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CAS 2674064-32-3

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  • BET/Aurora kinase-IN-1

    CAS:
    BET/Aurora kinase-IN-1 (Compound 38) is a dual inhibitor of BET and Aurora kinases. It exhibits antiproliferative activity against various tumor cell lines and demonstrates significant antitumor efficacy in xenograft models of renal cell carcinoma and colon cancer, with tumor growth inhibition (TGI) rates of 45.99% and 53.06%, respectively.
    Fórmula:C25H30FN7O
    Forma y color:Solid
    Peso molecular:463.55