(±)-WS 75624b

CAS: 188048-45-5

Ref. 3D-NHA04845

Produktinformation

• Name: (±)-WS 75624b
• Synonyme: Ws-75624B

Beschreibung

(±)-WS 75624b is a potent and selective activator of the human serotonin 5-HT2C receptor. The binding affinity of (±)-WS 75624b to the human serotonin 5-HT2C receptor was determined by measuring the Ki value with radioligand binding assays using [3H]-mesulergine as the radioligand. The Ki value for (±)-WS 75624b was determined to be 0.8 nM, which is in good agreement with the Ki values reported for other serotonin 5-HT2C receptor agonists.

(±)-WS 75624b binds to the serotonin 5-HT2C receptor with high affinity and selectivity, and it has been shown to activate this receptor in a number of cell types. It has been found to inhibit voltage-gated potassium currents in rat dorsal root ganglion neurons and also inhibits glutamate release from cultured rat cortical cells. These properties make

• Marke: Biosynth

Chemische Eigenschaften

• Molekulargewicht: 380.5 g/mol
• Formel: C₁₈H₂₄N₂O₅S
• Reinheit: Min. 95%