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CAS 2355304-05-9

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  • RGH-122

    CAS:
    <p>RGH-122 (compound 43), characterized as an orally active, potent, and selective hV1a receptor antagonist, demonstrates significant affinity with a K i value of 0.3 nM and an IC 50 of 0.9 nM. It exhibits microsomal stability, indicated by a CL int value of 13/28/25 μL/min/mg [1].</p>
    Fórmula:C24H25ClN4O3
    Forma y color:Solid
    Peso molecular:452.93