JTC-801

CAS: 244218-51-7

Ref. 3D-UJA21851

Produktinformation

• Name: JTC-801
• Synonyme: Jtc-801
• CAS: 244218-51-7

Beschreibung

JTC-801 is a selective agonist for the κ-opioid receptors and has been shown to inhibit the proliferation of tumor cells in vitro. It binds to κ-opioid receptors on the surface of cells and activates these receptors, which causes an increase in cytosolic calcium. This drug also inhibits the pro-apoptotic protein Bax, leading to apoptosis (cell death). JTC-801 has been shown to have a low toxicity profile in mice and does not cross the blood brain barrier. It also has been found to have a similar affinity for δ-opioid receptors as morphine and shows anti-inflammatory effects by inhibiting prostaglandin synthesis.

• Marke: Biosynth

Chemische Eigenschaften

• Molekulargewicht: 447.96 g/mol
• Formel: C₂₆H₂₅N₃O₂·HCl
• Reinheit: Min. 95%