.96%
    Color and Shape:Solid
    Molecular weight:754.48
  • Vofopitant dihydrochloride

    CAS:
    <p>Vofopitant dihydrochloride (GR 205171A) is a tachykinin NK1 receptor antagonist and a potential compound for the treatment of pathologic vomiting.</p>
    Formula:C21H25Cl2F3N6O
    Purity:98.99%
    Color and Shape:Solid
    Molecular weight:505.36
  • DN02


    <p>DN02: a potent, selective BRD8(1) bromodomain probe; Ki=32 nM; 30x more affine than BRD8(2).</p>
    Formula:C22H24FN3O3
    Purity:98.22% - 99.74%
    Color and Shape:Solid
    Molecular weight:397.44
  • Rupintrivir

    CAS:
    <p>Rupintrivirvr (AG7088) is a mimetic peptide inhibitor of rhinovirus (HRV) 3C cysteine protease with antiviral activity for the study of viral infections.</p>
    Formula:C31H39FN4O7
    Purity:97.72% - 99.35%
    Color and Shape:Solid
    Molecular weight:598.66
  • AZD5462

    CAS:
    <p>AZD5462 is a potent orally available relaxin receptor RXFP1 agonist for the study of heart failure and cancer.</p>
    Formula:C30H41FN2O6
    Purity:98.32% - 99.63%
    Color and Shape:Solid
    Molecular weight:544.65
  • Suzetrigine

    CAS:
    <p>Suzetrigine (VX-548) is an oral NaV1.8 inhibitor with analgesic properties for acute pain research.</p>
    Formula:C21H20F5N3O4
    Purity:98.08% - 99.27%
    Color and Shape:Solid
    Molecular weight:473.39
  • MIV-247

    CAS:
    <p>MIV-247 is a cathepsin S inhibitor that attenuates mechanically abnormal pain in preclinical neuropathic pain models and can be used to study myocardial injury.</p>
    Formula:C17H24F3N3O4
    Purity:99.27%
    Color and Shape:Solid
    Molecular weight:391.39
  • LSN3318839

    CAS:
    <p>LSN3318839 is a potent and orally available glucagon-like peptide-1 receptor (GLP-1R) modulator.LSN3318839 enhances GLP-1R G-protein-coupled signaling and can</p>
    Formula:C26H23Cl2N3O2
    Purity:99.21%
    Color and Shape:Solid
    Molecular weight:480.39
  • PREP inhibitor-1

    CAS:
    <p>PREP inhibitor-1 is a prolyl oligopeptidase (PREP) inhibitor for the study of Alzheimer's disease.</p>
    Formula:C22H28N4O2
    Purity:98.78%
    Color and Shape:Soild
    Molecular weight:380.48
  • AZD 3147

    CAS:
    <p>AZD 3147 inhibits mTORC1 (40.7 nM), mTORC2 (5.75 nM), and PI3Kα/β/δ/γ (912/5495/9333/6310 nM IC50s).</p>
    Formula:C24H31N5O4S2
    Purity:99.99%
    Color and Shape:Solid
    Molecular weight:517.66
  • SJ6986

    CAS:
    <p>SJ6986 is a potent, selective and orally active GSPT1/2 degrader. SJ6986 degrades GSPT1 with a DC 50 of 2.1 nM (D max 99%) [1].</p>
    Formula:C20H14F3N3O7S
    Purity:99.73%
    Color and Shape:Solid
    Molecular weight:497.4
  • Dersimelagon

    CAS:
    <p>Dersimelagon (MT-7117) is an orally active, selective melanocortin 1 receptor (MC1R) agonist.Cost-effective and quality-assured.</p>
    Formula:C36H45F4N3O5
    Purity:97.35% - 98.23%
    Color and Shape:Solid
    Molecular weight:675.75
  • NRX-252114

    CAS:
    <p>NRX-252114 promotes mutant β-catenin degradation, binding it to E3 ligase SCFβ-TrCP (EC50: 6.5 nM; Kd: 0.4 nM).</p>
    Formula:C22H12Cl2F3N3O2S
    Purity:99.70%
    Color and Shape:Solid
    Molecular weight:510.32
  • USP5-IN-1


    <p>USP5-IN-1, a powerful USP5 deubiquitinase inhibitor, selectively binds with 2.8 μM affinity, blocking USP5's di-ubiquitin cleavage.</p>
    Formula:C19H20ClN3O5S
    Purity:99.76%
    Color and Shape:Soild
    Molecular weight:437.9
  • ZD 7155 hydrochloride

    CAS:
    <p>ZD 7155 hydrochloride is an angiotensin II receptor type 1 (AT1 receptor) antagonist.</p>
    Formula:C26H27ClN6O
    Purity:99.8%
    Color and Shape:Solid
    Molecular weight:474.98
  • Moiramide B

    CAS:
    <p>Moiramide B is an acetyl coenzyme A carboxylase inhibitor with antimicrobial activity, strongly inhibiting Gram-positive bacteria.</p>
    Formula:C25H31N3O5
    Purity:98.53% - 99.90%
    Color and Shape:Solid
    Molecular weight:453.53
  • L-371,257

    CAS:
    <p>L-371,257 is a competitive antagonist of oxytocin receptor with pA2 of 8.4 and Ki of 19 nM. L-371,257 shows a Ki of 3.7 nM for vasopressin receptor 1a.</p>
    Formula:C28H33N3O6
    Purity:99.79%
    Color and Shape:Solid
    Molecular weight:507.58
  • FABPs ligand 6

    CAS:
    <p>FABPs ligand 6 (MF6) is an inhibitor of FABP5 and FABP7.</p>
    Formula:C28H27FN2O3
    Purity:97.45%
    Color and Shape:Solid
    Molecular weight:458.52
  • AZD-5672

    CAS:
    <p>AZD-5672 is an antagonist of CCR5 with an IC50 of 0.32 nM.</p>
    Formula:C32H38F2N2O5S2
    Purity:98.1%
    Color and Shape:Solid
    Molecular weight:632.78
  • Glycosyltransferase-IN-1


    <p>Glycosyltransferase-IN-1 is a glycosyltransferase inhibitor with bacteriostatic activity, inhibiting MSSA, MRSA, Bacillus subtilis, and Enterobacteriaceae.</p>
    Formula:C19H21N5O
    Purity:99.76%
    Color and Shape:Solid
    Molecular weight:335.4
  • DRB18

    CAS:
    <p>DRB18 inhibits GLUT proteins, altering glucose metabolism and inducing cancer cell death by G1/S arrest and oxidative stress.</p>
    Formula:C22H23ClN2O2
    Purity:99.54%
    Color and Shape:Solid
    Molecular weight:382.88
  • JNJ-6204

    CAS:
    <p>JNJ-6204 is a deuterated compound that efficiently inhibits CSNK1D and CSNK1E.</p>
    Formula:C19H11D6FN6O
    Purity:97.42% - 99.87%
    Color and Shape:Solid
    Molecular weight:370.41
  • BE1218

    CAS:
    <p>BE1218 is a liver X receptor (LXR) inverse agonist active on LXRα and LXRβ with an IC50 of 9 nM and 7 nM, respectively.</p>
    Formula:C30H30FNO4S2
    Purity:99.7%
    Color and Shape:Soild
    Molecular weight:551.69
  • Iclepertin

    CAS:
    <p>Iclepertin (BI-425809) is a GlyT1 inhibitor.Iclepertin is used for the treatment of Alzheimer;s disease and other CNS disorders.</p>
    Formula:C20H18F6N2O5S
    Purity:98.89% - 98.93%
    Color and Shape:Solid
    Molecular weight:512.42
  • Etamicastat hydrochloride

    CAS:
    <p>Etamicastat hydrochloride (BIA 5-453 hydrochloride) is a peripherally selective dopamine beta-hydroxylase inhibitor that reduces hypertension.</p>
    Formula:C14H16ClF2N3OS
    Purity:98.54%
    Color and Shape:Solid
    Molecular weight:347.81
  • ELOVL1-IN-2

    CAS:
    <p>ELOVL1-IN-2 weakly inhibits ELOVL1 enzyme (IC50: 21 μM) and shows moderate potency in HEK293 cells (IC50: 6.7 μM).</p>
    Formula:C18H15FN2O
    Purity:99.84%
    Color and Shape:Solid
    Molecular weight:294.32
  • JTK-109

    CAS:
    <p>JTK-109 is an inhibitor of hepatitis C virus NS5B RNA-dependent RNA polymerase inhibitor and inhibits G1b and G3a subgenomic replicons and recombinant enzymes.</p>
    Formula:C37H33ClFN3O4
    Purity:98.48% - 99.68%
    Color and Shape:Solid
    Molecular weight:638.13
  • Tigemonam

    CAS:
    <p>Tigemonam is a monobactam, a novel orally administered monobactam that protects against gram-negative aerobic bacterial pathogens. Cost-effective and quality-assured.</p>
    Formula:C12H15N5O9S2
    Purity:99.03% - >99.99%
    Color and Shape:Solid
    Molecular weight:437.41
  • Zotizalkib

    CAS:
    <p>TPX-0131: potent, selective, CNS-ready, oral ALK inhibitor (WT IC50: 1.4nM, G1202R/L1196M IC50: 0.3nM) with robust antitumor effects.</p>
    Formula:C21H20F3N5O3
    Purity:98.7%
    Color and Shape:Solid
    Molecular weight:447.41
  • PF-07258669

    CAS:
    <p>PF-07258669 is a selective melanocortin 4 receptor (MC4) antagonist used in the study of cachexia and loss of appetite.</p>
    Formula:C25H27FN6O2
    Purity:99.9%
    Color and Shape:Solid
    Molecular weight:462.52
  • Evixapodlin

    CAS:
    <p>Evixapodlin (PD-1/PD-L1-IN 7) is a human PD-1/PD-L1 protein/protein interaction inhibitor (IC50: 0.213).Evixapodlin has anticancer and antiviral activities.</p>
    Formula:C34H36Cl2N8O4
    Purity:99.07%
    Color and Shape:Solid
    Molecular weight:691.61
  • CCF0058981

    CAS:
    <p>CCF0058981: noncovalent inhibitor for SARS-CoV-2 &amp; -1 proteases; IC50s: 68 nM (SC2) &amp; 19 nM (SC1). Potential COVID-19 research use.</p>
    Formula:C24H19ClN6O
    Purity:98.94%
    Color and Shape:Soild
    Molecular weight:442.9
  • SR 11302

    CAS:
    <p>SR 11302 is an inhibitor of activator protein-1 (AP-1).</p>
    Formula:C26H32O2
    Purity:98.65%
    Color and Shape:Solid
    Molecular weight:376.53
  • XMD-17-51 Trifluoroacetate

    CAS:
    <p>XMD-17-51 Trifluoroacetate is a pyrimido-diazepinone compound that regulates protein kinases.</p>
    Formula:C23H25F3N8O3
    Purity:99.65%
    Color and Shape:Solid
    Molecular weight:518.49
  • JAK2-IN-7

    CAS:
    <p>JAK2-IN-7 selectively inhibits JAK2 (IC50: 3 nM), shows 14-fold selectivity over JAK1/3, FLT3, induces G0/G1 arrest, apoptosis, and has antitumor effects.</p>
    Formula:C26H33N7O
    Purity:99.54%
    Color and Shape:Solid
    Molecular weight:459.59
  • Gemcitabine elaidate hydrochloride

    CAS:
    <p>CP-4126, a lipophilic pro-drug of Gemcitabine, converts to active form by esterases, allowing oral administration with dose-dependent effects.</p>
    Formula:C27H44ClF2N3O5
    Purity:98.50% - 99.6%
    Color and Shape:Solid
    Molecular weight:564.11
  • PD 151746

    CAS:
    <p>PD151746: calpain inhibitor, Ki μ-calpain=0.26μM, Ki m-calpain=5.33μM; reduces oxLDL cytotoxicity.</p>
    Formula:C11H8FNO2S
    Purity:98.63% - ≥95%
    Color and Shape:Solid
    Molecular weight:237.25
  • Rineterkib

    CAS:
    <p>Rineterkib (ERK-IN-1) is an inhibitor of RAF and ERK1/2 activating mutations in the MAPK pathway.</p>
    Formula:C26H27BrF3N5O2
    Purity:99.73%
    Color and Shape:Solid
    Molecular weight:578.42
  • Sinefungin

    CAS:
    <p>Sinefungin (Adenosyl-Ornithine) is an effective inhibitor of virion mRNA(guanine-7-)-methyltransferase, mRNA(nucleoside-2'-)-methyltransferase, and viral</p>
    Formula:C15H23N7O5
    Purity:98.12%
    Color and Shape:Solid
    Molecular weight:381.39
  • ARN19702

    CAS:
    <p>ARN19702: orally active, brain-penetrant, selective NAAA inhibitor, IC50 230 nM, broad analgesic profile.</p>
    Formula:C21H22FN3O3S2
    Purity:99.86%
    Color and Shape:Solid
    Molecular weight:447.55
  • BRD0639

    CAS:
    <p>BRD0639 is a first-in-class PRMT5-substrate interaction inhibitor for PBM-dependent PRMT5 activity studies.</p>
    Formula:C21H22ClN5O4S
    Purity:99.85%
    Color and Shape:Solid
    Molecular weight:475.95
  • 10-Methoxycamptothecin

    CAS:
    <p>10-Methoxycamptothecin is a natural bioactive derivative of camptothecin (CPT) isolated from Camptotheca acuminata and possesses high anti-cancer properties.</p>
    Formula:C21H18N2O5
    Purity:98.36%
    Color and Shape:Solid
    Molecular weight:378.38
  • CK2 inhibitor 2

    CAS:
    <p>CK2 Inhibitor 2, characterized as a potent, selective, and orally active inhibitor of CK2, demonstrates an impressive IC50 value of 0.66 nM.</p>
    Formula:C21H17ClN4O2
    Purity:99.02%
    Color and Shape:Solid
    Molecular weight:392.84
  • TGFβRI-IN-3

    CAS:
    <p>TGFβRI-IN-3 inhibits TGFβR1 with an IC 50 of 0.79 nM with 2000-fold selectivity against MAP4K4.</p>
    Formula:C28H23N3O2S
    Purity:99.85%
    Color and Shape:Soild
    Molecular weight:465.57
  • LY3143921 hydrate

    CAS:
    <p>LY3143921 ((S)-Example 2) hydrate is an orally active CDC7 kinase inhibitor with broad in vitro anticancer activity [1].</p>
    Formula:C16H14FN5O2
    Purity:98.43%
    Color and Shape:Solid
    Molecular weight:327.31
  • FGI-106 tetrahydrochloride

    CAS:
    <p>FGI-106 tetrahydrochloride demonstrates potent inhibitory activity across a broad spectrum of viruses, including those causing hemorrhagic fevers such as Ebola</p>
    Formula:C28H42Cl4N6
    Purity:99.68%
    Color and Shape:Solid
    Molecular weight:604.48
  • BAY-8400


    <p>BAY-8400 is an orally active, potent and selective DNA-dependent protein kinase ( DNA-PK ) inhibitor ( IC 50 =81 nM) which shows synergistic efficacy in</p>
    Formula:C21H17F2N5O
    Purity:99.53%
    Color and Shape:Solid
    Molecular weight:393.39
  • (E/Z)-GSK5182

    CAS:
    <p>GSK5182 is a racemic mix of (E/Z) isomers, a selective ERRγ inverse agonist (IC50: 79 nM), and induces ROS in liver cancer.</p>
    Formula:C27H31NO3
    Purity:97.58%
    Color and Shape:Solid
    Molecular weight:417.54
  • Rolapitant hydrochloride

    CAS:
    <p>Rolapitant HCl is a potent NK1 antagonist, non-CYP3A4 interactive, with anti-emetic effects and a Ki of 0.66 nM.</p>
    Formula:C25H27ClF6N2O2
    Purity:98.35% - 99.79%
    Color and Shape:Solid
    Molecular weight:536.94
  • Durlobactam sodium salt

    CAS:
    <p>Durlobactam sodium salt (ETX2514) have an IC50 values of 4, 14 and 190 nM against class A KPC-2, class C AmpC and class D OXA-24.Cost-effective and quality-assured.</p>
    Formula:C8H10N3NaO6S
    Purity:97.01% - 99.03%
    Color and Shape:Solid
    Molecular weight:299.23
  • FX-11

    CAS:
    <p>FX-11: potent LDHA inhibitor (Ki 8 μM), activates PKM2, reduces ATP, induces oxidative stress/ROS, cell death, shows antitumor effects.</p>
    Formula:C22H22O4
    Purity:98.95%
    Color and Shape:Solid
    Molecular weight:350.41
  • INCB086550

    CAS:
    <p>INCB086550 (PD-1/PD-L1-IN-8) (example 24) is a PD-1/PD-L1 inhibitor, with an IC50 &lt;= 10 nM.</p>
    Formula:C41H39N7O4
    Purity:98.49%
    Color and Shape:Solid
    Molecular weight:693.79
  • LSZ-102

    CAS:
    <p>LSZ-102 is an effective and selective degrader of estrogen receptor (IC50 = 0.2 nM) and can be used in studies about ERα positive breast cancer.</p>
    Formula:C25H17F3O4S
    Purity:98.56%
    Color and Shape:Solid
    Molecular weight:470.46
  • Sebetralstat

    CAS:
    <p>Sebetralstat (KVD900) is an inhibitor of plasma kallikrein and can be used in studies about metabolic diseases.</p>
    Formula:C26H26FN5O4
    Purity:99.85%
    Color and Shape:Solid
    Molecular weight:491.51
  • Clorophene

    CAS:
    <p>Clorophene (Clorofene) is an antimicrobial agent and can be used in personal care products.</p>
    Formula:C13H11ClO
    Purity:99.87%
    Color and Shape:White To Light Tan Or Pink Flakes Phenolic Odor (Ntp 1992)
    Molecular weight:218.68
  • TEM1/CD248 Protein, Mouse, Recombinant (His)


    <p>TEM1/CD248 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with C-His tag. The predicted molecular weight is 73.6 kDa and the accession number is Q91V98.</p>
    Color and Shape:Solid
    Molecular weight:73.6 kDa (predicted). Due to glycosylation, the protein migrates to 75-140 kDa based on Tris-Bis PAGE result.

    Ref: TM-TMPK

    1mg
    Discontinued
    100µg
    Discontinued
    500µg
    Discontinued
    Discontinued product
  • GAS6 Protein, Human, Recombinant (His)


    <p>GAS6 (Growth arrest-specific protein 6) is also known as AXL receptor tyrosine kinase ligand, AXLLG, is a multimodular protein that is up-regulated by a wide variety of cell types in response to growth arrest. Gas6 binds and induces signaling through the receptor tyrosine kinases Axl, Dtk, and Mer whose signaling is implicated in cell growth and survival, cell adhesion and cell migration. GAS6/AXL signaling plays a role in various processes such as endothelial cell survival during acidification by preventing apoptosis, optimal cytokine signaling during human natural killer cell development, hepatic regeneration, gonadotropin-releasing hormone neuron survival and migration, platelet activation, or regulation of thrombotic responses. GAS6 Protein, Human, Recombinant (His) is expressed in HEK293 cells.</p>
    Purity:>99.90%
    Color and Shape:Soild
    Molecular weight:72.7 KDa (Predicted), 80-90 KDa (Reducing conditions)

    Ref: TM-TMPY

    50µg
    Discontinued
    Discontinued product
  • TCblR Protein, Human, Recombinant (His)


    <p>TCblR Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with C-6xHis tag. The predicted molecular weight is 32-58 KDa and the accession number is Q9NPF0.</p>
    Color and Shape:Solid
    Molecular weight:32-58 KDa (reducing condition)

    Ref: TM-TMPJ

    1mg
    Discontinued
    10µg
    Discontinued
    50µg
    Discontinued
    500µg
    Discontinued
    Discontinued product
  • Relacorilant

    CAS:
    <p>Relacorilant is an oral glucocorticoid receptor antagonist with Ki of 7.2 nM, potential for treating Cushing's syndrome.</p>
    Formula:C27H22F4N6O3S
    Purity:98.53% - 99%
    Color and Shape:Solid
    Molecular weight:586.56

    Ref: TM-T16727

    1mg
    Discontinued
    5mg
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    10mg
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    25mg
    Discontinued
    50mg
    Discontinued
    100mg
    Discontinued
    500mg
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    1ml*10 (DMSO)
    Discontinued
    1mL*10mM (DMSO)_old
    Discontinued
    Discontinued product
  • 3-Acetylcoumarin

    CAS:
    <p>3-Acetylcoumarin as a practical ligand for copper-catalyzed CN coupling reactions at room temperature. It has neuroprotective and acaricidal properties.</p>
    Formula:C11H8O3
    Purity:99.41%
    Color and Shape:Yellow Crystalline Powder
    Molecular weight:188.18

    Ref: TM-FR12596

    5mg
    Discontinued
    1ml*10 (DMSO)
    Discontinued
    Discontinued product
  • 2'-Hydroxy-4'-methylacetophenone

    CAS:
    <p>2'-Hydroxy-4'-methylacetophenone, a phenolic compound isolated from Angelicae koreana roots possesses acaricidal property. 2'-Hydroxy-4'-methylacetophenone has acaricidal activity, it could be used in the preparation of 4'-methyl-2'-[(p-tolylsulfonyl) oxy] acetophenone.</p>
    Formula:C9H10O2
    Purity:99.88%
    Color and Shape:Black Liquid
    Molecular weight:150.17

    Ref: TM-FR14298

    1g
    Discontinued
    1ml*10 (DMSO)
    Discontinued
    Discontinued product
  • α-Terpineol

    CAS:
    <p>Terpineol possesses antifungal activity against Trichophyton mentagrophytes, it also exhibits strong antimicrobial activity against periodontopathic and cariogenic bacteria. α-Terpineol (Terpineol) shows anticonvulsant, and anti-inflammatory activities, it inhibits the gene expression of the IL-6 receptor.</p>
    Formula:C10H18O
    Purity:97.55%
    Color and Shape:Colorless Liquid
    Molecular weight:154.25

    Ref: TM-FR14115

    5g
    Discontinued
    10g
    Discontinued
    1ml*10 (DMSO)
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    Discontinued product
  • PRGL493

    CAS:
    <p>PRGL493 blocks ACSL4, halts PC3/MDA-MB-231 cancer cell spread, and inhibits MA-10 tumor progesterone. Effective in mouse PC3 tumor model at 0.25 mg/kg.</p>
    Formula:C25H21N7O2
    Purity:98.80% - 99.11%
    Color and Shape:Solid
    Molecular weight:451.48

    Ref: TM-T35666

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  • Anisylacetone

    CAS:
    <p>Anisylacetone (Anisylacetone) is an effective lure for the male melon fly.</p>
    Formula:C11H14O2
    Purity:99.74%
    Color and Shape:Liquid
    Molecular weight:178.23

    Ref: TM-FR12339

    5g
    Discontinued
    50g
    Discontinued
    1ml*10 (DMSO)
    Discontinued
    Discontinued product
  • (-)-Isopulegol

    CAS:
    <p>Isopulegol has antioxidant, and neuroactive properties. It also has gastroprotective effects induced by isopulegol appear to be mediated, at least in part, by endogenous prostaglandins, K+ATP channel opening and antioxidant proprieties related to GSH increased.</p>
    Formula:C10H18O
    Purity:99.89%
    Color and Shape:Liquid
    Molecular weight:154.25

    Ref: TM-FR14207

    100mg
    Discontinued
    1ml*10 (DMSO)
    Discontinued
    Discontinued product
  • 3-Methoxyphenylacetic acid

    CAS:
    <p>3-Methoxyphenylacetic acid belongs to the class of organic compounds known as anisoles. 3-Methoxyphenylacetic acid is slightly soluble (in water) and a weakly acidic compound (based on its pKa).3-Methoxyphenylacetic acid (m-Methoxyphenylacetic acid), a m-hydroxyphenylacetic acid (m-OHPAA) derivative, is a phytotoxin in Rhizoctonia solani. 3-Methoxyphenylacetic acid is used to develop a toxin-mediated bioassay for resistance to rhizoctonia root rot</p>
    Formula:C9H10O3
    Purity:98.61%
    Color and Shape:White Solid
    Molecular weight:166.17

    Ref: TM-FR13883

    500mg
    Discontinued
    1ml*10 (DMSO)
    Discontinued
    Discontinued product
  • 4-Ethoxycoumarin

    CAS:
    <p>4-Ethoxycoumarin has antimicrobial activity.</p>
    Formula:C11H10O3
    Purity:99.64%
    Color and Shape:Solid
    Molecular weight:190.2

    Ref: TM-FR12662

    50mg
    Discontinued
    100mg
    Discontinued
    1ml*10 (DMSO)
    Discontinued
    Discontinued product
  • EGFR-IN-7

    CAS:
    <p>EGFR-IN-7 (TQB3804) is a selective and potent EGFR kinase inhibitor.</p>
    Formula:C32H41BrN9O2P
    Purity:95.32% - 99.64%
    Color and Shape:Solid
    Molecular weight:694.6

    Ref: TM-T11161

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  • ANNINE-6plus

    CAS:
    <p>ANNINE-6plus, a water-soluble dye from Germany's Max Planck Institute, tracks cell voltage changes with 30% (1-photon) &amp; &gt;50% (2-photon) intensity shifts.</p>
    Formula:C39H47Br2N3
    Color and Shape:Solid
    Molecular weight:717.62

    Ref: TM-T30078

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    Discontinued
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    Discontinued product
  • 1-(2,3-Dichlorphenyl)-piperazine

    CAS:
    <p>1-(2,3-Dichlorphenyl)-piperazine (DCPP) is a potent DHCR7 inhibitor. DHCR7 is the last enzyme in cholesterol biosynthesis.</p>
    Formula:C10H12Cl2N2
    Purity:98%
    Color and Shape:Brown Oil
    Molecular weight:231.12

    Ref: TM-T20999

    5mg
    Discontinued
    Discontinued product
  • PEG2-bis(phosphonic acid)

    CAS:
    <p>PEG2-bis(phosphonic acid) is a PEG Linker.</p>
    Formula:C6H16O8P2
    Color and Shape:Solid
    Molecular weight:278.13

    Ref: TM-T33906

    100mg
    Discontinued
    500mg
    Discontinued
    Discontinued product
  • Kbz probe 1

    CAS:
    <p>Kbz probe 1, an adaptable probe utilized for examining histone benzoylation and interactions within living cells, showcases extensive versatility.</p>
    Formula:C13H17ClF2N2O3
    Color and Shape:Solid
    Molecular weight:322.73

    Ref: TM-T40235

    25mg
    Discontinued
    Discontinued product
  • Azido-PEG12-t-butyl ester

    CAS:
    <p>Azido-PEG12-t-butyl ester, a soluble PEG with azide/reactive t-butyl, forms triazoles via Click Chemistry; deprotectable in acid.</p>
    Formula:C31H62N3O14
    Color and Shape:Solid
    Molecular weight:700.84

    Ref: TM-T30272

    100mg
    Discontinued
    500mg
    Discontinued
    Discontinued product
  • m-Ciaamp

    CAS:
    <p>3-Carboxyphenyl((N-((4-iodophenyl)acetyl)amino)methyl)phosphonate is a bioactive chemical.</p>
    Formula:C16H15INO6P
    Color and Shape:Solid
    Molecular weight:475.175

    Ref: TM-T29390

    25mg
    Discontinued
    Discontinued product
  • Questiomycin A derivatives 12


    <p>Questiomycin A derivatives 12 is a Questiomycin A derivative.</p>
    Formula:C16H14N2O3
    Purity:99.79%
    Color and Shape:Soild
    Molecular weight:282.29

    Ref: TM-T67711

    1mg
    Discontinued
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  • Anticancer agent 11

    CAS:
    <p>Anticancer agent 11 suppresses angiogenesis and induces DNA cross-links for broad-spectrum efficacy.</p>
    Formula:C20H21N3O2
    Color and Shape:Solid
    Molecular weight:335.40

    Ref: TM-T39868

    25mg
    Discontinued
    Discontinued product
  • Questiomycin A derivatives 13


    <p>Questiomycin A derivatives 13 is a Questiomycin A derivative.</p>
    Formula:C17H14N2O3
    Purity:98.30%
    Color and Shape:Soild
    Molecular weight:294.30

    Ref: TM-T67712

    1mg
    Discontinued
    5mg
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    Discontinued product
  • Trk-IN-6

    CAS:
    <p>Trk-IN-6 shows excellent in vitro potency on a panel of TRK mutants ( IC 50 = 0.2-0.7 nM).</p>
    Formula:C21H21F3N6O2
    Color and Shape:Solid
    Molecular weight:446.43

    Ref: TM-T40150

    25mg
    Discontinued
    Discontinued product
  • PROTAC MDM2 Degrader-2

    CAS:
    <p>PROTAC MDM2 Degrader-2: A potent MDM2-targeting compound with PROTAC tech for E3 ligase-mediated degradation.</p>
    Formula:C70H76Cl4N10O12
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1391.22

    Ref: TM-T18632

    100mg
    Discontinued
    500mg
    Discontinued
    Discontinued product
  • AS-604850


    <p>AS-604850: PI3Kγ inhibitor, ATP-competitive, IC50=2.5μM, 30x&gt; PI3Kδ/β, 18x&gt; PI3Kα.</p>
    Formula:C11H5F2NO4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:285.22

    Ref: TM-T22587

    5mg
    Discontinued
    10mg
    Discontinued
    25mg
    Discontinued
    Discontinued product
  • Phosalacine

    CAS:
    <p>Phosalacine, isolated from Kitasatosporia phosalacinea, is a new herbicidal antibiotic that contains phosphinothricin.</p>
    Formula:C14H28N3O6P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:365.367

    Ref: TM-T25950

    25mg
    Discontinued
    Discontinued product
  • Apratoxin A

    CAS:
    <p>Apratoxin A is a potent cytotoxin isolated from the marine cyanobacterium Lyngbya majuscula Harvey ex Gomont.</p>
    Formula:C45H69N5O8S
    Color and Shape:Solid
    Molecular weight:840.13

    Ref: TM-T30104

    5mg
    Discontinued
    Discontinued product
  • PROTAC BRD4 Degrader-6

    CAS:
    <p>Compound 32a: PROTAC BRD4 Degrader-6, IC50 = 2.7 nM, degrades BRD4, halts BxPC3 pancreatic cancer cell growth, induces apoptosis for research.</p>
    Formula:C43H40F2N10O10S
    Color and Shape:Solid
    Molecular weight:926.9

    Ref: TM-T73958

    5mg
    Discontinued
    50mg
    Discontinued
    Discontinued product
  • C12 NBD Sphingomyelin

    CAS:
    <p>C12 NBD sphingomyelin, a fluorescent sphingomyelin derivative, serves as a sphingomyelinase substrate (Ex=470 nm, Em=525 nm).</p>
    Formula:C41H73N6O9P
    Color and Shape:Solid
    Molecular weight:825.03

    Ref: TM-T75371

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    Discontinued
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    100mg
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    Discontinued product
  • TPPS

    CAS:
    <p>Tetraphenylporphine sulfonate (TPPS) serves as a non-cytotoxic probe suitable for tumor localization detection [1].</p>
    Formula:C44H30N4O12S4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:934.99

    Ref: TM-T78448

    5mg
    Discontinued
    Discontinued product
  • Arsenazo I

    CAS:
    <p>Arsenazo I is a calcium-sensitive, metallochromic dye used as reagent.</p>
    Formula:C16H13AsN2O11S2
    Color and Shape:Solid
    Molecular weight:548.32

    Ref: TM-T30144

    100mg
    Discontinued
    500mg
    Discontinued
    Discontinued product
  • Yimitasvir diphosphate

    CAS:
    <p>Yimitasvir (Emitasvir) diphosphate,一种针对丙型肝炎病毒(HCV)非结构蛋白5A (NS5A)的口服活性抑制剂,适用于慢性丙型肝炎病毒感染的研究。</p>
    Formula:C49H64N8O14P2
    Color and Shape:Solid
    Molecular weight:1051.03

    Ref: TM-T74588

    5mg
    Discontinued
    50mg
    Discontinued
    Discontinued product
  • Pyrromethene 597

    CAS:
    <p>Pyrromethene 597, a BODIPY laser dye, exhibits a wide tuning range of lasing wavelengths along with high photostability, and can serve as a thermal probe [1] [2</p>
    Formula:C22H33BF2N2
    Color and Shape:Solid
    Molecular weight:374.32

    Ref: TM-T78457

    ne
    Discontinued
    Discontinued product
  • (D)-PPA 1

    CAS:
    <p>PD-1/PD-L1 binder, Kd 0.51 μM; blocks interaction in flow cytometry at 1 mg/mL; inhibits tumors, extends mouse survival.</p>
    Formula:C70H98N20O21
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1555.67

    Ref: TM-TP1960

    1mg
    Discontinued
    Discontinued product
  • Antibacterial agent 28

    CAS:
    <p>Antibacterial agent 28 targets MRSA with 0.5-2 μg/mL MIC, showing high potential.</p>
    Formula:C40H64Br2N4O4
    Color and Shape:Solid
    Molecular weight:824.77

    Ref: TM-T40301

    25mg
    Discontinued
    Discontinued product
  • Pomalidomide-amido-PEG3-C2-NH2

    CAS:
    <p>Cereblon Ligand-Linker 22: A pomalidomide-based E3 ligase conjugate with a PEG3 linker for PROTACs.</p>
    Formula:C22H28N4O8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:476.48

    Ref: TM-T18553

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    Discontinued
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    Discontinued product
  • HDAC3/6-IN-2

    CAS:
    <p>HDAC3/6-IN-2 inhibits HDAC6/3 with IC50s 0.368/0.635 μM; promotes cancer cell apoptosis and histone acetylation.</p>
    Formula:C49H67N5O6
    Color and Shape:Solid
    Molecular weight:822.09

    Ref: TM-T74003

    5mg
    Discontinued
    50mg
    Discontinued
    Discontinued product
  • HJM-561

    CAS:
    <p>HJM-561 is a potent and selective EGFR PROTAC with oral bioavailability, capable of overcoming osimertinib-resistant EGFR triple mutations and demonstrating</p>
    Formula:C45H51ClN9O5P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:864.37

    Ref: TM-T82193

    5mg
    Discontinued
    50mg
    Discontinued
    Discontinued product
  • 7-(Diethylamino)-4-methyl-2H-chromen-2-one

    CAS:
    <p>7-(Diethylamino)-4-methyl-2H-chromen-2-one is a useful organic compound for research related to life sciences.</p>
    Formula:C14H17NO2
    Color and Shape:Solid
    Molecular weight:231.30

    Ref: TM-T66262

    ne
    Discontinued
    Discontinued product
  • m-PEG11-Tos


    <p>m-PEG11-Tos is a PEG-based PROTAC linker that can be used in the synthesis of PROTACs[1].</p>
    Formula:C28H50O13S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:626.75

    Ref: TM-T18131

    100mg
    Discontinued
    500mg
    Discontinued
    Discontinued product
  • Fungicide5

    CAS:
    <p>Fungicide5 is a fungicide candidate targeting succinate dehydrogenase ( K i = 0.095 μM).</p>
    Formula:C20H13F8N3O2
    Color and Shape:Solid
    Molecular weight:479.33

    Ref: TM-T39882

    25mg
    Discontinued
    Discontinued product
  • NT 2 Toxin

    CAS:
    <p>NT 2 Toxin is a useful organic compound for research related to life sciences. The catalog number is T124258 and the CAS number is 76348-84-0.</p>
    Formula:C17H24O7
    Color and Shape:Solid
    Molecular weight:340.372

    Ref: TM-T124258

    1mg
    Discontinued
    5mg
    Discontinued
    Discontinued product
  • 5'-O-TBDMS-dT

    CAS:
    <p>5’-O-TBDMS-dT is a nucleoside with protective and modification effects.</p>
    Formula:C16H28N2O5Si
    Color and Shape:Solid
    Molecular weight:356.49

    Ref: TM-T37145

    1ml*10 (DMSO)
    Discontinued
    1mL*10mM (DMSO)_old
    Discontinued
    Discontinued product
  • Telmisartan Acyl-β-D-Glucuronide

    CAS:
    <p>Telmisartan acyl-β-D-glucuronide is a major metabolite of the angiotensin II receptor antagonist telmisartan .</p>
    Formula:C39H38N4O8
    Color and Shape:Solid
    Molecular weight:690.753

    Ref: TM-T35865

    1mg
    Discontinued
    Discontinued product
  • PYBG

    CAS:
    <p>PYBG serves as a flexible precursor for facile conjugation with diverse fluorescent dyes using 'Click chemistry' and Sonogashira coupling reactions.</p>
    Formula:C16H15N5O2
    Color and Shape:Solid
    Molecular weight:309.329

    Ref: TM-T40788

    ne
    Discontinued
    Discontinued product
  • PROTAC PARP/EGFR ligand 1

    CAS:
    <p>PROTAC PARP/EGFR ligand 1 enables dual PARP EGFR degrader synthesis via PROTAC.</p>
    Formula:C53H56ClF2N9O8
    Color and Shape:Solid
    Molecular weight:1020.52

    Ref: TM-T74173

    5mg
    Discontinued
    50mg
    Discontinued
    Discontinued product
  • Pulcherriminic acid

    CAS:
    <p>Pulcherriminic acid, a cyclic dipeptide, chelates Fe3+, forms pulcherrimin, and has antimicrobial properties used in food, agriculture, and medicine.</p>
    Formula:C12H20N2O4
    Color and Shape:Solid
    Molecular weight:256.30

    Ref: TM-T75509

    5mg
    Discontinued
    50mg
    Discontinued
    Discontinued product