Melatoninrezeptor
Los receptores de ácido lisofosfatídico (LPA) son un grupo de GPCR que responden al LPA, un lípido bioactivo involucrado en la proliferación, migración y supervivencia celular. La señalización de LPA juega un papel crucial en varios procesos fisiológicos, incluyendo la cicatrización de heridas, el desarrollo vascular y la metástasis del cáncer. La modulación de la actividad de los receptores de LPA se está explorando para aplicaciones terapéuticas en el cáncer, la fibrosis y las enfermedades inflamatorias. En CymitQuimica, ofrecemos una gama de moduladores de receptores de LPA de alta calidad para apoyar su investigación en señalización celular, oncología y trastornos inflamatorios.
24 Produkte aus dem Bereich "Melatoninrezeptor" gefunden
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Agomelatine
CAS:<p>Agomelatine (Valdoxan), like melatonin, boosts mood by targeting melatonin and 5-HT2C receptors.</p>Formel:C15H17NO2Reinheit:99.92%Farbe und Form:White SolidMolekulargewicht:243.3Ramelteon
CAS:<p>Ramelteon (TAK-375) is a Melatonin Receptor Agonist. The mechanism of action of ramelteon is as a Melatonin Receptor Agonist.</p>Formel:C16H21NO2Reinheit:97.21% - 99.92%Farbe und Form:Crystalline SolidMolekulargewicht:259.34Luzindole
CAS:<p>Luzindole (N-0774) is a selective melatonin receptor antagonist.</p>Formel:C19H20N2OReinheit:98.53%Farbe und Form:Off-White Amorphous SolidMolekulargewicht:292.37Melatonin-Tamoxifen Conjugate
<p>Melatonin-Tamoxifen Conjugate (compound 16c) is an anticancer drug conjugate made of Melatonin and Tamoxifen, serving as an effective antagonist of ERα (IC50 = 863 nM). In cells expressing the hMT1 receptor, it binds to MLT receptors (Ki = 3.1 nM) and exhibits the ability to promote β-arrestin activation (EC50 = 914 nM) and ERK activation (EC50 = 98 nM). The IC50 values for Melatonin-Tamoxifen Conjugate in MCF-7, MDA-MB-231, and HT-1080 cell lines are 6.8 μM, 6.4 μM, and 1.7 μM, respectively.</p>Formel:C47H58N4O4Farbe und Form:SolidMolekulargewicht:742.99UCM 549
CAS:<p>UCM 549 is a bioactive chemical.</p>Formel:C19H21NO2Farbe und Form:SolidMolekulargewicht:295.384-P-PDOT
CAS:<p>4-P-PDOT (4-phenyl-2- propionamidotetralin) is a potent, selective and affinity Melatonin receptor (MT2) antagonist.</p>Formel:C19H21NOReinheit:99.91%Farbe und Form:SolidMolekulargewicht:279.38Histamine & Melatonin Receptor-Targeted Compound Library
<p>A unique collection of xnum compounds targeting histaminergic receptor and melatonin receptor for high throughput screening (HTS) and high content screening (HCS</p>Farbe und Form:Odour SolidRamelteon-d5
CAS:<p>Ramelteon-d5 is a deuterated compound of Ramelteon.</p>Formel:C16H16D5NO2Farbe und Form:SolidMolekulargewicht:264.37N-ACETYLTRYPTAMINE
CAS:<p>N-ACETYLTRYPTAMINE is a partial agonist for melatonin receptors in the retina. Also used for determination of serotonin N-acetyl transferase.</p>Formel:C12H14N2OReinheit:98.79%Farbe und Form:PowderMolekulargewicht:202.25Tasimelteon
CAS:<p>Tasimelteon (BMS-214778) is a melatonin receptor agonist that is used for the treatment of non-24 hour sleep-wake disorder in blind individuals.</p>Formel:C15H19NO2Reinheit:98.93% - 99.93%Farbe und Form:SolidMolekulargewicht:245.32S26131
CAS:<p>S26131 (N-[2-[7-[3-[8-(2-acetamidoethyl)naphthalen-2-yl]oxypropoxy]naphthalen-1-yl]ethyl]acetamide) behaves as an antagonist on MT1 and MT2 receptors with Ki of</p>Formel:C31H34N2O4Reinheit:99.77%Farbe und Form:SolidMolekulargewicht:498.61Melatonin
CAS:<p>Melatonin (Melatonine) is a natural hormone that activates melatonin receptors. Melatonin regulates the biological clock. Cost-effective and quality-assured.</p>Formel:C13H16N2O2Reinheit:98% - 99.89%Farbe und Form:Pale Yellow Leaflets From Benzene SolidMolekulargewicht:232.28ACH-000143
CAS:<p>ACH-000143 是一种可口服的褪黑素受体激动剂，对 MT1 和 MT2 的EC50值分别为0.06 和0.32 nM。</p>Formel:C13H16ClN3O3Reinheit:98.15%Farbe und Form:SolidMolekulargewicht:297.74UCM 608
CAS:<p>UCM 608 (2-Phenylmelatonin) is an antagonist of melatonin-induced contractile responses at low concentrations and induces an increase in GDP-GTP exchange.</p>Formel:C19H20N2O2Reinheit:98.88%Farbe und Form:SolidMolekulargewicht:308.37DH97
CAS:<p>MT2 melatonin receptor antagonist</p>Formel:C22H26N2OReinheit:98%Farbe und Form:SolidMolekulargewicht:334.45S20928
CAS:<p>S20928 is an antagonist of melatonin receptor.</p>Formel:C17H19NOFarbe und Form:SolidMolekulargewicht:253.34Melatonin receptor agonist 1
CAS:<p>Melatonin receptor agonist 1 (compound 20c) is a potent agonist of melatonin receptor (MT) with Ki values of 108 nM for MT2 and 1140 nM for MT 1 [1].</p>Formel:C15H19N3O2Farbe und Form:SolidMolekulargewicht:273.338-M-PDOT
CAS:<p>8-M-PDOT (AH-002) is an MT2 receptor agonist that inhibits MT1.8-M-PDOT has anxiolytic activity and may be used in the study of neuropathic pain.</p>Formel:C14H19NO2Reinheit:99.54% - 99.54%Farbe und Form:SolidMolekulargewicht:233.312-Iodomelatonin
CAS:<p>2-Iodomelatonin, Ki 28 pM, is an MT1 agonist, >5x selective over MT2, used to map melatonin sites in brain/tissues.</p>Formel:C13H15IN2O2Reinheit:99.7%Farbe und Form:SolidMolekulargewicht:358.17GR 196429
CAS:<p>GR 196429: MT1-selective melatonin receptor agonist; induces sleep, alters circadian rhythm, stimulates melatonin in mice.</p>Formel:C14H18N2O2Reinheit:98%Farbe und Form:SolidMolekulargewicht:246.3
