N-(3-Butenyl)norbuprenorphine

CAS: 457071-73-7

Ref. TR-B690070

Produktinformation

• Name: N-(3-Butenyl)norbuprenorphine
• Synonyme: (αS,5α,7α)-17-(3-Buten-1-yl)-α-(1,1-dimethylethyl)-4,5-epoxy-18,19-dihydro-3-hydroxy-6-methoxy-α-methyl-6,14-ethenomorphinan-7-methanol, 6,14-Ethenomorphinan-7-methanol, 17-(3-butenyl)-α-(1,1-dimethylethyl)-4,5-epoxy-18,19-dihydro-3-hydroxy-6-methoxy-α-methyl-, (αS,5α,7α)- (9CI), (2S)-2-[17-(But-3-enyl)-4,5α-epoxy-3-hydroxy-6-methoxy-6α,14-ethano-14α-morphinan-7α-yl]-3,3-dimethylbutan-2-ol, N-But-3-enylnorbuprenorphine, Buprenorphine Imp. A (EP)
• CAS: 457071-73-7

Beschreibung

Applications An impurity in the synthesis of Buprenorphine (B689570), which is a controllled substance (narcotic). Analgesic that demonstrates narcotic agonist-antagonist properties.
References Martin, W.R., et al.: J. Pharmacol. Exp. Ther., 197, 517 (1976), Rance, M.J., Biochem. Pharmacol., 25, 735 (1976), Heel, R.C., et al.: Drugs, 17, 81 (1979),

• Marke: TRC

Chemische Eigenschaften

• Molekulargewicht: 467.64
• Formel: C₂₉H₄₁NO₄
• Farbe/Form: White To Light Yellow
• InChl: InChI=1S/C29H41NO4/c1-7-8-14-30-15-13-28-22-18-9-10-19(31)23(22)34-24(28)29(33-6)12-11-27(28,21(30)16-18)17-20(29)26(5,32)25(2,3)4/h7,9-10,20-21,24,31-32H,1,8,11-17H2,2-6H3/t20-,21-,24-,26+,27-,28+,29?/m1/s1