5-Methylgramine

CAS: 30218-58-7

Ref. 3D-FM52381

Produktinformation

• Name: 5-Methylgramine
• Synonyme: 3-(Dimethylaminomethyl)-5-methylindole, Indole, 3-(dimethylamino)methyl-5-methyl-, Brn 0144975, Nsc 88884, 1H-Indole-3-methanamine, N,N,5-trimethyl- (9CI), N,N-dimethyl-1-(5-methyl-1H-indol-3-yl)methanamine

Beschreibung

5-Methylgramine is a centrally acting adrenergic (5-HT) receptor antagonist that is used for the treatment of allergic disorders and as an antiemetic. It has been shown to be effective in treating allergic rhinitis, urticaria, and pruritus. 5-Methylgramine blocks the binding of 5-hydroxytryptamine at the peripheral 5-ht receptors and also antagonizes the action of endogenous or exogenous histamine at central 5-ht receptors. It has been shown to have a maximal effect on the constrictor responses mediated by the adventitia in guinea pigs. The drug can be given orally or intravenously.

• Marke: Biosynth

Chemische Eigenschaften

• Molekulargewicht: 188.27 g/mol
• Formel: C₁₂H₁₆N₂
• Reinheit: Min. 95%