CAS 75696-02-5

Cinolazepam

Descripción:

Cinolazepam es un derivado de benzodiazepina utilizado principalmente por sus propiedades ansiolíticas, sedantes y relajantes musculares. Se caracteriza por su capacidad para potenciar los efectos del neurotransmisor ácido gamma-aminobutírico (GABA) en el receptor GABA-A, lo que lleva a una mayor inhibición neuronal. Este mecanismo contribuye a sus efectos terapéuticos en el tratamiento de trastornos de ansiedad y alteraciones del sueño. Cinolazepam se administra típicamente por vía oral y tiene una vida media relativamente larga, lo que puede resultar en efectos prolongados. La sustancia es conocida por su bajo potencial de abuso en comparación con otras benzodiazepinas, aunque se aconseja precaución debido al riesgo de dependencia con el uso prolongado. Los efectos secundarios comunes pueden incluir somnolencia, mareos y deterioro cognitivo. Al igual que con otros medicamentos de su clase, es esencial usar Cinolazepam bajo supervisión médica para mitigar riesgos y asegurar una dosificación adecuada. Su estructura química incluye un anillo de diazepina, que es característico de las benzodiazepinas, contribuyendo a su perfil farmacológico.

Fórmula: C₁₈H₁₃ClFN₃O₂

InChI: InChI=1S/C18H13ClFN3O2/c19-11-6-7-15-13(10-11)16(12-4-1-2-5-14(12)20)22-17(24)18(25)23(15)9-3-8-21/h1-2,4-7,10,17,24H,3,9H2

Clave InChI: InChIKey=XAXMYHMKTCNRRZ-UHFFFAOYSA-N

SMILES: C(CC#N)N1C=2C(C(=NC(O)C1=O)C3=C(F)C=CC=C3)=CC(Cl)=CC2

Sinónimos:

• 1H-1,4-Benzodiazepine-1-propanenitrile, 2,3-dihydro-7-chloro-5-(2-fluorophenyl)-2-oxo-
• 1H-1,4-Benzodiazepine-1-propanenitrile, 7-chloro-5-(2-fluorophenyl)-2,3-dihydro-3-hydroxy-2-oxo-
• 3-[7-chloro-5-(2-fluorophenyl)-3-hydroxy-2-oxo-2,3-dihydro-1H-1,4-benzodiazepin-1-yl]propanenitrile
• 7-Chloro-5-(2-fluorophenyl)-2,3-dihydro-3-hydroxy-2-oxo-1H-1,4-benzodiazepine-1-propanenitrile
• 7-Chloro-5-(o-fluorophenyl)-2,3-dihydro-3-hydroxy-2-oxo-1H-1,4-benzodiazepine-1-propionitrile
• Brn 5359831
• Cinolazepam [INN]
• Cinolazepamum
• Cinolazepamum [INN-Latin]
• Gerodorm
• Ox 373
• Unii-68P0556B0U

Cinolazepam

Producto controlado

CAS: 75696-02-5

Fórmula: C₁₈H₁₃ClFN₃O₂

Forma y color: Neat

Peso molecular: 357.766

Ref: TR-C475805

Cinolazepam

CAS: 75696-02-5

Cinolazepam is a benzodiazepine derivative drug.It has a powerful sedative effect, so it is mainly used as a hypnotic.

Fórmula: C₁₈H₁₃ClFN₃O₂

Forma y color: Solid

Peso molecular: 357.77

Ref: TM-T30945

Cinolazepam

Producto controlado

CAS: 75696-02-5

Cinolazepam is a benzodiazepine derivative, which is a synthetic product that acts primarily as a central nervous system depressant. Its mode of action involves enhancing the effect of the neurotransmitter gamma-aminobutyric acid (GABA) at the GABA-A receptor, resulting in increased inhibitory effects and neuronal hyperpolarization. This leads to its characteristic sedative and anxiolytic properties.Cinolazepam is utilized in therapeutic settings primarily as a hypnotic for the management of insomnia, particularly in cases involving difficulty in sleep initiation. It may also offer anxiolytic benefits, although it is less commonly prescribed for generalized anxiety disorders compared to other benzodiazepines. Its pharmacokinetic profile includes a relatively short half-life, favoring its use as a sleep aid with reduced risk of next-day residual effects. However, caution is warranted due to the potential for tolerance, dependence, and withdrawal phenomena typical of benzodiazepines. Therefore, its use is recommended for short-term treatment periods under strict medical supervision.

Fórmula: C₁₈H₁₃ClFN₃O₂

Pureza: Min. 95%

Peso molecular: 357.8 g/mol

Ref: 3D-ADA69602