Tianeptine sodium salt

CAS: 30123-17-2

Ref. 3D-FT28266

Produktinformation

• Name: Tianeptine sodium salt
• Synonyme: 7-[(3-Chloro-6,11-dihydro-6-methyldibenzo[c,f][1,2]thiazepin-11-yl)amino]heptanoic acid S,S-dioxide sodium saltS-1574Stablon
• Marke: Biosynth
• Beschreibung: Full agonist of the μ-opioid receptor (MOR) with Ki of 383 nM. It also weakly agonizes the δ-opioid receptor (DOR) with a Ki >10 μM. Tianeptine has antidepressant effects but can also regulate neuroplasticity in the amygdala and stress-induced release of glutamate. It can generate analgesia and reward, typical opiate-like behavioural effects, but does not induce tolerance or withdrawal.

Chemische Eigenschaften

• Molekulargewicht: 458.93 g/mol
• Formel: C₂₁H₂₄ClN₂NaO₄S
• Reinheit: Min. 98.5 Area-%
• Farbe/Form: White Slightly Yellow Powder