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CAS 2173508-07-9

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  • CGRP antagonist 7

    CAS:
    CGRP antagonist 7 is a potent calcitonin gene-related peptide receptor (CGRP) antagonist with a Ki value of 0.029 nM. It effectively inhibits CGRP receptor-mediated cyclic adenosine monophosphate (cAMP) production, with an IC50 value of 1.5 nM. This compound is useful in migraine research.
    Fórmula:C30H32FN5O3
    Forma y color:Solid
    Peso molecular:529.61