AZD1283

CAS: 919351-41-0

Ref. TM-T3536

Produktinformation

• Name: AZD1283
• Synonyme: AZD-1283
• CAS: 919351-41-0

Beschreibung

AZD1283 is an effective P2Y12 receptor antagonist (EC50: 3.0 ug/kg/min, binding IC50: 11 nM). AZD1283 dose-dependently induced increases in blood flow and inhibition of ADP-induced platelet aggregation with antithrombotic ED50 values of 3.0 and 10 μg/kg/min, respectively. The doses induced the increase in bleeding time at 33 and 100 μg/kg/min for 3- and 13-fold, respectively. Thus, the therapeutic index (TI) was ≥10 for both compounds.

• Marke: Targetmol

Chemische Eigenschaften

• Molekulargewicht: 470.54
• Formel: C₂₃H₂₆N₄O₅S
• Reinheit: 99.621%
• Farbe/Form: Solid