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Unter den Marken unserer mehr als 25 Partner sticht TargetMol hervor

Unter den Marken unserer mehr als 25 Partner sticht TargetMol hervor

We have reached an agreement with TargetMol: CymitQuimica clients will benefit for a 20% discount on all TargetMol products until the end of the year.On our website you can find the products offered by this partner, which has become one of the world's most recognised compound libraries and small molecule inhibitors supplier. TargetMol offers approximately 120 compound libraries and a wide range of chemical products and kits for life sciences.

Endet am 31. Dez.( 8 verbleibende Tage )

Produkte pro Seite.111931 Produkte in dieser Werbeaktion.
  • Eberconazole

    CAS:
    Eberconazole, a potent antifungal, is an imidazole derivative effective against dermatophytes. Administered topically.
    Formel:C18H14Cl2N2
    Farbe und Form:Solid
    Molekulargewicht:329.22
  • Justicidin B

    CAS:
    Justicidin B: anticancer, proapoptotic, inhibits bone resorption & platelets, antiviral, fungicidal, antiprotozoal.
    Formel:C21H16O6
    Farbe und Form:Solid
    Molekulargewicht:364.35
  • D-threo-PDMP

    CAS:
    D-threo-PDMP inhibits glucoceramide synthase, cutting cell surface glycosphingolipids and hindering neurite growth.
    Formel:C23H38N2O3
    Farbe und Form:Solid
    Molekulargewicht:390.56
  • JNJ-49095397

    CAS:
    <p>JNJ-49095397 (RV568) is a p38 MAPK-α and p38 MAPK-γ kinase inhibitor for the study of respiratory syncytial virus infection.</p>
    Formel:C34H36N6O4
    Reinheit:98.33% - 99.04%
    Farbe und Form:Solid
    Molekulargewicht:592.69
  • PKCiota-IN-1

    CAS:
    <p>PKCiota-IN-1: Strong PKC-ι inhibitor (IC50=2.7 nM); also blocks PKC-α/ε (IC50s=45/450 nM).</p>
    Formel:C25H22FN5O
    Farbe und Form:Solid
    Molekulargewicht:427.47
  • FITM

    CAS:
    FITM is a potent negative allosteric modulator of mGlu1 receptor(Ki : 2.5 nM).
    Formel:C18H18FN5OS
    Reinheit:97.25%
    Farbe und Form:Solid
    Molekulargewicht:371.43
  • Azaphilone-9

    CAS:
    <p>AZA-9 inhibits cancer growth by blocking HuR-ARE RNA binding; IC50=1.2μM.</p>
    Formel:C21H23BrO5
    Farbe und Form:Solid
    Molekulargewicht:435.31
  • TNKS1/2-IN-1

    CAS:
    <p>TNKS1/2-IN-1: potent inhibitor for cancer, fibrosis research; pIC50 7.1-8.2.</p>
    Formel:C26H23F4N3O4
    Farbe und Form:Solid
    Molekulargewicht:517.47
  • VEGFR-3-IN-1

    CAS:
    VEGFR-3-IN-1, a potent VEGFR3 inhibitor (IC50=110.4 nM), hinders tumor growth and VEGFR3 signaling, affecting HDLEC and MDA-MB cell proliferation/migration.
    Formel:C29H29ClF3N7OS
    Reinheit:99.95%
    Farbe und Form:Solid
    Molekulargewicht:616.1
  • Naloxonazine

    CAS:
    <p>Naloxonazine, a potent, selective opiate mu-1 (μ1) antagonist, also influences leishmania through the modulation of host coding function.</p>
    Formel:C38H42N4O6
    Farbe und Form:Solid
    Molekulargewicht:650.76
  • IMD-vanillin

    CAS:
    IMD-vanillin is a novel compound characterized as an imidazoquinolinone-derived dimer with NF-κB immunomodulatory properties.
    Formel:C37H45N7O4
    Reinheit:98%
    Farbe und Form:Solid
    Molekulargewicht:651.8
  • IMD-catechol

    CAS:
    IMD-catechol: an imidazoquinolinone-based dimer with NF-κB activity; improves CT26 cancer treatment, low toxicity.
    Formel:C31H34N6O3
    Reinheit:98%
    Farbe und Form:Solid
    Molekulargewicht:538.64
  • CDK4/6-IN-15

    CAS:
    CDK4/6-IN-15: Oral, selective CDK4/6 inhibitor, halts cancer cell growth, G1 arrest, suppresses Rb phosphorylation.
    Formel:C21H27FN8S
    Farbe und Form:Solid
    Molekulargewicht:442.56
  • 18:0-22:6 DG

    CAS:
    1-Stearoyl-2-docosahexaenoyl-sn-glycerol (18:0-22:6 DG) is a diacylglycerol capable of binding to RasGRP and modulating the activation of MAP kinases.
    Formel:C43H72O5
    Farbe und Form:Solid
    Molekulargewicht:669.03
  • EC330

    CAS:
    EC330, a novel steroidal LIF inhibitor showed cytotoxicity in various cancer cell lines and NCI-60 cell line panel at low nano-molar range.
    Formel:C30H32F2O2
    Reinheit:97.83%
    Farbe und Form:Solid
    Molekulargewicht:462.57
  • NCGC00138783


    NCGC00138783 blocks CD47/SIRPα interaction; IC50 of 50 µM.
    Formel:C30H28F7N7O5S
    Farbe und Form:Solid
    Molekulargewicht:731.64
  • TRK/ALK-IN-1


    TRK/ALK-IN-1: Potent dual TRK & ALK inhibitor; IC50s: 2.2nM (TRKA), 9.3nM (ALK WT), 38nM (ALK L1196M); cancer research potential.
    Formel:C31H35ClF2N8O2S
    Farbe und Form:Solid
    Molekulargewicht:657.18
  • Triphen diol

    CAS:
    Triphen diol, a phenol diol, fights pancreatic cancer & cholangiocarcinoma, inducing apoptosis via caspase-dependent & -independent paths.
    Formel:C22H20O4
    Farbe und Form:Solid
    Molekulargewicht:348.39
  • ChemR23-IN-3


    <p>ChemR23-IN-3 is a potent thiazole-based ChemR23 inhibitor with an IC 80 value of 12 nM.</p>
    Formel:C31H33N5O5S2
    Farbe und Form:Solid
    Molekulargewicht:619.75
  • Epothilone E

    CAS:
    <p>Epothilone E, a derivative of epothilone, functions by inhibiting microtubule protein activity, thereby halting cell division and exhibiting anti-tumor</p>
    Formel:C26H39NO7S
    Farbe und Form:Solid
    Molekulargewicht:509.66
  • Aramchol

    CAS:
    Aramchol (C20-FABAC), a mix of arachidic & cholic acid, lessens cholesterol crystallization & dissolves crystals in bile.
    Formel:C44H79NO5
    Reinheit:≥95%
    Farbe und Form:Solid
    Molekulargewicht:702.1
  • eIF4A3-IN-17

    CAS:
    <p>eIF4A3-IN-17, a silvestrol analogue, disrupts eIF4F assembly; EC50: 0.9-15 nM. Used in cancer pathogenesis research.</p>
    Formel:C28H25NO7
    Farbe und Form:Solid
    Molekulargewicht:487.5
  • eIF4A3-IN-18

    CAS:
    eIF4A3-IN-18, a silvestrol analogue with EC50s: 0.8/35/2 nM, inhibits eIF4F complex and is cytotoxic (LC50: 0.06 nM) for cancer research.
    Formel:C29H28N2O6
    Farbe und Form:Solid
    Molekulargewicht:500.54
  • Palazestrant

    CAS:
    Palazestrant, an antiestrogen and antineoplastic agent, effectively targets ER+/HER2+ cancer when used in conjunction with a HER2 inhibitor.
    Formel:C28H36FN3O
    Reinheit:97.55%
    Farbe und Form:Solid
    Molekulargewicht:449.6
  • G4/HDAC-IN-1


    <p>G4/HDAC-IN-1, a G4/HDAC dual inhibitor, IC50 1.1 µM, blocks TNBC growth, useful in cancer research.</p>
    Formel:C36H49ClFN7O4
    Farbe und Form:Solid
    Molekulargewicht:698.27
  • JBSNF-000028


    <p>JBSNF-000028: potent oral NNMT inhibitor; IC50s—human 0.033 μM, monkey 0.19 μM, mouse 0.21 μM; aids insulin sensitivity &amp; weight loss.</p>
    Formel:C11H13N3
    Reinheit:99.23%
    Farbe und Form:Solid
    Molekulargewicht:187.24
  • hDHODH-IN-11

    CAS:
    hDHODH-IN-11: potent hDHODH inhibitor, IC50 7.2 nM, low cytotoxicity, for AML research.
    Formel:C24H23N3O3
    Farbe und Form:Solid
    Molekulargewicht:401.46
  • Miridesap

    CAS:
    <p>Miridesap (GSK2315698) rapidly depletes SAP in blood, cerebrospinal fluid, and amyloid deposits via liver clearance.</p>
    Formel:C16H24N2O6
    Reinheit:≥95%
    Farbe und Form:Solid
    Molekulargewicht:340.37
  • 15-PGDH-IN-1

    CAS:
    15-PGDH-IN-1: potent oral 15-PGDH inhibitor, IC50=3nM, useful for tissue repair research.
    Formel:C24H22N4O2
    Farbe und Form:Solid
    Molekulargewicht:398.46
  • CDK4/6-IN-14

    CAS:
    CDK4/6-IN-14: potent CDK4/6 inhibitor, IC50s 10/16 nM, >60-fold selectivity over CDKs 1/2/7/9, selective across 205 kinases.
    Formel:C24H27ClFN7O
    Farbe und Form:Solid
    Molekulargewicht:483.97
  • Dynamin IN-1

    CAS:
    Dynamin IN-1 is a potent dynamin inhibitor with an IC 50 value of 1.0 µM .
    Formel:C23H24N2O
    Farbe und Form:Solid
    Molekulargewicht:344.45
  • Zidesamtinib

    CAS:
    <p>Zidesamtinib (NVL-520) is a ROS1 fusion and resistance mutation inhibitor that inhibits ROS1 and can be used to study non-small cell lung cancer.</p>
    Formel:C22H22FN7O
    Reinheit:99.74%
    Farbe und Form:Solid
    Molekulargewicht:419.455
  • Fazamorexant

    CAS:
    Fazamorexant (YZJ-1139) is a powerful orexin receptor antagonist effective for insomnia research.
    Formel:C25H25FN4O2
    Farbe und Form:Solid
    Molekulargewicht:432.49
  • Gumelutamide

    CAS:
    Gumelutamide, a tetrahydropyridopyrimidine compound, functions as both an antiandrogen and an antineoplastic agent by acting as an androgen antagonist.
    Formel:C22H21ClN6O
    Farbe und Form:Solid
    Molekulargewicht:420.89
  • Darizmetinib

    CAS:
    Darizmetinib (HRX215) is an MKK4 inhibitor.
    Formel:C21H17F2N5O3S
    Reinheit:98.03% - 99.57%
    Farbe und Form:Solid
    Molekulargewicht:457.45
  • DRAK1/2-IN-1

    CAS:
    DRAK1/2-IN-1 is a potent inhibitor targeting both DRAK1 and DRAK2, displaying dissociation constants (Kd) of 1 µM and 6 µM, respectively.
    Formel:C22H24N2O3S
    Farbe und Form:Solid
    Molekulargewicht:396.5
  • BCR-ABL-IN-7

    CAS:
    BCR-ABL-IN-7 is an inhibitor of ABL kinase activity in WT and T315I mutants.BCR-ABL-IN-7 can be used in chronic myeloid leukemia (CML) research.
    Formel:C19H16FN3O3S
    Reinheit:98.28%
    Farbe und Form:Solid
    Molekulargewicht:385.41
  • NUCC-0000323

    CAS:
    NUCC-0000323: potent SOD1 inhibitor, curbs expression, used in ALS research.
    Formel:C15H13BrN4S
    Farbe und Form:Solid
    Molekulargewicht:361.26
  • THZ2

    CAS:
    THZ2 (CDK7-IN-1), an analog of THZ1, is a potent and selective CDK7 inhibitor(IC50:13.9 nM),with the potential to treat Triple-negative breast cancer (TNBC).
    Formel:C31H28ClN7O2
    Reinheit:98.28%
    Farbe und Form:Solid
    Molekulargewicht:566.05
  • Falcarindiol

    CAS:
    Falcarindiol is an orally active natural polyacetylene compound, anti-inflammatory and antiproliferative. inhibits NO production, suppressing iNOS expression.
    Formel:C17H24O2
    Reinheit:99.38%
    Farbe und Form:Solid
    Molekulargewicht:260.37
  • Sycosterol A


    <p>Sycosterol A is an α-synuclein (α-syn) inhibitory sterol .</p>
    Formel:C27H48O9S
    Farbe und Form:Solid
    Molekulargewicht:548.73
  • Anserinone B

    CAS:
    Anserinone B: Antifungal, antibacterial; inhibits S.fimicola (50%), A. furfuraceus (37%); cytotoxic to human tumor cells (GI50=4.4 µg/mL).
    Formel:C11H14O4
    Farbe und Form:Solid
    Molekulargewicht:210.23
  • Dictyostatin

    CAS:
    Dictyostatin: potent microtubule stabilizer & anticancer agent with antiproliferative effects; researched for tauopathies.
    Formel:C32H52O6
    Farbe und Form:Solid
    Molekulargewicht:532.75
  • Inuviscolide

    CAS:
    Inuviscolide induces apoptosis, G2/M arrest in melanoma, and has anti-cancer, anti-inflammatory effects.
    Formel:C15H20O3
    Farbe und Form:Solid
    Molekulargewicht:248.32
  • ZINC00640089

    CAS:
    <p>ZINC00640089: Selective LCN2 inhibitor; curbs SUM149 cell growth and AKT activity; useful for IBC research.</p>
    Formel:C20H13F3N2O2
    Reinheit:98.41% - 99.80%
    Farbe und Form:Solid
    Molekulargewicht:370.32
  • Actinoquinol

    CAS:
    Actinoquinol, a compound effective in absorbing UVB radiation, plays a crucial role in protecting the human eye from photooxidative and other oxidative
    Formel:C11H11NO4S
    Farbe und Form:Solid
    Molekulargewicht:253.27
  • KG-501

    CAS:
    KG-501 (Naphthol AS-E phosphate) is a cAMP response element-binding protein (CREB) inhibitor(IC50 : 6.89 μM).
    Formel:C17H13ClNO5P
    Reinheit:97.81%
    Farbe und Form:Solid
    Molekulargewicht:377.72
  • Rosolic Acid

    CAS:
    Rosolic Acid activates Nrf2, boosts angiogenesis, reduces inflammation, deters apoptosis, aids pancreatic cells, and shields ECs from stress.
    Formel:C19H14O3
    Farbe und Form:Solid
    Molekulargewicht:290.31
  • (S)-JDQ-443

    CAS:
    <p>(S)-JDQ-443, an isomer of JDQ-443, is a selective, potent oral KRAS G12C inhibitor with antitumor properties.</p>
    Formel:C29H28ClN7O
    Farbe und Form:Solid
    Molekulargewicht:526.03
  • Octotiamine

    CAS:
    Octotiamine (TATD), a Vitamin B1 analogue and component of the vitamin complex, is utilized in research related to Vitamin B1 deficiency.
    Formel:C23H36N4O5S3
    Farbe und Form:Solid
    Molekulargewicht:544.75
  • Aflibercept

    CAS:
    <p>Aflibercept has a wide range of applications in life science related research.</p>
    Farbe und Form:Liquid
  • TGFβRI-IN-6

    CAS:
    <p>TGFβRI-IN-6 is a potent TGFβRI inhibitor with an IC50 value of 0.55 nM.TGFβRI-IN-6 has the potential to enhance anti-tumour immunity.</p>
    Formel:C17H10F4N6
    Farbe und Form:Solid
    Molekulargewicht:374.3
  • Cyprodenate

    CAS:
    Cyprodenate (Actebral) is a potent orally active brain-activating agent with appetite-suppressing properties, useful in studying metabolic.
    Formel:C13H25NO2
    Farbe und Form:Solid
    Molekulargewicht:227.34
  • c-Met-IN-16

    CAS:
    c-Met-IN-16 is a c-Met inhibitor that can be used for cancer research .
    Formel:C21H17F2N9O
    Farbe und Form:Solid
    Molekulargewicht:449.42
  • LEM-14-1189

    CAS:
    <p>LEM-14-1189 inhibits NSD1/2/3 (IC50: 418/111/60 μM), targets nuclear receptors, and may treat cancer and blood diseases.</p>
    Formel:C35H34N6O5S2
    Reinheit:98.06%
    Farbe und Form:Solid
    Molekulargewicht:682.81
  • FT011

    CAS:
    <p>FT011, a direct anti-fibrotic agent,attenuates cardiac remodelling and dysfunction in experimental diabetic cardiomyopathy.</p>
    Formel:C20H17NO5
    Reinheit:98.98%
    Farbe und Form:Solid
    Molekulargewicht:351.35
  • DPNB-ABT594


    DPNB-ABT594, a nitrobenzyl-caged ABT594, selectively activates α4β2 over α7 nAChRs; used to study Ca²⁺ signaling in MHb.
    Formel:C31H46ClN3O11
    Farbe und Form:Solid
    Molekulargewicht:672.16
  • eeAChE-IN-2

    CAS:
    eeAChE-IN-2 is a potent inhibitor of eeAChE, exhibiting inhibitory potency with an IC50 of 2 nM.
    Formel:C37H40N8O5S
    Farbe und Form:Solid
    Molekulargewicht:708.83
  • (Rac)-SHIN2

    CAS:
    (Rac)-SHIN2 is a serine hydroxymethyltransferase (SHMT) inhibitor for the study of T-cell acute lymphoblastic leukemia (T-ALL).
    Formel:C23H26N4O3
    Reinheit:98.165% - 99.48%
    Farbe und Form:Solid
    Molekulargewicht:406.48
  • Masofaniten

    CAS:
    Masofaniten (EPI-7386) is an orally active androgen receptor (AR) inhibitor with antitumor activity for the study of prostate and breast cancer.
    Formel:C24H24Cl2N4O4S
    Reinheit:98.42% - 98.66%
    Farbe und Form:Solid
    Molekulargewicht:535.44
  • IMD-ferulic


    <p>IMD-ferulic, a compound that forms covalent bonds, acts as an NF-κB modulator, enhancing the adjuvanticity of small molecule immune potentiators.</p>
    Formel:C36H41N7O4
    Farbe und Form:Solid
    Molekulargewicht:635.76
  • photoCORM-1


    photoCORM-1: a CORM with real-time CO monitoring via color change, exhibits cellular uptake and anti-tumor activity.
    Formel:C33H32Cl2N2O6
    Farbe und Form:Solid
    Molekulargewicht:623.52
  • photoCORM-2

    CAS:
    photoCORM-2 releases CO, changes color for real-time monitoring, has good cellular uptake, and anti-tumor properties.
    Formel:C17H13NO3
    Farbe und Form:Solid
    Molekulargewicht:279.29
  • hGGPPS-IN-3

    CAS:
    13h (hGGPPS-IN-3), a strong C2-ThP-BPs hGGPPS blocker, triggers MM cell apoptosis and shows in vivo anti-myeloma effects.
    Formel:C21H19BrN4O7P2S
    Reinheit:98%
    Farbe und Form:Solid
    Molekulargewicht:613.31
  • β-Estradiol 17-acetate

    CAS:
    <p>β-Estradiol 17-acetate (1,3,5(10)-Estratriene-3,17β-diol 17-acetate) is a metabolite of estradiol.</p>
    Formel:C20H26O3
    Reinheit:98.11% - 99.88%
    Farbe und Form:Solid
    Molekulargewicht:314.42
  • BAY 1214784

    CAS:
    <p>BAY 1214784: potent, oral hGnRH-R antagonist, reduces LH levels, low variability, good tolerance, may research uterine fibroids.</p>
    Formel:C29H26ClF4N3O5S2
    Farbe und Form:Solid
    Molekulargewicht:672.11
  • Bis-Pro-5FU

    CAS:
    Bis-Pro-5FU enhances oral uptake and safety of 5-FU, an anti-cancer drug for colorectal and pancreatic tumors.
    Formel:C10H7FN2O2
    Farbe und Form:Solid
    Molekulargewicht:206.17
  • Hsp90-IN-17

    CAS:
    Hsp90-IN-17 (Example 5) is an inhibitor of HSP90, applicable in researching proliferative diseases, including cancer and neurodegenerative conditions.
    Formel:C21H20N4O7
    Farbe und Form:Solid
    Molekulargewicht:440.41
  • HIF-2α-IN-7

    CAS:
    HIF-2α-IN-7 is a hypoxia inducible factor 2α (HIF-2α) inhibitor.
    Formel:C18H9F6NO2
    Farbe und Form:Solid
    Molekulargewicht:385.26
  • L-Afegostat

    CAS:
    <p>L-Afegostat (5-epi-Isofagomine), an iminosugar, inhibits glycosidase and β-Glucosidase (K i 30 μM), aids in carbohydrate synthesis.</p>
    Formel:C6H13NO3
    Farbe und Form:Solid
    Molekulargewicht:147.17
  • PF-06455943

    CAS:
    PF-06455943: LRRK2 inhibitor, IC50=3nM, PET radioligand, used for ADME/neuro PK & Parkinson's research.
    Formel:C17H14FN5O
    Farbe und Form:Solid
    Molekulargewicht:323.32
  • GDC-0575

    CAS:
    <p>GDC-0575 (ARRY-575) is a highly-selective oral small-molecule Chk1 inhibitor(IC50 of 1.2 nM).</p>
    Formel:C16H20BrN5O
    Reinheit:≥95%
    Farbe und Form:Solid
    Molekulargewicht:378.27
  • SIRT2-IN-11

    CAS:
    SIRT2-IN-11 (AEM1), a SIRT2 inhibitor (IC50 18.5μM), induces apoptosis and affects p53, used in cancer research.
    Formel:C21H22N2O
    Farbe und Form:Solid
    Molekulargewicht:318.41
  • eIF4A3-IN-9

    CAS:
    eIF4A3-IN-9, a silvestrol analogue, disrupts eIF4F complex assembly; EC50s: 29/450/80 nM (myc/tub-LUC, MB-231 cells); for cancer research.
    Formel:C28H27NO8
    Farbe und Form:Solid
    Molekulargewicht:505.52
  • METTL3-IN-1

    CAS:
    <p>METTL3-IN-1 is a polyheterocyclic compound, acts as METTL3 inhibitor .</p>
    Formel:C25H24FN5O2
    Farbe und Form:Solid
    Molekulargewicht:445.49
  • METTL3-IN-2

    CAS:
    METTL3-IN-2, a potent METTL3 inhibitor, exhibits an IC50 value of 6.1 nM, effectively impairing the proliferation of Caov3 cancer cells.
    Formel:C25H26N8O
    Farbe und Form:Solid
    Molekulargewicht:454.53
  • METTL3-IN-3

    CAS:
    METTL3-IN-3 is a polyheterocyclic compound, acts as METTL3 inhibitor .
    Formel:C26H28BrFN6O2
    Farbe und Form:Solid
    Molekulargewicht:555.44
  • PF-07054894

    CAS:
    PF-07054894: potent CCR6 antagonist, targets GPCR, for inflammatory bowel disease research.
    Formel:C24H30N6O4
    Farbe und Form:Solid
    Molekulargewicht:466.53
  • cis-ccc_R08

    CAS:
    cis-ccc_R08 infection . cis-ccc_R08 is a cccDNA (covalently closed circular DNA) inhibitor .
    Formel:C22H19ClO6
    Farbe und Form:Solid
    Molekulargewicht:414.84
  • PARP10-IN-2

    CAS:
    <p>PARP10-IN-2 is a potent inhibitor of PARP10, a mono-ADP-ribosyltransferase, with an IC50 value of 3.64 μM for human PARP10.PARP10-IN-2 also inhibited PARP2 and</p>
    Formel:C14H10N2O2
    Reinheit:99.27%
    Farbe und Form:Solid
    Molekulargewicht:238.24
  • PCSK9-IN-13

    CAS:
    PCSK9-IN-13 is a potent inhibitor of PCSK9, effectively preventing the binding of PCSK9 to low-density lipoprotein (LDL) receptors through its mechanism of
    Formel:C30H33N5O2
    Farbe und Form:Solid
    Molekulargewicht:495.62
  • Vemtoberant

    CAS:
    Vemtoberant is a β3 adrenergic antagonist used in β3-related disorder research like heart failure.
    Formel:C29H37N3O8S2
    Farbe und Form:Solid
    Molekulargewicht:619.75
  • BDP5290

    CAS:
    BDP5290 is a potent inhibitor of both ROCK and MRCK(IC50s of 5 nM, 50 nM, 10 nM and 100 nM for ROCK1, ROCK2, MRCKα and MRCKβ, respectively.)
    Formel:C17H18ClN7O
    Reinheit:97.22%
    Farbe und Form:Solid
    Molekulargewicht:371.82
  • HSP90-IN-20

    CAS:
    HSP90-IN-20, a potent inhibitor of HSP90, exhibits an IC50 of ≤10 μM, indicating its potential application in cancer research.
    Formel:C26H32N4O4
    Farbe und Form:Solid
    Molekulargewicht:464.56
  • NLRP3-IN-14

    CAS:
    NLRP3-IN-14, potent selective NLRP3 inhibitor, KD 5.87μM; IC50 0.131μM for IL-1β; for inflammation research.
    Formel:C27H28N2O4
    Farbe und Form:Solid
    Molekulargewicht:444.52
  • NLRP3-IN-15

    CAS:
    NLRP3-IN-15: potent, selective NLRP3 inflammasome inhibitor; IC50 0.114 μM for IL-1β; for inflammation research.
    Formel:C22H19NO4
    Farbe und Form:Solid
    Molekulargewicht:361.39
  • NLRP3-IN-16

    CAS:
    NLRP3-IN-16: potent NLRP3 inflammasome inhibitor; IC50=0.065μM; curbs IL-1β; used in inflammation studies.
    Formel:C25H25NO5
    Reinheit:98%
    Farbe und Form:Solid
    Molekulargewicht:419.47
  • THRX-144644

    CAS:
    THRX-144644: lung-specific ALK5 inhibitor, 0.14 nM IC50, no systemic TGFβ toxicity.
    Formel:C26H28ClF2N7
    Farbe und Form:Solid
    Molekulargewicht:512
  • ONO-0740556

    CAS:
    ONO-0740556 is a potent agonist of the Gi-coupled human lysophosphatidic acid receptor 1 (LPA1), exhibiting an EC50 value of 0.26 nM.
    Formel:C20H34NO6P
    Farbe und Form:Solid
    Molekulargewicht:415.46
  • NLRP3-IN-13

    CAS:
    <p>NLRP3-IN-13 is an NLRP3 inhibitor that inhibits NLRP3-associated inflammation.NLRP3-IN-13 can be used in the study of neurological disorders and inflammation.</p>
    Formel:C19H15N3O3S
    Reinheit:99.16%
    Farbe und Form:Solid
    Molekulargewicht:365.41
  • MALT1-IN-11

    CAS:
    <p>MALT1-IN-11: MALT1 inhibitor, IC50 &lt;10-100 nM, reduces IL10, for cancer/autoimmune research.</p>
    Formel:C20H16F4N8O
    Farbe und Form:Solid
    Molekulargewicht:460.39
  • CU-CPT9b

    CAS:
    <p>CU-CPT9b (TLR8-specific antagonist 1) is an antagonist of toll-like receptor 8 (TLR8; Kd = 21 nM).</p>
    Formel:C16H13NO2
    Reinheit:98.1%
    Farbe und Form:Solid
    Molekulargewicht:251.28
  • c-Met-IN-14

    CAS:
    c-Met-IN-14: selective c-Met kinase inhibitor, IC50 2.89 nM, anticancer, stops G2/M phase, induces A549 cell apoptosis.
    Formel:C34H38ClFN4O7S
    Farbe und Form:Solid
    Molekulargewicht:701.2
  • PARP1-IN-12


    PARP1-IN-12: potent PARP1 inhibitor, IC50 2.99 nM, triggers cell apoptosis, G2/M arrest, induces DSBs in BRCA-deficient cells.
    Formel:C43H56FN5O5
    Farbe und Form:Solid
    Molekulargewicht:741.93
  • PARP7-IN-12

    CAS:
    PARP7-IN-12, a potent inhibitor targeting PARP7, exhibits an IC50 of 7.836 nM. This compound is applicable in cancer research.
    Formel:C23H27ClF3N5O5
    Farbe und Form:Solid
    Molekulargewicht:545.94
  • PARP-2-IN-3

    CAS:
    <p>PARP-2-IN-3 is used in the study of breast cancer as a PARP-2 inhibitor with antitumor activity that induces apoptosis (apoptosis) and necrosis in cancer cells.</p>
    Formel:C20H20ClN3O3
    Reinheit:99.33%
    Farbe und Form:Solid
    Molekulargewicht:385.84
  • hCAIX-IN-16

    CAS:
    hCAIX-IN-16 (Compound 12d), an inhibitor of hCA IX, exhibits inhibition constants (K i) of 190.0 nM for hCA IX and 187.9 nM for hCA XII.
    Formel:C20H20N8O2S
    Reinheit:98%
    Farbe und Form:Solid
    Molekulargewicht:436.49
  • hCAIX-IN-15

    CAS:
    hCAIX-IN-15 is a potent inhibitor of human carbonic anhydrase IX (hCA IX) with an inhibition constant (Ki) of 38.8 nM, exhibiting broad-spectrum anticancer
    Formel:C18H14FN7O2S
    Reinheit:98%
    Farbe und Form:Solid
    Molekulargewicht:411.41
  • LIXIVAPTAN

    CAS:
    Lixivaptan (VPA-985) is an orally active and selective vasopressin receptor V2 antagonist(Ki = 2.3 nM)
    Formel:C27H21ClFN3O2
    Reinheit:98.36%
    Farbe und Form:Solid
    Molekulargewicht:473.93
  • hCAIX-IN-14

    CAS:
    hCAIX-IN-14 is a potent inhibitor of human CA IX with a K i value of 134.8 nM .
    Formel:C11H17ClN6O2S
    Farbe und Form:Solid
    Molekulargewicht:332.81