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CAS 3017180-18-3

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  • DDO-8958

    CAS:
    DDO-8958 is an orally active and selective BET BD1 inhibitor, exhibiting a KD of 5.6 nM for BRD4 BD1. It shows low nanomolar inhibitory activity across all BET BD1 bromodomains except for BRDT BD1. DDO-8958 inhibits tumor cell proliferation and migration, induces apoptosis and cell cycle arrest, and demonstrates antitumor activity.
    Fórmula:C22H22FN5O2
    Forma y color:Solid
    Peso molecular:407.441