CAS 1936422-33-1

GNE-781

CAS: 1936422-33-1

GNE-781: potent CBP inhibitor (IC50: 0.94 nM), also targets BRET/BRD4(1) (IC50: 6.2/5100 nM).

Fórmula: C₂₇H₃₃F₂N₇O₂

Pureza: 99.25% - 99.64%

Forma y color: Solid

Peso molecular: 525.59

Ref: TM-T15405

GNE-781

CAS: 1936422-33-1

GNE-781

Pureza: ≥98%

Peso molecular: 525.59g/mol

Ref: 54-BUP04443

GNE-781

Producto controlado

CAS: 1936422-33-1

Fórmula: C₄H₁₁NO·HCl

Forma y color: Neat

Peso molecular: 125.597

Ref: TR-D447825

GNE 781

CAS: 1936422-33-1

A selective inhibitor of the bromodomain of Cyclic adenosine monophosphate Response Element Binding protein Binding Protein (CREBBP or CBP) with anti-tumoral activity. The CBP inhibition regulates oncogene MYC and impairs differentiation of regulatory T cells.

Fórmula: C₂₇H₃₃F₂N₇O₂

Pureza: Min. 95%

Peso molecular: 525.59 g/mol

Ref: 3D-BG166815