CAS 1671088-84-8

CAY10727

CAS: 1671088-84-8

CAY10727 selectively inhibits PAD3 (15,600 M^-1min^-1) over PAD1, PAD2, and PAD4.

Fórmula: C₂₁H₂₂Cl₂N₄O₂

Forma y color: Solid

Peso molecular: 433.33

Ref: TM-T36393

CAY10727

CAS: 1671088-84-8

CAY10727 is a potent biochemical inhibitor, which is derived from synthetic sources with specific action targeting cyclooxygenase-2 (COX-2) enzymes. It functions by selectively blocking the enzymatic activity of COX-2, which plays a critical role in the biosynthesis of prostaglandins involved in inflammatory responses. This targeted inhibition allows the study of COX-2-related pathways without interference from COX-1, which is significant for maintaining gastrointestinal integrity.The use and applications of CAY10727 are primarily in research settings where understanding the pathways involved in inflammation, pain, and cancer progression are critical. This compound is utilized in various in vitro experiments to delineate the role of COX-2 in cellular and molecular contexts, enabling scientists to dissect complex signaling networks. Given its specificity, CAY10727 is instrumental in the development of new therapeutic approaches where selective COX-2 inhibition might offer benefits over non-selective inhibitors.

Fórmula: C₂₁H₂₂Cl₂N₄O₂

Pureza: Min. 95%

Peso molecular: 433.3 g/mol

Ref: 3D-WRC08884