CAS 512-15-2

Ciclopentolato

Descripción:

Ciclopentolato es una amina terciaria y un derivado del ácido trópico, utilizado principalmente como agente midriático en oftalmología para dilatar las pupilas durante los exámenes oculares. Se caracteriza por su capacidad para bloquear la acción de la acetilcolina en los receptores muscarínicos del músculo esfínter del iris, lo que conduce a la dilatación de la pupila. Ciclopentolato se administra típicamente como una solución en gotas para los ojos y tiene un inicio de acción rápido, con efectos que duran varias horas. El compuesto es conocido por su relativamente baja absorción sistémica, lo que minimiza los efectos secundarios. En términos de propiedades físicas, Ciclopentolato es un polvo cristalino blanco a blanco sucio que es soluble en agua y presenta un perfil de solubilidad dependiente del pH. Su estructura química incluye un anillo de ciclopentano, lo que contribuye a sus propiedades farmacológicas únicas. Al igual que con cualquier medicamento, es esencial considerar los posibles efectos secundarios, incluyendo el aumento de la presión intraocular y la sensibilidad a la luz, particularmente en individuos susceptibles.

Fórmula: C₁₇H₂₅NO₃

InChI: InChI=1S/C17H25NO3/c1-18(2)12-13-21-16(19)15(14-8-4-3-5-9-14)17(20)10-6-7-11-17/h3-5,8-9,15,20H,6-7,10-13H2,1-2H3

Clave InChI: InChIKey=SKYSRIRYMSLOIN-UHFFFAOYSA-N

SMILES: C(C(OCCN(C)C)=O)(C1(O)CCCC1)C2=CC=CC=C2

Sinónimos:

• 1-Hydroxy-α-phenylcyclopentaneacetic acid, 2-(dimethylamino)ethyl ester
• 2-(Dimethylamino)Ethyl (1-Hydroxycyclopentyl)(Phenyl)Acetate
• 2-(Dimethylamino)ethyl 2-(1-hydroxycyclopentyl)-2-phenylacetate
• 2-Dimethylaminoethyl 1-hydroxy-α-phenylcyclopentaneacetate
• 2-Dimethylaminoethyl 2-(1-Hydroxycyclopentyl)-2-Phenylacetate
• <span class="text-smallcaps">DL</span>-Cyclopentolate
• Benzeneacetic acid, α-(1-hydroxycyclopentyl)-, 2-(dimethylamino)ethyl ester
• Ciclopentolato
• Cyclogyl
• Cyclopentaneacetic acid, 1-hydroxy-α-phenyl-, 2-(dimethylamino)ethyl ester
• Cyclopentoiate
• Cyclopentolat
• Cyclopentylate
• DL-Cyclopentolate
• Tsiklopentolat
• β-Dimethylaminoethyl (1-hydroxycyclopentyl)phenylacetate
• Mydrilate
• 2-Dimethylaminoethyl 1-hydroxy-alpha-phenylcyclopentaneacetate
• 2-dimethylaminoethyl 2-(1-hydroxycyclopentyl)-2-phenyl-ethanoate
• CYCLOPENTOLATE
• Benzeneacetic acid, a-(1-hydroxycyclopentyl)-, 2-(dimethylamino)ethylester
• 1-Hydroxy-alpha-phenylcyclopentaneacetic acid, 2-(dimethylamino)ethyl ester
• 2-(1-hydroxycyclopentyl)-2-phenyl-acetic acid 2-dimethylaminoethyl ester
• yclopentolate
• Benzeneacetic acid, alpha-(1-hydroxycyclopentyl)-, 2-(dimethylamino)ethyl ester
• α-(1-Hydroxycyclopentyl)benzeneacetic acid 2-(dimethylamino)ethyl
• beta-(Dimethylamino)ethyl (1-hydroxycyclopentyl)phenylacetate
• Cyplegin

2-(Dimethylamino)ethyl 2-(1-hydroxycyclopentyl)-2-phenylacetate

CAS: 512-15-2

Fórmula: C₁₇H₂₅NO₃

Peso molecular: 291.3853

Ref: IN-DA00I95X

Cyclopentolate

Producto controlado

CAS: 512-15-2

Cyclopentolate is a muscarinic antagonist and is used as an ophthalmic drug to produce mydriasis. Cyclopentolate inhibits the metabolism of cyclopentyl-CoA via the 3-hydroxyacyl-CoA dehydrogenase, which leads to the accumulation of cyclopentyl-CoA in cells. This inhibition can cause metabolic disorders such as hyperlipidemia and diabetes mellitus, which are characterized by increased acid formation and reduced glucose uptake. Cyclopentolate also binds to DNA, inhibiting transcription, replication, and repair of DNA. The binding affinity of cyclopentolate to DNA is approximately 2500 times higher than that of other drugs in its class. Cyclopentolate has been shown to inhibit leukemia inhibitory factor (LIF) and the production of acid from fluorescein angiography

Fórmula: C₁₇H₂₅NO₃

Pureza: Min. 95%

Forma y color: White/Off-White Solid

Peso molecular: 291.39 g/mol

Ref: 3D-FC61687

2-(Dimethylamino)ethyl 2-(1-hydroxycyclopentyl)-2-phenylacetate

CAS: 512-15-2

Fórmula: C₁₇H₂₅NO₃

Pureza: 95.0%

Peso molecular: 291.391

Ref: 10-F449906