Pepstatin A

CAS: 26305-03-3

Ref. 3D-FP29630

Produktinformation

• Name: Pepstatin A
• Synonyme: pepstatin A from microbial source, Pepstatin (microbial product), Isovaleryl-Val-Val-Sta-Ala-Sta-OH, N-(3-methylbutanoyl)-L-valyl-N-[(1S,2S)-4-{[(1S)-2-({(1S)-1-[(1S)-2-carboxy-1-hydroxyethyl]-3-methylbutyl}amino)-1-methyl-2-oxoethyl]amino}-2-hydroxy-1-(2-methylpropyl)-4-oxobutyl]-L-valinamide, (3S,4R)-3-hydroxy-4-[[(2R)-2-[[(3R,4S)-3-hydroxy-6-methyl-4-[[(2R)-3-methyl-2-[[(2R)-3-methyl-2-(3-methylbutanoylamino)butanoyl]amino]butanoyl]amino]heptanoyl]amino]propanoyl]amino]-6-methyl-heptanoic acid, Pepstatin

Beschreibung

Pepstatin A is a natural product that inhibits the activity of aspartyl proteases. It has inhibitory effects on the mitochondrial membrane potential and can be used to study the protein-protein interactions involved in signal transduction. Pepstatin A also interacts with other drugs and can inhibit their action, which may lead to drug interactions. Moreover, it is a potent inducer of platelet aggregation and has been shown to be effective in experimental models of inflammation. Pepstatin A is found in many biological samples, such as human plasma and rat liver extracts, and wild-type strains are resistant to its inhibitory effects.

• Marke: Biosynth

Chemische Eigenschaften

• Molekulargewicht: 685.90 g/mol
• Formel: C₃₄H₆₃N₅O₉
• Reinheit: Min. 98 Area-%
• Farbe/Form: Powder