Irdabisant

CAS: 1005402-19-6

Ref. TM-T32191

Produktinformation

• Name: Irdabisant
• Synonyme: CEP-26401, CEP 26401, CEP26401
• CAS: 1005402-19-6

Beschreibung

Irdabisant (CEP-26401) (CEP-26401) is a selective, orally active and blood-brain barrier (BBB) penetrant antagonist/inverse agonist of histamine H3 receptor (H3R) (rat H3R Ki= 7.2 nM, human H3R Ki= 2.0 nM). Irdabisant exhibits relatively low inhibitory activity against hERG current (IC50= 13.8 μM). Irdabisant exhibits cognition-enhancing and wake-promoting activities in the rat social recognition model. Irdabisant can be used for research on schizophrenia or cognitive impairment.

• Marke: Targetmol

Chemische Eigenschaften

• Molekulargewicht: 313.39
• Formel: C₁₈H₂₃N₃O₂
• Reinheit: 99.77%
• Farbe/Form: Solid