CAS 2056261-42-6

BRD5648

CAS: 2056261-42-6

BRD5648

Reinheit: ≥98%

Molekulargewicht: 321.42g/mol

Ref: 54-BUP14260

(4R)-4-Ethyl-7,7-dimethyl-4-phenyl-1,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-one

CAS: 2056261-42-6

4-Ethyl-7,7-dimethyl-4-phenyl-1,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-one (EDQ) is a potent inhibitor of the voltage dependent ion channels. It has been shown to be an effective inhibitor of the Na+ and Ca2+ channels in mammalian cells. EDQ binds to the extracellular loops of these channels and inhibits their function by blocking the opening of the channel pore. The inhibition of these ion channels leads to a decrease in neurotransmitter release and prevents neuronal depolarization. This compound can be used as a research tool for studying cell biology, peptides, pharmacology and ligands. It is also used as a reagent for testing receptor activation with high purity.

Formel: C₂₀H₂₃N₃O

Reinheit: Min. 95%

Molekulargewicht: 321.4 g/mol

Ref: 3D-GHD26142

BRD5648

CAS: 2056261-42-6

BRD5648 ((R)-BRD0705) is an inactive (R)-enantiomer of BRD0705.

Formel: C₂₀H₂₃N₃O

Reinheit: 99.89%

Farbe und Form: Solid

Molekulargewicht: 321.42

Ref: TM-T10608