CAS 130049-85-3
:Sortieren nach
Reinheit (%)
0
100
|
0
|
50
|
90
|
95
|
100
8 Produkte.
Risperidone EP Impurity C ((R)-Isomer)-d4 ((R)-9-Hydroxy Risperidone-d4, (R)-Paliperidone-d4)
CAS:Formel:C23H23D4FN4O3Farbe und Form:Pale Yellow SolidMolekulargewicht:430.52Risperidone EP Impurity C ((R)-Isomer) ((R)-9-Hydroxy Risperidone, (R)-Paliperidone)
CAS:Formel:C23H27FN4O3Farbe und Form:Pale Yellow SolidMolekulargewicht:426.49(R)-9-Hydroxy Risperidone-d4
CAS:Kontrolliertes ProduktFormel:C23H23D4FN4O3Farbe und Form:NeatMolekulargewicht:430.51(+)-9-Hydroxyrisperidone
CAS:Kontrolliertes Produkt(+)-9-Hydroxyrisperidone is an active metabolite of risperidone, which is an atypical antipsychotic. It functions as a dopamine (D2) receptor antagonist and serotonin (5-HT2A) receptor antagonist. The (+)-9-hydroxyrisperidone binds to the D2 receptor in the brain and prevents dopamine from binding, thereby blocking dopamine D2 receptors. This blocks the action of dopamine on postsynaptic cells, which results in a decrease in dopaminergic effects such as extrapyramidal symptoms and akathisia. In addition, (+)-9-hydroxyrisperidone binds to serotonin 5-HT2A receptors and blocks serotonin from binding, thereby blocking serotonin effects such as hallucinations and suicidal thoughts.Formel:C23H27FN4O3Reinheit:Min. 95%Farbe und Form:PowderMolekulargewicht:426.48 g/mol(R)-9-Hydroxy Risperidone
CAS:Kontrolliertes ProduktApplications The R-enantiomer metabolite of Risperidone (R525000), a combined serotonin (5-HT2) and dopamine (D2) receptor antagonist.
Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package
References Tiberghien, F., et al.: Anticancer Drugs, 7, 568 (1996), Kansy, M., et al.: J. Med. Chem., 41, 1007 (1998), Kerns, E., et al.: J. Pharm. Sci., 90, 1838 (2001), Kerr, K., et al.: J. Biol. Chem., 276, 8657 (2001), Doran, A., et al.: Drug Metab. Dispos., 33, 165 (2005),Formel:C23H27FN4O3Farbe und Form:NeatMolekulargewicht:426.48
