Bazedoxifene 5-β-D-glucuronide

CAS: 328933-56-8

Ref. 3D-DNA93356

Produktinformation

• Name: Bazedoxifene 5-β-D-glucuronide

Beschreibung

Bazedoxifene 5-β-D-glucuronide is an analog of bazedoxifene, a selective estrogen receptor modulator used in the treatment of osteoporosis. This compound has shown promising anticancer properties and has been studied extensively in Chinese hamster ovary cells. Bazedoxifene 5-β-D-glucuronide has been found to induce apoptosis in cancer cells and inhibit the activity of kinases involved in tumor growth. It is a potent inhibitor of several human protein kinases, including cyclin-dependent kinase 2 (CDK2) and glycogen synthase kinase 3 beta (GSK3β), which are important targets for medicinal chemists developing kinase inhibitors. This compound is excreted primarily in urine and may have potential as a therapeutic agent for various types of cancer.

• Marke: Biosynth

Chemische Eigenschaften

• Molekulargewicht: 646.7 g/mol
• Formel: C₃₆H₄₂N₂O₉
• Reinheit: Min. 95%
• Farbe/Form: Powder