CAS 2251753-58-7

N-[2-[[[1-[[(4-Fluorophenyl)amino]carbonyl]cyclopropyl]carbonyl]amino]ethyl]-2-methylene-3-oxoolean-12-en-28-amide

CAS: 2251753-58-7

N-[2-[[[1-[[(4-Fluorophenyl)amino]carbonyl]cyclopropyl]carbonyl]amino]ethyl]-2-methylene-3-oxoolean-12-en-28-amide is a research tool for the study of protein interactions and the development of new drugs. It has shown to be a potent inhibitor of ion channels, including voltage gated sodium channels. This compound binds to the extracellular domain of these channels and prevents activation, leading to inhibition of nerve impulse transmission. N-[2-[[[1-[[(4-Fluorophenyl)amino]carbonyl]cyclopropyl]carbonyl]amino]ethyl]-2-methylene-3-oxoolean-12-en-28 amide also inhibits ligand binding to its receptor by binding in an allosteric site that is distinct from the active site.

Formel: C₄₄H₆₀FN₃O₄

Reinheit: Min. 95%

Molekulargewicht: 714.00 g/mol

Ref: 3D-BQD75358

CAY10735

CAS: 2251753-58-7

CAY10735: Anticancer agent; inhibits growth/migration in various cancer cells; reduces tumor in mouse models. IC50=0.674-11.56μM.

Formel: C₄₄H₆₀FN₃O₄

Farbe und Form: Solid

Molekulargewicht: 713.979

Ref: TM-T36497