E 52862 (S1RA)

CAS: 878141-96-9

Ref. 3D-BE177449

Produktinformation

• Name: E 52862 (S1RA)
• Synonyme: E 52862, MR-309, 4-[2-[[5-Methyl-1-(2-naphthalenyl)-1H-pyrazol-3-yl]oxy]ethyl]morpholine, S1RA, Morpholine, 4-[2-[[5-methyl-1-(2-naphthalenyl)-1H-pyrazol-3-yl]oxy]ethyl]-

Beschreibung

E 52862 (S1RA) is a monoclonal antibody that targets the α2δ subunit of voltage-gated calcium channels. It blocks the binding of ATP and reduces neuronal excitability, providing antinociception without causing dependence or addiction. E 52862 has been shown to be an effective treatment for diabetic neuropathy in vivo models. The drug has also been shown to have a sub-effective dose, which may reduce its side effects. E 52862's receptor activity may be due to its ability to inhibit glutamate release and cyclin D2 expression, which are both involved in pain transmission.

• Marke: Biosynth

Chemische Eigenschaften

• Molekulargewicht: 337.42 g/mol
• Formel: C₂₀H₂₃N₃O₂
• Reinheit: Min. 95%