CAS 1904611-63-7

PDE1-IN-2

CAS: 1904611-63-7

Fórmula: C₁₆H₂₁BrN₄O₂

Pureza: 98%

Peso molecular: 381.2675

Ref: IN-DA01EOF4

PDE1-IN-2

CAS: 1904611-63-7

PDE1-IN-2 is a potent and selective activator of phosphodiesterase type 1 (PDE1). The PDE1-IN-2 ligand binds to the receptor on the cell surface, activating it and resulting in an increase in intracellular cAMP. This intracellular messenger molecule is involved in many cellular processes, including protein synthesis, ion channels, and cell signaling. PDE1-IN-2 has been shown to be a potent inhibitor of the antibody response, as well as having potential use as a therapeutic agent for chronic immune disorders.
Protein interactions:
PDE1-IN-2 binds to protein kinase A (PKA) and the cAMP response element binding protein (CREB), which are both involved in cellular processes such as gene transcription.

Fórmula: C₁₆H₂₁BrN₄O₂

Pureza: Min. 95%

Peso molecular: 381.27 g/mol

Ref: 3D-EBD61163

PDE1-IN-2

CAS: 1904611-63-7

PDE1-IN-2 is an PDE1 inhibitor(PDE1C, PDE1B and PDE1A with IC50 values of 6, 140 and 164 nM, respectvely).

Fórmula: C₁₆H₂₁BrN₄O₂

Pureza: 98%

Forma y color: Solid

Peso molecular: 381.27

Ref: TM-T12390