KH-4-43

CAS: 2813310-07-3

Ref. TM-T84685

Produktinformation

• Name: KH-4-43
• Marke: Targetmol
• Beschreibung: KH-4-43, an inhibitor of the E3 CRL4 ligase complex, demonstrates anticancer activity by targeting the core of the E3 CRL4. It exhibits a binding affinity (Kd) of 83 nM to the E3 ROC1-CUL4A CTD and 9.4 μM to the closely related ROC1-CUL1 CTD [1].

Chemische Eigenschaften

• Molekulargewicht: 422.74
• Formel: C₁₉H₁₀ClF₃N₂O₄
• Farbe/Form: Solid