CAS 69-22-7

Citrato de cafeína

Descripción:

Citrato de cafeína es un compuesto químico que combina cafeína, un estimulante del sistema nervioso central, con ácido cítrico. Se utiliza principalmente en entornos médicos, particularmente para el tratamiento de la apnea en bebés prematuros, ya que ayuda a estimular la respiración. Citrato de cafeína es un polvo cristalino blanco a blanco amarillento que es soluble en agua, lo que facilita su administración en entornos clínicos. El compuesto exhibe las propiedades estimulantes de la cafeína, promoviendo la alerta y reduciendo la fatiga. Su farmacocinética implica una rápida absorción y metabolismo en el hígado, lo que lleva a un aumento de las concentraciones plasmáticas de cafeína. El componente de citrato mejora la solubilidad y biodisponibilidad de la cafeína, haciéndola más efectiva para el uso terapéutico. Citrato de cafeína generalmente es bien tolerado, pero los efectos secundarios potenciales pueden incluir aumento de la frecuencia cardíaca, trastornos gastrointestinales y nerviosismo, particularmente a dosis más altas. Al igual que con cualquier medicamento, es importante usar Citrato de cafeína bajo supervisión médica para garantizar la seguridad y eficacia.

Fórmula: C₁₄H₁₈N₄O₉

InChI: InChI=1/C8H10N4O2.C6H8O7/c1-10-4-9-6-5(10)7(13)12(3)8(14)11(6)2;7-3(8)1-6(13,5(11)12)2-4(9)10/h4H,1-3H3;13H,1-2H2,(H,7,8)(H,9,10)(H,11,12)

Clave InChI: InChIKey=RCQXSQPPHJPGOF-UHFFFAOYSA-N

SMILES: C(CC(O)=O)(CC(O)=O)(C(O)=O)O.O=C1C2=C(N(C)C(=O)N1C)N=CN2C

Sinónimos:

• 1,2,3-Propanetricarboxylic acid, 2-hydroxy-, mixt. with 3,7-dihydro-1,3,7-trimethyl-1H-purine-2,6-dione
• 1H-Purine-2,6-dione, 3,7-dihydro-1,3,7-trimethyl-, mixt. contg.
• 1H-purine-2,6-dione, 3,7-dihydro-1,3,7-trimethyl-, 2-hydroxy-1,2,3-propanetricarboxylate (1:1) (salt)
• Cafcit
• Caffeina citrate
• Caffeine Citrated
• Caffeine citrate
• Caffeine citrate (1:1)
• Caffeine, citrated [USAN]
• Cafnea
• Citrated caffein
• Citrated caffeine
• Citric acid, compd. with caffeine (1:1)
• Gencebok
• Peyona
• 1,3,7-Trimethyl-3,7-dihydro-1H-purine-2,6-dione 2-hydroxypropane-1,2,3-tricarboxylate (1:1)
• 1,3,7-TRIMETHYL-2,6-DIOXOPURINE CITRATE
• 1,3,7-Trimethyl-3,7-dihydro-purin-2,6-dion2-hydroxypropane-1,2,3-tricarboxylic acid,1,3,7-trimethyl
• thyl-1h-purine-2,6-dione
• 1,3,7-TRIMETHYLXANTHINE CITRATE
• Coffeinum-citrate
• citricacid,compd.withcaffeine(1:1)
• caffeinecitrate(1:1)
• CAFFEINE CITRATED GRANULAR
• caffeinacitrate
• Kaffein,Citrat
• COFFEINE CITRATE
• METHYLTHEOBROMINE CITRATE
• Caffeine Citrate USP
• Mixture with citric acid
• CAFFEINE,CITRATED,POWDER,PURIFIED
• GUARANINE CITRATE
• Caffeine, Citrated, Powder
• 2-HYDROXYPROPANE-1,2,3-TRICARBOXYLIC ACID,1,3,7-TRIMETHYLPURINE-2,6-DIONE
• citratedcaffein

Caffeine Citrate

Producto controlado

CAS: 69-22-7

Fórmula: C₈H₁₀N₄O₂·C₆H₈O₇

Forma y color: Neat

Peso molecular: 386.31

Ref: 86-MM1851.00

Caffeine Citrate

CAS: 69-22-7

Fórmula: C₈H₁₀N₄O₂C₆H₈O₇

Peso molecular: 194.2 : 192.1

Ref: ST-EA-CP-C47008

Caffeine citrate

Producto controlado

CAS: 69-22-7

Caffeine citrate is a low-dose caffeine product that has been shown to increase locomotor activity in rats. Caffeine citrate is an ester of caffeine and citric acid. It inhibits the enzyme that breaks down acetylcholine, which may lead to an increase in brain functions. Caffeine citrate is used as a treatment for apnea in pediatric patients, and it has also been shown to prevent bacterial translocation and reduce liver impairment caused by certain drugs. The therapeutic effect of caffeine citrate may be due to its ability to inhibit mitochondrial membrane potential, or its effects on basic proteins such as sodium citrate, or both.

Fórmula: C₈H₁₀N₄O₂·C₆H₈O₇

Forma y color: White Powder

Peso molecular: 386.31 g/mol

Ref: 3D-FC35311

Caffeine Citrate

CAS: 69-22-7

Applications Caffeine citrate (Cafcit) is a citrate salt of Caffeine, sometimes used in medical treatment, including short-term treatment of apnea of prematurity (lack of breathing in premature infants). Caffeine citrate functions in much the same capacity as does caffeine, but takes effect more quickly; its speed of dissociation is faster than that of Caffeine. Caffeine citrate is typically only used to treat severe migraines.
References Zubair, U.M., et al.: Anal. Profiles Drug Subs., 15, 71 (1986); Cherrah, Y., et al.: Biochem. Pharmacol., 37, 1311 (1988); Grillon, C., et al.: Clin. Neurophysiol., 114, 1557 (2003); Duangdao, D., et al.: Behav. Brain Res., 205, 1 (2009);

Fórmula: C₈H₁₀N₄O₂·C₆H₈O₇

Forma y color: White

Peso molecular: 386.31

Ref: TR-C080115

Caffeine Citrate

CAS: 69-22-7

Forma y color: Neat

Ref: 61-FOR1851.00