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CAS 1980821-53-1

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  • pan-Raf/RTK inhibitor 1

    CAS:
    Pan-Raf/RTK inhibitor 1 (compound I-16) is a potent pan-Raf inhibitor with IC50 values of 3.49 nM (BRafV600E), 8.86 nM (ARaf), 5.78 nM (BRafWT), and 1.65 nM (CRaf). It exhibits antiproliferative activity against various cancer cell lines and can be utilized in cancer research.
    Fórmula:C29H28F3N7O3
    Forma y color:Solid
    Peso molecular:579.573