Sarafotoxin 6c

CAS: 121695-87-2

Ref. 3D-FS73598

Produktinformation

• Name: Sarafotoxin 6c
• Synonyme: Srtx-C, Sarafotoxin S6C (Atractaspis Engaddensis), Sarafotoxin S6C, Atractaspsis Engaddensis, Sarafotoxin 6C, Sarafotoxin C, Sarafotoxin C (Atractaspis Engaddensis), Cys-Thr-Cys-Asn-Asp-Met-Thr-Asp-Glu-Glu-Cys-Leu-Asn-Phe-Cys-His-Gln-Asp-Val-Ile-Trp

Beschreibung

Sarafotoxin 6c is a potent, selective, and noncompetitive endothelin-1 receptor antagonist. Sarafotoxin 6c binds to the extracellular domain of the endothelin-1 receptor and prevents endothelin-1 from binding, thereby inhibiting its activity. Sarafotoxin 6c has been shown to inhibit the production of intracellular Ca2+ in mesenteric artery cells. Sarafotoxin 6c also inhibits the enzymatic inactivation of endothelin-1 by carboxypeptidases and calpains. Sarafotoxin 6c has been shown to be effective against a number of infectious diseases including myocardial infarction.

• Marke: Biosynth

Chemische Eigenschaften

• Molekulargewicht: 2,515.76 g/mol
• Formel: C₁₀₃H₁₄₇N₂₇O₃₇S₅
• Reinheit: Min. 95%