Methyl 5-fluoro-2-(2-(1-methyl-1H-1,2,4-triazol-5-yl)acetyl)-3-nitrobenzoate

CAS: 1322879-81-1

Ref. 3D-XCC87981

Produktinformation

• Name: Methyl 5-fluoro-2-(2-(1-methyl-1H-1,2,4-triazol-5-yl)acetyl)-3-nitrobenzoate

Beschreibung

Methyl 5-fluoro-2-(2-(1-methyl-1H-1,2,4-triazol-5-yl)acetyl)-3-nitrobenzoate is a cell permeable inhibitor of the protease cathepsin B. It has been used as a research tool to study the protein interactions of this enzyme. Methyl 5-fluoro-2-(2-(1-methyl-1H-1,2,4-triazol-5-yl)acetyl)-3-nitrobenzoate is also an inhibitor of other proteinases and peptidases. The inhibition is reversible and competitive. The inhibition constant (Ki) for this drug are in the range of 0.02 - 1 µM. This compound has been shown to be an activator of G proteins by binding to the regulatory domain on the alpha subunit with high affinity and specificity. Methyl 5 - fluoro - 2 - (

• Marke: Biosynth

Chemische Eigenschaften

• Molekulargewicht: 322.25 g/mol
• Formel: C₁₃H₁₁FN₄O₅
• Reinheit: Min. 95%