CAS 1467052-75-0

Tazemetostat hydrobromide

CAS: 1467052-75-0

Fórmula: C₃₄H₄₅BrN₄O₄

Pureza: 98%

Peso molecular: 653.6495

Ref: IN-DA01V3MX

Tazemetostat hydrobromide

CAS: 1467052-75-0

Tazemetostat hydrobromide

Pureza: ≥98%

Peso molecular: 653.65g/mol

Ref: 54-BUP15347

Tazemetostat hydrobromide

CAS: 1467052-75-0

Tazemetostat hydrobromide: potent, selective EZH2 inhibitor; blocks PRC2/wild-type EZH2 (Ki: 2.5 nM) & EZH1 (IC50: 392 nM).

Fórmula: C₃₄H₄₅BrN₄O₄

Pureza: 99.8%

Forma y color: Solid

Peso molecular: 653.65

Ref: TM-T17002

Tazemetostat hydrobromide

CAS: 1467052-75-0

Tazemetostat hydrobromide is a potent and selective inhibitor of histone methyltransferase. This drug binds to the active site of the enzyme, preventing it from transferring methyl groups. Tazemetostat hydrobromide prevents the activation of cancer-related genes, which has been demonstrated in vitro using various cancer cell lines. Furthermore, this drug acts as an inhibitor of viral replication by inhibiting the production of new viruses. The polymorphic form of tazemetostat hydrobromide is found in human plasma and urine samples and may be used as a biomarker for cancer susceptibility. Tazemetostat hydrobromide may also be used as an antineoplastic agent against certain types of cancers due to its inhibition of histone methylation.

Fórmula: C₃₄H₄₅BrN₄O₄

Pureza: Min. 95%

Peso molecular: 653.6 g/mol

Ref: 3D-SIC05275