CAS 107788-00-1

Tyrphostin ag 658

CAS: 107788-00-1

Tyrphostin ag 658 is a protein kinase inhibitor that inhibits the activity of the ubiquitin-proteasome system. Tyrphostin ag 658 has been shown to inhibit the activity of ubiquitin ligases and targets, which are enzymes involved in protein degradation. The drug binds to a specific moiety on the enzyme and prevents it from functioning. Tyrphostin ag 658 has been used as a linker for photolabile drugs, including puromycin and doxorubicin, to target proteins that are not accessible with traditional inhibitors. As with other tyrosine kinase inhibitors, tyrphostin ag 658 inhibits protein synthesis by preventing the phosphorylation of proteins at tyrosine residues. This inhibition prevents cellular proliferation and division by blocking cell cycle progression.

Fórmula: C₁₈H₁₆N₂O₃S

Pureza: Min. 95%

Peso molecular: 340.4 g/mol

Ref: 3D-HEA78800