CAS 106266-06-2

Risperidona

Descripción:

Risperidona es un medicamento antipsicótico atípico que se utiliza principalmente para tratar la esquizofrenia, el trastorno bipolar y la irritabilidad asociada con el autismo. Funciona como un antagonista de la serotonina y la dopamina, influyendo en la actividad de los neurotransmisores en el cerebro, particularmente en los receptores de serotonina y dopamina. Risperidona se caracteriza por su fórmula química C23H27N3O2 y un peso molecular de aproximadamente 410.48 g/mol. La sustancia aparece como un polvo cristalino blanco a blanco amarillento y se administra típicamente en forma oral, aunque también están disponibles formulaciones inyectables. Su farmacocinética indica una vida media relativamente larga, lo que permite una dosificación una vez al día en muchos casos. Los efectos secundarios comunes pueden incluir sedación, aumento de peso y cambios metabólicos, lo que requiere un monitoreo durante el tratamiento. El perfil de eficacia y seguridad de Risperidona lo convierte en una opción ampliamente prescrita en el cuidado psiquiátrico, aunque es esencial adaptar el tratamiento a las necesidades individuales del paciente y monitorear posibles efectos adversos.

Fórmula: C₂₃H₂₇FN₄O₂

InChI: InChI=1/C23H27FN4O2/c1-15-18(23(29)28-10-3-2-4-21(28)25-15)9-13-27-11-7-16(8-12-27)22-19-6-5-17(24)14-20(19)30-26-22/h5-6,14,16H,2-4,7-13H2,1H3

Clave InChI: InChIKey=RAPZEAPATHNIPO-UHFFFAOYSA-N

SMILES: FC=1C=C2C(C(=NO2)C3CCN(CCC=4C(=O)N5C(=NC4C)CCCC5)CC3)=CC1

Sinónimos:

• 1,2-Benzisoxazole, 4H-pyrido[1,2-a]pyrimidin-4-one deriv.
• 3-(2-(4-(6-Fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl)ethyl)-6,7,8,9-tetrahydro-2-methyl-4H-pyrido[1,2-α]pyrimidin-4-one
• 3-[2-[4-(6-Fluor-1,2-benzisoxazol-3-yl)piperidino]ethyl]-2-methyl-6,7,8,9-tetrahydro-4H-pyrido[1,2-a]pyrimidin-4-on
• 3-{2-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]ethyl}-2-methyl-6,7,8,9-tetrahydro-4H-pyrido[1,2-a]pyrimidin-4-one
• 4H-Pyrido[1,2-a]pyrimidin-4-one, 3-[2-[4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-2-methyl-
• Apexidone
• Psychodal
• R 64766
• Rbp 7000
• Resperidone
• Ripedon
• Risbiodal
• Rispa
• Rispadal
• Risperdal
• Risperdal Consta
• Risperdine
• Risperid
• Risperid fort
• Risperidal
• Risperidone ACIS
• Risperidone intermediates
• Spiron
• Zophrenal
• Risperidone
• 4H-Pyrido[1,2-a]pyrimidin-4-one, 3-[2-[4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-2-methyl-(9CI)
• 3-[2-4-(6-Fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl-6,7,8,9-tetrahydro-2-methyl-4H-pyrido[1,2-α]pyrimidin-4-one, R-64766, Belivon, Risperdal
• Risoeridone
• 3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-
• Kesperidone
• 3-[2-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]ethyl]-2-methyl-6,7,8,9-tetrahydropyrido[2,1-b]pyrimidin-4-one
• 3-[2-4-(6-Fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl-6,7,8,9-tetrahydro-2-methyl-4H-pyrido[1,2-a]pyrimidin-4-one, R-64766, Belivon, Risperdal
• 4h-pyrido(1,2-a)pyrimidin-4-one,6,7,8,9-tetrahydro-3-(2-(4-(6-fluoro-1,2-benzi
• 3-[2-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-
• soxazol-3-yl)-1-piperidinyl)ethyl)-2-methyl-
• 3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin-1-yl]-ethyl}-2-methyl-6,7,8,9-tetrahydro-pyrido[1,2,a]pyrimidin-4-one

Risperidone

CAS: 106266-06-2

Applications Risperidone is a combined serotonin (5-HT2) and dopamine (D2) receptor antagonist.
Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package
References Jannssen, P.A.J., et al.: J. Pharmacol. Exp. Ther., 244, 685 (1988); Gelders, Y.G., et al.: Pharmacopsychiatry, 23, 206 (1990); Green, B.: Curr. Med. Res. Opin., 16, 57 (2000);

Fórmula: C₂₃H₂₇FN₄O₂

Forma y color: Neat

Peso molecular: 410.48

Ref: TR-R525000

Risperidone

Producto controlado

CAS: 106266-06-2

Risperidone can be used as an antipsychotic drug in the treatment of schizophrenia and mania. This is due to it binding to the 5-HT2 receptor and antagonizing serotonin, leading to a reduction in symptoms such as delusions and hallucinations. This product can also act on the D1 and D2 Dopamine receptors. It is thought, that as a result of Risperidone’s antagonistic activity against D2 receptors within the tuberoinfundibular pathway, an increase in the level of prolactin occurs. Consequently leading to hyperprolactinemia, a negative adverse effect when Risperidone is used as a drug. Risperidone has been shown to have cardiac effects, including increasing heart rate and QT interval. It is also metabolized by cytochrome P450 enzymes and can be detected in wastewater after oral administration of a single dose (0.5 mg/kg).

Fórmula: C₂₃H₂₇FN₄O₂

Pureza: Min. 98.5 Area-%

Forma y color: White Off-White Powder

Peso molecular: 410.48 g/mol

Ref: 3D-FR27737

Risperidone - Bio-X ™

Producto controlado

CAS: 106266-06-2

Risperidone can be used as an antipsychotic drug in the treatment of schizophrenia and mania. This is due to it binding to the 5-HT2 receptor and antagonizing serotonin, leading to a reduction in symptoms such as delusions and hallucinations. This product can also act on the D1 and D2 Dopamine receptors. It is thought, that as a result of Risperidone’s antagonistic activity against D2 receptors within the tuberoinfundibular pathway, an increase in the level of prolactin occurs. Risperidone is part of our Bio-X ™ Range. These products are aimed at life science researchers who need high quality ready-to-use products for assay development, screening or other R&D work. With a solubility datasheet and convenient vials, all of our Bio-X ™ products are in stock across our global warehouses for rapid delivery and ease of use.

Fórmula: C₂₃H₂₇FN₄O₂

Pureza: Min. 99.0 Area-%

Forma y color: White Powder

Peso molecular: 410.48 g/mol

Ref: 3D-BR164349

Risperidone

CAS: 106266-06-2

Ref: BE-MU-7140

Risperidone

CAS: 106266-06-2

Ref: BE-RMCR091000

Risperidone in Methanol

CAS: 106266-06-2

Methanol

Ref: BE-MU-7140LM-10

Risperidone in Methanol

CAS: 106266-06-2

Methanol

Ref: BE-MU-7140YM-1000

Risperidone

CAS: 106266-06-2

Fórmula: C₂₃H₂₇FN₄O₂

Pureza: 98%

Forma y color: Solid, White to off-white powder

Peso molecular: 410.212

Ref: 10-F036563