Selonsertib hydrochloride

CAS: 1448428-05-4

Ref. 3D-YHC42805

Produktinformation

• Name: Selonsertib hydrochloride

Beschreibung

Selonsertib is a small molecule that inhibits the serine/threonine kinase RSK2. It has been shown to inhibit the proliferation of cells and induce cell death in vitro. Selonsertib selectively binds to the ATP-binding site of RSK2, which is essential for its function as a protein kinase, and prevents it from phosphorylating other proteins on threonine and serine residues. Selonsertib also inhibits the activity of TGF-β1, a cytokine that can cause tumor growth.

Selonsertib hydrochloride is an inhibitor of receptor tyrosine kinases (RTKs) such as insulin-like growth factor 1 receptor (IGF-1R), vascular endothelial growth factor receptor 2 (VEGFR2), platelet-derived growth factor receptor β (PDGFRβ), or fibroblast growth factor receptor 2 (FGFR2). Selonsertib hydrochloride is

• Marke: Biosynth

Chemische Eigenschaften

• Molekulargewicht: 482 g/mol
• Formel: C₂₄H₂₅ClFN₇O
• Reinheit: Min. 95%