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CAS 2196448-47-0

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  • EN1441

    CAS:
    <p>EN1441 is a covalent degrader that targets the androgen receptor (AR) with an EC50 value of 4.2 μM, as well as its truncated variant AR-V7. It selectively and effectively degrades AR and AR-V7 in androgen-independent prostate cancer cells. EN1441 holds potential for research into androgen-independent prostate cancer.</p>
    Fórmula:C13H13ClN2O2
    Forma y color:Solid
    Peso molecular:264.708