EGFR kinase inhibitor 3

CAS: 2922402-03-5

Ref. TM-T86341

Produktinformation

• Name: EGFR kinase inhibitor 3
• Marke: Targetmol
• Beschreibung: EGFR kinase inhibitor 3 (compound 2) serves as a dual-action inhibitor targeting both ATP and allosteric sites of the EGFR kinase, exhibiting potent IC50 values of less than 10 nM for wild-type EGFR, 1.5 nM for the L858R mutation, 0.059 nM for the L858R/T790M mutation, and 0.064 nM for the L858R/T790M/C797S mutation. It is classified as a C-linked inhibitor [1].

Chemische Eigenschaften

• Molekulargewicht: 575.64
• Formel: C₃₁H₂₅N₇O₃S
• Farbe/Form: Solid